Affinity DataKi: 4.70E+3nMAssay Description:Competitive inhibition of human LDH-A using pyruvate as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of human LDH-A using pyruvate as substrate and NADH as cofactor at 125 uM after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 8.90E+3nMAssay Description:Competitive inhibition of human LDH-A using NADH as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 1.04E+4nMAssay Description:Competitive inhibition of human LDH-A using NADH as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 1.57E+4nMAssay Description:Competitive inhibition of human LDH-A using pyruvate as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 1.98E+4nMAssay Description:Competitive inhibition of human LDH-A using NADH as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 3.54E+4nMAssay Description:Competitive inhibition of human LDH-A using pyruvate as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 1.38E+5nMAssay Description:Inhibition of human LDH-A using pyruvate as substrate and NADH as cofactor at 125 uM after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of PH domain lacking AKT1 (unknown origin) using Tamara-labeled GRPRTSSFAEG peptide as substrate after 90 mins by fluorescence polarizatio...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 4.70nMAssay Description:Antagonistic affinity against Alpha-1A adrenergic receptor was determined in isolated prostatic vas deferens tissue from ratMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 8.20nMAssay Description:Antagonistic affinity against Alpha-1B adrenergic receptor was determined in isolated spleen tissue from ratMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Antagonistic affinity against Alpha-1D adrenergic receptor was determined in isolated thoracic aorta from ratMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of PH domain lacking AKT1 (unknown origin) using Tamara-labeled GRPRTSSFAEG peptide as substrate after 90 mins by fluorescence polarizatio...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 115nMAssay Description:Inhibition of PH domain lacking AKT1 (unknown origin) using Tamara-labeled GRPRTSSFAEG peptide as substrate after 90 mins by fluorescence polarizatio...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 176nMAssay Description:Inhibition of PH domain lacking AKT1 (unknown origin) using Tamara-labeled GRPRTSSFAEG peptide as substrate after 90 mins by fluorescence polarizatio...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Antagonistic potency for NK-3 receptor was determined in vitro, using isolated rat portal vein.More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 311nMAssay Description:Antagonistic affinity against Alpha-1A adrenergic receptor was determined in isolated prostatic vas deferens tissue from ratMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 313nMAssay Description:Antagonistic potency for NK-1 receptor was determined in vitro,using isolated rabbit vena cava.More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 432nMAssay Description:Antagonistic affinity against Alpha-1A adrenergic receptor was determined in isolated prostatic vas deferens tissue from ratMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 482nMAssay Description:Antagonistic affinity against Alpha-1B adrenergic receptor was determined in isolated spleen tissue from ratMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:Antagonistic affinity against Alpha-1A adrenergic receptor was determined in isolated prostatic vas deferens tissue from ratMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 738nMAssay Description:Antagonistic potency for NK-3 receptor was determined in vitro, using isolated rat portal vein.More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Svkm'S Dr. Bhanuben Nanavati College Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 980nMAssay Description:Compound was evaluated for in vitro inhibition of human immunodeficiency virus type 1 (HIV-1) ProteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human LDH-A using pyruvate as substrate and NADH as cofactor at 125 uM after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of human LDH-A using pyruvate as substrate and NADH as cofactor at 125 uM after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair