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Found 46 with Last Name = 'phuwapraisirisan' and Initial = 'p'
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439692(CHEMBL2418233)
Affinity DataKi:  2.24E+4nMAssay Description:Competitive inhibition of rat intestine sucrase using sucrose as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439692(CHEMBL2418233)
Affinity DataKi:  2.38E+4nMAssay Description:Competitive inhibition of rat intestine maltase using maltose as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439692(CHEMBL2418233)
Affinity DataKi:  4.75E+4nMAssay Description:Non-competitive inhibition of rat intestine sucrase using sucrose as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439692(CHEMBL2418233)
Affinity DataKi:  6.45E+4nMAssay Description:Non-competitive inhibition of rat intestine maltase using maltose as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50208826((+)-Pinoresinol | 4-[(1S,3aR,4S,6aR)-4-(4-hydroxy-...)
Affinity DataKi:  2.88E+5nMAssay Description:Competitive inhibition of rat intestinal maltase using maltose as substrate assessed as dissociation of enzyme-inhibitor complex at 0.1 to 1 mg/ml by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50123929(CHEMBL3621760)
Affinity DataKi:  3.80E+5nMAssay Description:Non-competitive inhibition of rat intestinal Sucrase using sucrose as substrate assessed as glucose release after 40 mins by Lineweaver-Burk plot ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50123930(CHEMBL3621759)
Affinity DataKi:  4.80E+5nMAssay Description:Non-competitive inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by Lineweaver-Burk plot ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50123929(CHEMBL3621760)
Affinity DataKi:  5.30E+5nMAssay Description:Non-competitive inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by Lineweaver-Burk plot ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50123930(CHEMBL3621759)
Affinity DataKi:  5.40E+5nMAssay Description:Non-competitive inhibition of rat intestinal Sucrase using sucrose as substrate assessed as glucose release after 40 mins by Lineweaver-Burk plot ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50123930(CHEMBL3621759)
Affinity DataKi:  1.09E+6nMAssay Description:Competitive inhibition of rat intestinal Sucrase using sucrose as substrate assessed as glucose release after 40 mins by Lineweaver-Burk plot analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50208826((+)-Pinoresinol | 4-[(1S,3aR,4S,6aR)-4-(4-hydroxy-...)
Affinity DataKi:  1.34E+6nMAssay Description:Non-competitive inhibition of rat intestinal maltase using maltose as substrate assessed as dissociation of enzyme-substrate-inhibitor complex at 0.1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50123930(CHEMBL3621759)
Affinity DataKi:  1.64E+6nMAssay Description:Competitive inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by Lineweaver-Burk plot analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50123929(CHEMBL3621760)
Affinity DataKi:  1.96E+6nMAssay Description:Competitive inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by Lineweaver-Burk plot analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50123929(CHEMBL3621760)
Affinity DataKi:  3.07E+6nMAssay Description:Competitive inhibition of rat intestinal Sucrase using sucrose as substrate assessed as glucose release after 40 mins by Lineweaver-Burk plot analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50333465((2R,3R,4R,5R,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50333465((2R,3R,4R,5R,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of rat intestinal alpha-glucosidase maltase using maltose as substrate preincubated for 10 mins prior substrate addition measured after 40...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50333465((2R,3R,4R,5R,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by glucose oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50333465((2R,3R,4R,5R,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50333465((2R,3R,4R,5R,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50:  2.38E+3nMAssay Description:Inhibition of rat intestinal alpha-glucosidase sucrase using sucrose as substrate preincubated for 10 mins prior substrate addition measured after 40...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50333465((2R,3R,4R,5R,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of rat intestinal sucrase using sucrose substrate incubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50036139(CHEMBL3358660)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of rat intestinal sucrase using sucrose substrate incubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50036147(CHEMBL3358661)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of rat intestinal sucrase using sucrose substrate incubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439692(CHEMBL2418233)
Affinity DataIC50:  5.31E+3nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50035933(CHEMBL3358659)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of rat intestinal sucrase using sucrose substrate incubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50035932(CHEMBL3358658)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of rat intestinal sucrase using sucrose substrate incubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439694(CHEMBL2418237)
Affinity DataIC50:  2.08E+4nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439695(CHEMBL2418236)
Affinity DataIC50:  2.11E+4nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50333465((2R,3R,4R,5R,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of rat intestinal Sucrase using sucrose as substrate assessed as glucose release after 40 mins by glucose oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50123929(CHEMBL3621760)
Affinity DataIC50:  3.39E+4nMAssay Description:Inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by glucose oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50208826((+)-Pinoresinol | 4-[(1S,3aR,4S,6aR)-4-(4-hydroxy-...)
Affinity DataIC50:  3.43E+4nMAssay Description:Inhibition of rat intestinal maltase using maltose as substrate preincubated for 10 mins before substrate addition by glucose oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM4375((2E)-3-(3,4-dihydroxyphenyl)prop-2-enoic acid | (2...)
Affinity DataIC50:  3.47E+4nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439692(CHEMBL2418233)
Affinity DataIC50:  4.37E+4nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50123930(CHEMBL3621759)
Affinity DataIC50:  4.72E+4nMAssay Description:Inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by glucose oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50123929(CHEMBL3621760)
Affinity DataIC50:  4.74E+4nMAssay Description:Inhibition of rat intestinal Sucrase using sucrose as substrate assessed as glucose release after 40 mins by glucose oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439696(CHEMBL2418235)
Affinity DataIC50:  5.19E+4nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439694(CHEMBL2418237)
Affinity DataIC50:  5.30E+4nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439696(CHEMBL2418235)
Affinity DataIC50:  6.72E+4nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM4375((2E)-3-(3,4-dihydroxyphenyl)prop-2-enoic acid | (2...)
Affinity DataIC50:  8.75E+4nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50123930(CHEMBL3621759)
Affinity DataIC50:  9.49E+4nMAssay Description:Inhibition of rat intestinal Sucrase using sucrose as substrate assessed as glucose release after 40 mins by glucose oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439695(CHEMBL2418236)
Affinity DataIC50:  1.71E+5nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439693(CHEMBL2418238)
Affinity DataIC50:  3.67E+5nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439697(CHEMBL2418234)
Affinity DataIC50:  4.97E+5nMAssay Description:Inhibition of rat intestine maltase using maltose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-galactosidase(Homo sapiens (Human))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50365006(CHEMBL1950779)
Affinity DataIC50:  6.00E+5nMAssay Description:Inhibition of beta-galactosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439693(CHEMBL2418238)
Affinity DataIC50:  8.05E+5nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50439697(CHEMBL2418234)
Affinity DataIC50:  9.54E+5nMAssay Description:Inhibition of rat intestine sucrase using sucrose as substrate incubated for 10 mins prior to substrate addition measured after 40 mins by glucose ox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Chulalongkorn University

Curated by ChEMBL
LigandPNGBDBM50123931(CHEMBL3621761)
Affinity DataIC50:  1.85E+6nMAssay Description:Inhibition of rat intestinal Maltase using maltose as substrate assessed as glucose release after 10 mins by glucose oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed