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Found 398 with Last Name = 'paul' and Initial = 'b'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306528((6aR,10aR)-6,6,9-trimethyl-3-(2-methyloctan-2-yl)-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306528((6aR,10aR)-6,6,9-trimethyl-3-(2-methyloctan-2-yl)-...)
Affinity DataKi:  0.240nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]-U69593 from kappa opioid receptor (unknown origin) assessed as inhibition constant incubated for 180 mins by competitive radioli...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) assessed as inhibition constant incubated for 180 mins by competitive radioligand ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306530((6aR,10aR)-6,6,9-trimethyl-3-(2-methyloctan-2-yl)-...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of human cloned CA12 catalytic domain by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Affinity DataKi:  5nMAssay Description:Inhibition of human cloned CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM10888(1,2-benzoxazol-3-ylmethanesulfonamide | CHEMBL750 ...)
Affinity DataKi:  5nMAssay Description:Inhibition of human cloned CA9 catalytic domain by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306529((6aR,10aR)-6,6,9-trimethyl-3-(2-methyloctan-2-yl)-...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human cloned CA12 catalytic domain by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306530((6aR,10aR)-6,6,9-trimethyl-3-(2-methyloctan-2-yl)-...)
Affinity DataKi:  11.7nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Inhibition of human cloned CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613007(CHEMBL5290432)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) assessed as inhibition constant incubated for 180 mins by competitive radioligand ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  25nMAssay Description:Inhibition of human cloned CA9 catalytic domain by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM10888(1,2-benzoxazol-3-ylmethanesulfonamide | CHEMBL750 ...)
Affinity DataKi:  35nMAssay Description:Inhibition of human cloned CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613008(CHEMBL5288483)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]-U69593 from kappa opioid receptor (unknown origin) assessed as inhibition constant incubated for 180 mins by competitive radioli...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613008(CHEMBL5288483)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) assessed as inhibition constant incubated for 180 mins by competitive radioligand ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM10888(1,2-benzoxazol-3-ylmethanesulfonamide | CHEMBL750 ...)
Affinity DataKi:  56nMAssay Description:Inhibition of human cloned CA1 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCarbonic anhydrase 9(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Affinity DataKi:  58nMAssay Description:Inhibition of human cloned CA9 catalytic domain by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306529((6aR,10aR)-6,6,9-trimethyl-3-(2-methyloctan-2-yl)-...)
Affinity DataKi:  67.8nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613009(CHEMBL5280172)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) assessed as inhibition constant incubated for 180 mins by competitive radioligand ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613011(CHEMBL5291340)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) assessed as inhibition constant incubated for 180 mins by competitive radioligand ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306542((6aR,10aR)-6,6,9-trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  215nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306531(CHEMBL600195 | N-((6aR,10aR)-6,6,9-trimethyl-3-(2-...)
Affinity DataKi:  216nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613010(CHEMBL5276128)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) assessed as inhibition constant incubated for 180 mins by competitive radioligand ...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM10887(Sulfamate 7 | Topiramate (TPM) | US11535599, Examp...)
Affinity DataKi:  250nMAssay Description:Inhibition of human cloned CA1 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  250nMAssay Description:Inhibition of human cloned CA1 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306534(CHEMBL601865 | N-((6aR,10aR)-6,6,9-trimethyl-3-(2-...)
Affinity DataKi:  255nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306532(1-methyl-3-(6aR,10aR)-6,6,9-trimethyl-3-(2-methylo...)
Affinity DataKi:  257nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50568638(CHEMBL4871880)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) assessed as inhibition constant incubated for 180 mins by competitive radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50568639(CHEMBL4846243)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) assessed as inhibition constant incubated for 180 mins by competitive radioligand ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613011(CHEMBL5291340)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]-U69593 from kappa opioid receptor (unknown origin) assessed as inhibition constant incubated for 180 mins by competitive radioli...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306532(1-methyl-3-(6aR,10aR)-6,6,9-trimethyl-3-(2-methylo...)
Affinity DataKi:  333nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306543((6aR,10aR)-6,6,9-trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  387nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306526((6aR,10aR)-6,6,9-trimethyl-1-(methylthio)-3-pentyl...)
Affinity DataKi:  469nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613007(CHEMBL5290432)
Affinity DataKi:  580nMAssay Description:Displacement of [3H]-U69593 from kappa opioid receptor (unknown origin) assessed as inhibition constant incubated for 180 mins by competitive radioli...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613010(CHEMBL5276128)
Affinity DataKi:  580nMAssay Description:Displacement of [3H]-U69593 from kappa opioid receptor (unknown origin) assessed as inhibition constant incubated for 180 mins by competitive radioli...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306542((6aR,10aR)-6,6,9-trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  616nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306524(1-(((6aR,10aR)-6,6,9-trimethyl-3-pentyl-6a,7,8,10a...)
Affinity DataKi:  782nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306526((6aR,10aR)-6,6,9-trimethyl-1-(methylthio)-3-pentyl...)
Affinity DataKi:  955nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306533(CHEMBL600397 | N-((6aR,10aR)-6,6,9-trimethyl-3-(2-...)
Affinity DataKi:  1.09E+3nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50613009(CHEMBL5280172)
Affinity DataKi:  1.17E+3nMAssay Description:Displacement of [3H]-U69593 from kappa opioid receptor (unknown origin) assessed as inhibition constant incubated for 180 mins by competitive radioli...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306539((6aR,10aR)-N,N,6,6,9-pentamethyl-3-pentyl-6a,7,8,1...)
Affinity DataKi:  1.21E+3nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306538((6aR,10aR)-N,6,6,9-tetramethyl-3-pentyl-6a,7,8,10a...)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306531(CHEMBL600195 | N-((6aR,10aR)-6,6,9-trimethyl-3-(2-...)
Affinity DataKi:  1.34E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306544(CHEMBL605128 | methyl(6aR,10aR)-6,6,9-trimethyl-3-...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306535(CHEMBL602857 | N-((6aR,10aR)-6,6,9-trimethyl-3-pen...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50306525(CHEMBL604329 | N-(((6aR,10aR)-6,6,9-trimethyl-3-pe...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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