Affinity DataIC50: 0.5nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in CHOK1 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.70nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 11.6nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 12.3nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 12.7nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 13.1nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 13.2nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 16.3nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in CHOK1 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 19.5nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Korea Research Institute Of Bioscience And Biotechnology
Curated by ChEMBL
Korea Research Institute Of Bioscience And Biotechnology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against rat liver microsomal Acyl coenzyme A:cholesterol acyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in CHOK1 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 29.1nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 34.6nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 35.3nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 35.9nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 38.8nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in CHOK1 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in CHOK1 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in CHOK1 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 45.7nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 49.6nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 50.7nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in CHOK1 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 59.9nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5HT2A receptor expressed in avCHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 66.5nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair