TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataKi: 690nMAssay Description:Competitive inhibition of recombinant HePTP expressed in Escherichia coli by Michaelis-Menten kinetic analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
University of California San Diego
Curated by ChEMBL
University of California San Diego
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Binding affinity at 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in rat brain.More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Brown University
Curated by ChEMBL
Brown University
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
TargetMetallo-beta-lactamase type 2(Serratia marcescens)
University of California San Diego
Curated by ChEMBL
University of California San Diego
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of Serratia marcescens IMP1 expressed in Escherichia coli BL21(DE3) using chromacef as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Brown University
Curated by ChEMBL
Brown University
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
Affinity DataIC50: 910nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant HePTP expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Brown University
Curated by ChEMBL
Brown University
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant HePTP expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Brown University
Curated by ChEMBL
Brown University
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
TargetMetallo-beta-lactamase VIM-2(Pseudomonas aeruginosa (g-Proteobacteria))
University of California San Diego
Curated by ChEMBL
University of California San Diego
Curated by ChEMBL
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa VIM2 expressed in Escherichia coli BL21(DE3) using chromacef as substrate preincubated for 10 mins followed by s...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of recombinant HePTP expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
Brown University
Curated by ChEMBL
Brown University
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
TargetMetallo-beta-lactamase type 2(Serratia marcescens)
University of California San Diego
Curated by ChEMBL
University of California San Diego
Curated by ChEMBL
Affinity DataIC50: 3.03E+3nMAssay Description:Binding affinity at 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in rat brain.More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
Brown University
Curated by ChEMBL
Brown University
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of recombinant HePTP expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
Brown University
Curated by ChEMBL
Brown University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of recombinant VHR expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of recombinant HePTP expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
Brown University
Curated by ChEMBL
Brown University
Curated by ChEMBL
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of recombinant VHR expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of recombinant VHR expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of recombinant VHR expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibition of recombinant VHR expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of HePTPMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of HePTPMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 6(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of recombinant MKP3 expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 6(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of recombinant MKP3 expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 6(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of recombinant MKP3 expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 6(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant MKP3 expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 6(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant MKP3 expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 6(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant MKP3 expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant HePTP expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Sanford-Burnham Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant VHR expressed in Escherichia coliMore data for this Ligand-Target Pair