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Found 46 with Last Name = 'oza' and Initial = 'sl'
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117542(2-Amino-4-[1-(hydroxycarbamoylmethyl-carbamoyl)-3-...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibitory constant against amidase free Glutathionylspermidine Synthetase mutant (C79A)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118638(2-[(S)-2-((S)-4-Amino-4-carboxy-butyrylamino)-4-me...)
Affinity DataKi:  6.40E+3nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118638(2-[(S)-2-((S)-4-Amino-4-carboxy-butyrylamino)-4-me...)
Affinity DataKi:  6.40E+3nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118640((S)-2-Amino-4-[1-((S)-(S)-2-amino-1-carboxy-ethylc...)
Affinity DataKi:  7.20E+3nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118640((S)-2-Amino-4-[1-((S)-(S)-2-amino-1-carboxy-ethylc...)
Affinity DataKi:  7.20E+3nMAssay Description:In vitro binding affinity for Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118642(5-Amino-2-[(S)-2-((S)-4-amino-4-carboxy-butyrylami...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118642(5-Amino-2-[(S)-2-((S)-4-amino-4-carboxy-butyrylami...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118643((S)-2-Amino-4-[1-((S)-(S)-3-amino-1-carboxy-propyl...)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118643((S)-2-Amino-4-[1-((S)-(S)-3-amino-1-carboxy-propyl...)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118644((S)-2-Amino-4-[1-((S)-(S)-1-carboxy-2-hydroxy-ethy...)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118644((S)-2-Amino-4-[1-((S)-(S)-1-carboxy-2-hydroxy-ethy...)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118641(6-Amino-2-[(S)-2-((S)-4-amino-4-carboxy-butyrylami...)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118641(6-Amino-2-[(S)-2-((S)-4-amino-4-carboxy-butyrylami...)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118639(6-(4-Amino-butylamino)-2-[(S)-2-((S)-4-amino-4-car...)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118639(6-(4-Amino-butylamino)-2-[(S)-2-((S)-4-amino-4-car...)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118645(2-[(S)-2-((S)-4-Amino-4-carboxy-butyrylamino)-4-me...)
Affinity DataKi:  3.30E+4nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118645(2-[(S)-2-((S)-4-Amino-4-carboxy-butyrylamino)-4-me...)
Affinity DataKi:  3.30E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117547(2-Amino-4-[3-methyl-1-(phosphonomethyl-carbamoyl)-...)
Affinity DataKi:  6.00E+4nMAssay Description:Inhibition constant of the compound was evaluated against enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117544(2-amino-4-(1-dihydroxyboronylmethylcarbamoyl-3-met...)
Affinity DataKi:  8.10E+4nMAssay Description:Inhibition constant of the compound was evaluated against enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117544(2-amino-4-(1-dihydroxyboronylmethylcarbamoyl-3-met...)
Affinity DataKi:  8.10E+4nMAssay Description:Concentration of the compound required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione synthetase(Trypanosoma cruzi)
University of Dundee

LigandPNGBDBM92592(DDD85811)
Affinity DataIC50:  95nMpH: 8.0 T: 2°CAssay Description:Hit compounds identified from the high throughput screen were also tested using orthogonal assay platform, namely the coupled assay described previou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypanothione synthetase(Trypanosoma cruzi)
University of Dundee

LigandPNGBDBM92593(DDD86243)
Affinity DataIC50:  140nMpH: 8.0 T: 2°CAssay Description:Hit compounds identified from the high throughput screen were also tested using orthogonal assay platform, namely the coupled assay described previou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypanothione synthetase(Trypanosoma cruzi)
University of Dundee

LigandPNGBDBM92590(DDD60632)
Affinity DataIC50:  273nMpH: 8.0 T: 2°CAssay Description:Hit compounds identified from the high throughput screen were also tested using orthogonal assay platform, namely the coupled assay described previou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypanothione synthetase(Trypanosoma cruzi)
University of Dundee

LigandPNGBDBM92591(DDD73385)
Affinity DataIC50:  317nMpH: 8.0 T: 2°CAssay Description:Hit compounds identified from the high throughput screen were also tested using orthogonal assay platform, namely the coupled assay described previou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117546(2-Amino-4-[1-(carbamoylmethyl-carbamoyl)-3-methyl-...)
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibitory activity against amidase free Glutathionylspermidine Synthetase mutant (C79A)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117543(2-Amino-4-{3-methyl-1-[2-oxo-2-(toluene-4-sulfonyl...)
Affinity DataIC50:  2.00E+3nMAssay Description:Concentration of the compound required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117542(2-Amino-4-[1-(hydroxycarbamoylmethyl-carbamoyl)-3-...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory activity against amidase free Glutathionylspermidine Synthetase mutant (C79A)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118640((S)-2-Amino-4-[1-((S)-(S)-2-amino-1-carboxy-ethylc...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118638(2-[(S)-2-((S)-4-Amino-4-carboxy-butyrylamino)-4-me...)
Affinity DataIC50:  9.40E+3nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118642(5-Amino-2-[(S)-2-((S)-4-amino-4-carboxy-butyrylami...)
Affinity DataIC50:  1.03E+4nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118644((S)-2-Amino-4-[1-((S)-(S)-1-carboxy-2-hydroxy-ethy...)
Affinity DataIC50:  1.17E+4nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118643((S)-2-Amino-4-[1-((S)-(S)-3-amino-1-carboxy-propyl...)
Affinity DataIC50:  1.37E+4nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117544(2-amino-4-(1-dihydroxyboronylmethylcarbamoyl-3-met...)
Affinity DataIC50:  1.72E+4nMAssay Description:Concentration of the compound required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118641(6-Amino-2-[(S)-2-((S)-4-amino-4-carboxy-butyrylami...)
Affinity DataIC50:  1.80E+4nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118645(2-[(S)-2-((S)-4-Amino-4-carboxy-butyrylamino)-4-me...)
Affinity DataIC50:  2.30E+4nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118639(6-(4-Amino-butylamino)-2-[(S)-2-((S)-4-amino-4-car...)
Affinity DataIC50:  2.79E+4nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117547(2-Amino-4-[3-methyl-1-(phosphonomethyl-carbamoyl)-...)
Affinity DataIC50:  6.00E+4nMAssay Description:Concentration required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118652((S)-2-Amino-4-[1-((S)-(S)-1-carboxy-ethylcarbamoyl...)
Affinity DataIC50:  9.00E+4nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117546(2-Amino-4-[1-(carbamoylmethyl-carbamoyl)-3-methyl-...)
Affinity DataIC50:  1.05E+5nMAssay Description:Inhibitory constant against amidase free Glutathionylspermidine Synthetase mutant (C79A)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117545(2-Amino-4-{3-methyl-1-[(1H-tetrazol-5-ylmethyl)-ca...)
Affinity DataIC50:  1.38E+5nMAssay Description:Concentration of the compound required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118649((S)-2-Amino-4-[1-((S)-(S)-2-carbamoyl-1-carboxy-et...)
Affinity DataIC50:  1.42E+5nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118647(2-[(S)-2-((S)-4-Amino-4-carboxy-butyrylamino)-4-me...)
Affinity DataIC50:  1.45E+5nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118648(2-[(S)-2-((S)-4-Amino-4-carboxy-butyrylamino)-4-me...)
Affinity DataIC50:  1.56E+5nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118651((S)-6-(3-tert-Butoxycarbonylamino-propylamino)-2-[...)
Affinity DataIC50:  1.57E+5nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118650(2-[(S)-2-((S)-4-Amino-4-carboxy-butyrylamino)-4-me...)
Affinity DataIC50:  2.27E+5nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118646(2-[(S)-2-((S)-4-Amino-4-carboxy-butyrylamino)-4-me...)
Affinity DataIC50:  3.65E+5nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed