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Found 127 with Last Name = 'ozawa' and Initial = 'h'
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064330(CHEMBL3403710)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064331(CHEMBL3403711)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064332(CHEMBL3403712)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064356(CHEMBL3403708)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at Gal4-tagged LXRalpha (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064377(CHEMBL3403693)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at Gal4-tagged LXRalpha (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064378(CHEMBL3403692)
Affinity DataEC50:  1.10E+4nMAssay Description:Agonist activity at Gal4-tagged LXRalpha (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064379(CHEMBL3403691)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at Gal4-tagged LXRalpha (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064380(CHEMBL3403687)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity at Gal4-tagged LXRalpha (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064381(CHEMBL3403686)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity at Gal4-tagged LXRalpha (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM19992(2-[3-[3-[[2-chloro-3-(trifluoromethyl)phenyl]methy...)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at Gal4-tagged LXRalpha (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM19992(2-[3-[3-[[2-chloro-3-(trifluoromethyl)phenyl]methy...)
Affinity DataEC50:  420nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064381(CHEMBL3403686)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064380(CHEMBL3403687)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064382(CHEMBL3403688)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064383(CHEMBL3403689)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064379(CHEMBL3403691)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064378(CHEMBL3403692)
Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064377(CHEMBL3403693)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064384(CHEMBL3403695)
Affinity DataEC50:  5.30E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064385(CHEMBL3403696)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064386(CHEMBL3403699)
Affinity DataEC50:  960nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064387(CHEMBL3403701)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064388(CHEMBL3403704)
Affinity DataEC50:  8.00E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064389(CHEMBL3403707)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064356(CHEMBL3403708)
Affinity DataEC50:  1.02E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064390(CHEMBL3403709)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...)
Affinity DataEC50:  490nMAssay Description:Agonist activity at Gal4-tagged LXRalpha (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...)
Affinity DataEC50:  410nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064391(CHEMBL3403715)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at Gal4-tagged LXRalpha (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064391(CHEMBL3403715)
Affinity DataEC50:  690nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214884(2-(3-(((6-fluorobenzo[d]oxazol-2-yl)(3-phenoxyprop...)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human recombinant PPARgamma by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214885(2-(3-((benzo[d]oxazol-2-yl(2-phenoxyethyl)amino)me...)
Affinity DataEC50:  630nMAssay Description:Agonist activity at human recombinant PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214887(2-(3-((benzo[d]oxazol-2-yl(3-(4-fluorophenoxy)prop...)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human recombinant PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214886(2-(3-(((5-methylbenzo[d]oxazol-2-yl)(3-phenoxyprop...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human recombinant PPARgamma by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214888(2-(3-(((4-hydroxybenzo[d]oxazol-2-yl)(3-phenoxypro...)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at human recombinant PPARgamma by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214889(2-(3-(2-(benzo[d]oxazol-2-yl(3-phenoxypropyl)amino...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human recombinant PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214892(2-(3-((benzo[d]oxazol-2-yl(3-(2,4-difluorophenoxy)...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human recombinant PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214890((R)-2-(3-((benzo[d]oxazol-2-yl(3-(4-fluorophenoxy)...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human recombinant PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214893(2-(3-((benzo[d]oxazol-2-yl(3-(p-tolyloxy)propyl)am...)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human recombinant PPARgamma by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214891(2-(3-((benzo[d]oxazol-2-yl(3-(3,4-dimethylphenoxy)...)
Affinity DataEC50:  830nMAssay Description:Agonist activity at human recombinant PPARdelta by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214894(2-(3-((benzo[d]oxazol-2-yl(3-phenoxypropyl)amino)m...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human recombinant PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214896((S)-2-(3-((benzo[d]oxazol-2-yl(3-phenoxypropyl)ami...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human recombinant PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214895(2-(3-((benzo[d]oxazol-2-yl(3-phenoxypropyl)amino)m...)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at human recombinant PPARdelta by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214892(2-(3-((benzo[d]oxazol-2-yl(3-(2,4-difluorophenoxy)...)
Affinity DataEC50:  6.50E+3nMAssay Description:Agonist activity at human recombinant PPARdelta by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214897(2-(3-{[[1,3]dioxolo[4',5':4,5]benzo[1,2-d]oxazol-6...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human recombinant PPARgamma by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214889(2-(3-(2-(benzo[d]oxazol-2-yl(3-phenoxypropyl)amino...)
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at human recombinant PPARdelta by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214897(2-(3-{[[1,3]dioxolo[4',5':4,5]benzo[1,2-d]oxazol-6...)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human recombinant PPARdelta by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214898((S)-2-(3-((benzo[d]oxazol-2-yl(3-(4-methoxyphenoxy...)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at human recombinant PPARdelta by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214900(2-(3-(2-(benzo[d]oxazol-2-yl(2-phenoxyethyl)amino)...)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human recombinant PPARgamma by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50214899((R)-2-(3-((benzo[d]oxazol-2-yl(3-(4-methoxyphenoxy...)
Affinity DataEC50:  1.58E+3nMAssay Description:Agonist activity at human recombinant PPARdelta by GAL4 transactivation assayMore data for this Ligand-Target Pair
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