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Found 25 with Last Name = 'peters' and Initial = 'gj'
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Universita` Di Pisa

Curated by ChEMBL
LigandPNGBDBM50339607(1-Hydroxy-6-phenyl-4-trifluoromethyl-1H-indole-2-c...)
Affinity DataKi:  4.70E+3nMAssay Description:Competitive inhibition of human LDH-A using pyruvate as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Universita` Di Pisa

Curated by ChEMBL
LigandPNGBDBM50066974(7-Benzyl-2,3-dihydroxy-6-methyl-4-propyl-naphthale...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of human LDH-A using pyruvate as substrate and NADH as cofactor at 125 uM after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Universita` Di Pisa

Curated by ChEMBL
LigandPNGBDBM50339607(1-Hydroxy-6-phenyl-4-trifluoromethyl-1H-indole-2-c...)
Affinity DataKi:  8.90E+3nMAssay Description:Competitive inhibition of human LDH-A using NADH as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Universita` Di Pisa

Curated by ChEMBL
LigandPNGBDBM50339605(1-Hydroxy-5-phenyl-1H-indole-2-carboxylic Acid | C...)
Affinity DataKi:  1.04E+4nMAssay Description:Competitive inhibition of human LDH-A using NADH as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Universita` Di Pisa

Curated by ChEMBL
LigandPNGBDBM50339605(1-Hydroxy-5-phenyl-1H-indole-2-carboxylic Acid | C...)
Affinity DataKi:  1.57E+4nMAssay Description:Competitive inhibition of human LDH-A using pyruvate as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Universita` Di Pisa

Curated by ChEMBL
LigandPNGBDBM50339606(1-Hydroxy-6-phenyl-1H-indole-2-carboxylic Acid | C...)
Affinity DataKi:  1.98E+4nMAssay Description:Competitive inhibition of human LDH-A using NADH as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Universita` Di Pisa

Curated by ChEMBL
LigandPNGBDBM50339606(1-Hydroxy-6-phenyl-1H-indole-2-carboxylic Acid | C...)
Affinity DataKi:  3.54E+4nMAssay Description:Competitive inhibition of human LDH-A using pyruvate as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Universita` Di Pisa

Curated by ChEMBL
LigandPNGBDBM23222(Oxalamic acid | Oxamate | Oxamate, 3 | Oxamidic Ac...)
Affinity DataKi:  1.38E+5nMAssay Description:Inhibition of human LDH-A using pyruvate as substrate and NADH as cofactor at 125 uM after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278034(CHEMBL4169791)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of PH domain lacking AKT1 (unknown origin) using Tamara-labeled GRPRTSSFAEG peptide as substrate after 90 mins by fluorescence polarizatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278056(CHEMBL4163627)
Affinity DataIC50:  4.70nMAssay Description:Antagonistic affinity against Alpha-1A adrenergic receptor was determined in isolated prostatic vas deferens tissue from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278048(CHEMBL4160193)
Affinity DataIC50:  8.20nMAssay Description:Antagonistic affinity against Alpha-1B adrenergic receptor was determined in isolated spleen tissue from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278044(CHEMBL4173126)
Affinity DataIC50:  12nMAssay Description:Antagonistic affinity against Alpha-1D adrenergic receptor was determined in isolated thoracic aorta from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278019(CHEMBL4172716)
Affinity DataIC50:  56nMAssay Description:Inhibition of PH domain lacking AKT1 (unknown origin) using Tamara-labeled GRPRTSSFAEG peptide as substrate after 90 mins by fluorescence polarizatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278035(CHEMBL4171390)
Affinity DataIC50:  115nMAssay Description:Inhibition of PH domain lacking AKT1 (unknown origin) using Tamara-labeled GRPRTSSFAEG peptide as substrate after 90 mins by fluorescence polarizatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278033(CHEMBL4159491)
Affinity DataIC50:  176nMAssay Description:Inhibition of PH domain lacking AKT1 (unknown origin) using Tamara-labeled GRPRTSSFAEG peptide as substrate after 90 mins by fluorescence polarizatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278031(CHEMBL4163164)
Affinity DataIC50:  251nMAssay Description:Antagonistic potency for NK-3 receptor was determined in vitro, using isolated rat portal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278047(CHEMBL4160580)
Affinity DataIC50:  311nMAssay Description:Antagonistic affinity against Alpha-1A adrenergic receptor was determined in isolated prostatic vas deferens tissue from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278032(CHEMBL4169321)
Affinity DataIC50:  313nMAssay Description:Antagonistic potency for NK-1 receptor was determined in vitro,using isolated rabbit vena cava.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278057(CHEMBL4164809)
Affinity DataIC50:  432nMAssay Description:Antagonistic affinity against Alpha-1A adrenergic receptor was determined in isolated prostatic vas deferens tissue from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278046(CHEMBL4170874)
Affinity DataIC50:  482nMAssay Description:Antagonistic affinity against Alpha-1B adrenergic receptor was determined in isolated spleen tissue from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278045(CHEMBL4161394)
Affinity DataIC50:  640nMAssay Description:Antagonistic affinity against Alpha-1A adrenergic receptor was determined in isolated prostatic vas deferens tissue from ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278030(CHEMBL4176130)
Affinity DataIC50:  738nMAssay Description:Antagonistic potency for NK-3 receptor was determined in vitro, using isolated rat portal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50278043(CHEMBL4161273)
Affinity DataIC50:  980nMAssay Description:Compound was evaluated for in vitro inhibition of human immunodeficiency virus type 1 (HIV-1) ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Universita` Di Pisa

Curated by ChEMBL
LigandPNGBDBM23251(1,2,5-Thiadiazole, TDA1 | 4-hydroxy-1,2,5-thiadiaz...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human LDH-A using pyruvate as substrate and NADH as cofactor at 125 uM after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Universita` Di Pisa

Curated by ChEMBL
LigandPNGBDBM23242(1,2(1,5)-Isoxazole, IOA1 | 3-hydroxy-1,2-oxazole-4...)
Affinity DataIC50:  5.40E+4nMAssay Description:Inhibition of human LDH-A using pyruvate as substrate and NADH as cofactor at 125 uM after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed