Affinity DataKi: 19nMAssay Description:Antagonist activity at mouse MC4R expressed in HEK293 cells assessed as effect on MT2 peptide-induced response by CRE/beta-galactosidase reporter gen...More data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Antagonist activity at mouse MC3R expressed in HEK293 cells assessed as effect on MT2 peptide-induced response by CRE/beta-galactosidase reporter gen...More data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Antagonist activity at mouse MC3R expressed in HEK293 cells assessed as effect on MT2 peptide-induced response by CRE/beta-galactosidase reporter gen...More data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Antagonist activity at mouse MC3R expressed in HEK293 cells assessed as effect on MT2 peptide-induced response by CRE/beta-galactosidase reporter gen...More data for this Ligand-Target Pair
Affinity DataKi: 5.01E+3nMAssay Description:Antagonist activity at mouse MC3R expressed in HEK293 cells assessed as effect on MT2 peptide-induced response by CRE/beta-galactosidase reporter gen...More data for this Ligand-Target Pair
Affinity DataKi: 6.17E+3nMAssay Description:Antagonist activity at mouse MC3R expressed in HEK293 cells assessed as effect on MT2 peptide-induced response by CRE/beta-galactosidase reporter gen...More data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
Affinity DataEC50: 1.46E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0970nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 64nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 770nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0630nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.05E+4nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 7.75E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 0.0780nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 390nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 0.00800nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 550nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 7.42nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 22.4nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 8.03nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 7.41nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 2.60nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 1.47nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 2.04nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 17.6nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 2.85nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 51.1nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 340nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 5.20nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 226nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 730nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem
Curated by ChEMBL
The Hebrew University Of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 3.26nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.24E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair