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Found 28 with Last Name = 'porter' and Initial = 'v'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001590(CHEMBL3237722)
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]diprenorphine from rat mu opioid receptor expressed in rat C6 cell membranes after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001590(CHEMBL3237722)
Affinity DataKi:  0.930nMAssay Description:Displacement of [3H]diprenorphine from rat delta opioid receptor expressed in rat C6 cell membranes after 1 hr by liquid scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001608(CHEMBL3237723)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]diprenorphine from rat mu opioid receptor expressed in rat C6 cell membranes after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001588(CHEMBL3237720)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]diprenorphine from rat delta opioid receptor expressed in rat C6 cell membranes after 1 hr by liquid scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001588(CHEMBL3237720)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]diprenorphine from rat mu opioid receptor expressed in rat C6 cell membranes after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001608(CHEMBL3237723)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]diprenorphine from rat delta opioid receptor expressed in rat C6 cell membranes after 1 hr by liquid scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001589(CHEMBL3237721)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]diprenorphine from rat delta opioid receptor expressed in rat C6 cell membranes after 1 hr by liquid scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001589(CHEMBL3237721)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]diprenorphine from rat mu opioid receptor expressed in rat C6 cell membranes after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001590(CHEMBL3237722)
Affinity DataKi:  93nMAssay Description:Displacement of [3H]diprenorphine from human kappa opioid receptor expressed in CHO cell membranes after 1 hr by liquid scintillation counting analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001608(CHEMBL3237723)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]diprenorphine from human kappa opioid receptor expressed in CHO cell membranes after 1 hr by liquid scintillation counting analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001588(CHEMBL3237720)
Affinity DataKi:  776nMAssay Description:Displacement of [3H]diprenorphine from human kappa opioid receptor expressed in CHO cell membranes after 1 hr by liquid scintillation counting analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001589(CHEMBL3237721)
Affinity DataKi:  7.10E+3nMAssay Description:Displacement of [3H]diprenorphine from human kappa opioid receptor expressed in CHO cell membranes after 1 hr by liquid scintillation counting analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50359568(CHEMBL1927661)
Affinity DataIC50:  450nMAssay Description:Inhibition of human alpha-thrombin using sarcosine-Pro-Arg-p-nitroanilide as substrate preincubated for 5 mins before substrate addition measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50359569(CHEMBL1927660)
Affinity DataIC50:  510nMAssay Description:Inhibition of human alpha-thrombin using sarcosine-Pro-Arg-p-nitroanilide as substrate preincubated for 5 mins before substrate addition measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50359562(CHEMBL1927655)
Affinity DataIC50:  570nMAssay Description:Inhibition of human alpha-thrombin using sarcosine-Pro-Arg-p-nitroanilide as substrate preincubated for 5 mins before substrate addition measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50359559(CHEMBL1927658)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of human alpha-thrombin using sarcosine-Pro-Arg-p-nitroanilide as substrate preincubated for 5 mins before substrate addition measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50359560(CHEMBL1927657)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human alpha-thrombin using sarcosine-Pro-Arg-p-nitroanilide as substrate preincubated for 5 mins before substrate addition measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50359563(CHEMBL1927654)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of human alpha-thrombin using sarcosine-Pro-Arg-p-nitroanilide as substrate preincubated for 5 mins before substrate addition measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50359566(CHEMBL1927663)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of human alpha-thrombin using sarcosine-Pro-Arg-p-nitroanilide as substrate preincubated for 5 mins before substrate addition measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50359561(CHEMBL1927656)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibition of human alpha-thrombin using sarcosine-Pro-Arg-p-nitroanilide as substrate preincubated for 5 mins before substrate addition measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50359558(CHEMBL1927659)
Affinity DataIC50:  2.62E+4nMAssay Description:Inhibition of human alpha-thrombin using sarcosine-Pro-Arg-p-nitroanilide as substrate preincubated for 5 mins before substrate addition measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50359565(CHEMBL1927664)
Affinity DataIC50:  7.30E+4nMAssay Description:Inhibition of human alpha-thrombin using sarcosine-Pro-Arg-p-nitroanilide as substrate preincubated for 5 mins before substrate addition measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50359567(CHEMBL1927662)
Affinity DataIC50:  9.80E+4nMAssay Description:Inhibition of human alpha-thrombin using sarcosine-Pro-Arg-p-nitroanilide as substrate preincubated for 5 mins before substrate addition measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50359564(CHEMBL1927653)
Affinity DataIC50:  6.01E+5nMAssay Description:Inhibition of human alpha-thrombin using sarcosine-Pro-Arg-p-nitroanilide as substrate preincubated for 5 mins before substrate addition measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001589(CHEMBL3237721)
Affinity DataEC50:  35nMAssay Description:Agonist activity at rat mu opioid receptor expressed in rat C6 cells assessed as stimulation of [35S]-GTPgammaS binding after 1 hr by GF/C filtersMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001588(CHEMBL3237720)
Affinity DataEC50:  4.70nMAssay Description:Agonist activity at rat mu opioid receptor expressed in rat C6 cells assessed as stimulation of [35S]-GTPgammaS binding after 1 hr by GF/C filtersMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001590(CHEMBL3237722)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at rat mu opioid receptor expressed in rat C6 cells assessed as stimulation of [35S]-GTPgammaS binding after 1 hr by GF/C filtersMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50001608(CHEMBL3237723)
Affinity DataEC50:  37nMAssay Description:Agonist activity at rat mu opioid receptor expressed in rat C6 cells assessed as stimulation of [35S]-GTPgammaS binding after 1 hr by GF/C filtersMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed