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Found 108 with Last Name = 'pieroni' and Initial = 'm'
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50387827(CHEMBL2058635)
Affinity DataKi:  0.178nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane incubated for 30 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50021809((2,6-Dichloro-4-iodo-phenyl)-(4,5-dihydro-1H-imida...)
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane incubated for 30 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50091345(CHEMBL2092861)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM81807(ATIPAMEZOLE | CAS_104054-27-5 | NSC_71310)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50240366(2-(naphthalen-2-yl)-4,5-dihydro-1H-imidazole | 2-N...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane incubated for 30 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50601014(CHEMBL5170947)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50085683((+)-4-((S)-alpha,2,3-trimethylbenzyl)imidazole | 4...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50179393(Efaroxan)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50019646(2-(alpha-(2,6-Dichlorophenoxy)ethyl)2-imidazoline ...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane incubated for 30 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50070328(CHEBI:8862 | Rilmenidine)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane incubated for 30 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50601018(CHEMBL5207596)
Affinity DataKi:  27nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50179397(CHEMBL1162356)
Affinity DataKi:  28nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane incubated for 30 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50146549(CHEMBL3764222)
Affinity DataKi:  40nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50146407(CHEMBL3763469)
Affinity DataKi:  50nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50146448(CHEMBL3764351)
Affinity DataKi:  80nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50146526(CHEMBL3765396)
Affinity DataKi:  86nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50601022(CHEMBL5181500)
Affinity DataKi:  110nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  126nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane incubated for 30 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50029050((-)-(R)-epinephrine | (-)-3,4-dihydroxy-alpha-((me...)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50601016(CHEMBL5204588)
Affinity DataKi:  240nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50070328(CHEBI:8862 | Rilmenidine)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50412260(CHEMBL273485)
Affinity DataKi:  309nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  347nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50601013(CHEMBL5179589)
Affinity DataKi:  400nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50179396(CHEMBL1907831)
Affinity DataKi:  589nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50146579(Benzyl-O-Hydroxylamine | CHEMBL443652 | O-Benzylhy...)
Affinity DataKi:  600nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50179395(CHEMBL14640)
Affinity DataKi:  708nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50601019(CHEMBL5199538)
Affinity DataKi:  720nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50179391(CHEMBL3593723)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50019848(2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1...)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50601021(CHEMBL5207995)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50146551(CHEMBL3763498)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50146408(CHEMBL3764504)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50601020(CHEMBL5183689)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50138499(2-Phenethyl-4,5-dihydro-1H-imidazole | CHEMBL14210)
Affinity DataKi:  3.72E+3nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50146529(CHEMBL3764023)
Affinity DataKi:  3.78E+3nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50146461(CHEMBL3765807)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50601023(CHEMBL5195123)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50091347(CHEMBL71429)
Affinity DataKi:  6.31E+3nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50179394(CHEMBL68608)
Affinity DataKi:  7.24E+3nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50179392(CHEMBL3593725)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlanine--glyoxylate aminotransferase(Homo sapiens)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50146465(CHEMBL3765186)
Affinity DataKi:  1.70E+4nMAssay Description:Inhibition of recombinant wild type His-tagged AGT (unknown origin) expressed in Escherichia coli BL21 assessed as inhibition constant using L-alanin...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50179387(CHEMBL3814276)
Affinity DataKi:  2.70E+4nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50179384(CHEMBL3814220)
Affinity DataKi:  4.10E+4nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50179386(CHEMBL3814626)
Affinity DataKi:  5.20E+4nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50179382(CHEMBL3814535)
Affinity DataKi:  5.80E+4nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50179383(CHEMBL3814593)
Affinity DataKi:  6.20E+4nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Belgrade

Curated by ChEMBL
LigandPNGBDBM50179385(CHEMBL3814521)
Affinity DataKi:  8.00E+4nMAssay Description:Displacement of [3H]RS-79948-197 from recombinant human alpha2A adrenoreceptor expressed in CHOK1 cell membrane by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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