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Found 207 with Last Name = 'portillo' and Initial = 'f'
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50252902(Ac-His-DNal(2)-Arg-Trp-NH2 | CHEMBL454736)
Affinity DataKi:  19nMAssay Description:Antagonist activity at mouse MC4R expressed in HEK293 cells assessed as effect on MT2 peptide-induced response by CRE/beta-galactosidase reporter gen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50115373(2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionyl...)
Affinity DataKi:  260nMAssay Description:Antagonist activity at mouse MC3R expressed in HEK293 cells assessed as effect on MT2 peptide-induced response by CRE/beta-galactosidase reporter gen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50252903(Ac-His-DPhe(3,4-diCl)-Arg-Trp-NH2 | CHEMBL501394)
Affinity DataKi:  260nMAssay Description:Antagonist activity at mouse MC3R expressed in HEK293 cells assessed as effect on MT2 peptide-induced response by CRE/beta-galactosidase reporter gen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50252900(Ac-His-DPhe(pBr)-Arg-Trp-NH2 | CHEMBL502093)
Affinity DataKi:  350nMAssay Description:Antagonist activity at mouse MC3R expressed in HEK293 cells assessed as effect on MT2 peptide-induced response by CRE/beta-galactosidase reporter gen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50252902(Ac-His-DNal(2)-Arg-Trp-NH2 | CHEMBL454736)
Affinity DataKi:  5.01E+3nMAssay Description:Antagonist activity at mouse MC3R expressed in HEK293 cells assessed as effect on MT2 peptide-induced response by CRE/beta-galactosidase reporter gen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50252901(Ac-His-DPhe(pCF3)-Arg-Trp-NH2 | CHEMBL501679)
Affinity DataKi:  6.17E+3nMAssay Description:Antagonist activity at mouse MC3R expressed in HEK293 cells assessed as effect on MT2 peptide-induced response by CRE/beta-galactosidase reporter gen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374671(CHEMBL272660)
Affinity DataIC50:  60nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374672(CHEMBL271586)
Affinity DataIC50:  60nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374673(CHEMBL408398)
Affinity DataIC50:  90nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374670(CHEMBL270923)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50374669(CHEMBL406985)
Affinity DataEC50:  1.46E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.0970nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50374670(CHEMBL270923)
Affinity DataEC50:  150nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374671(CHEMBL272660)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374669(CHEMBL406985)
Affinity DataEC50:  120nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374672(CHEMBL271586)
Affinity DataEC50:  240nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374673(CHEMBL408398)
Affinity DataEC50:  64nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50374673(CHEMBL408398)
Affinity DataEC50:  770nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50374673(CHEMBL408398)
Affinity DataEC50:  4nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374673(CHEMBL408398)
Affinity DataEC50:  7nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.0630nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50374671(CHEMBL272660)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50374670(CHEMBL270923)
Affinity DataEC50:  2.05E+4nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50374672(CHEMBL271586)
Affinity DataEC50:  7.75E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50374669(CHEMBL406985)
Affinity DataEC50:  18nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50374671(CHEMBL272660)
Affinity DataEC50:  4nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50374672(CHEMBL271586)
Affinity DataEC50:  5nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.0780nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374669(CHEMBL406985)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374670(CHEMBL270923)
Affinity DataEC50:  390nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374672(CHEMBL271586)
Affinity DataEC50:  26nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.00800nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374671(CHEMBL272660)
Affinity DataEC50:  28nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374670(CHEMBL270923)
Affinity DataEC50:  550nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50252903(Ac-His-DPhe(3,4-diCl)-Arg-Trp-NH2 | CHEMBL501394)
Affinity DataEC50:  7.42nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50252902(Ac-His-DNal(2)-Arg-Trp-NH2 | CHEMBL454736)
Affinity DataEC50:  22.4nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50252901(Ac-His-DPhe(pCF3)-Arg-Trp-NH2 | CHEMBL501679)
Affinity DataEC50:  8.03nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50115373(2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionyl...)
Affinity DataEC50:  7.41nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50252900(Ac-His-DPhe(pBr)-Arg-Trp-NH2 | CHEMBL502093)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50252899(Ac-His-DPhe(pCl)-Arg-Trp-NH2 | CHEMBL491870)
Affinity DataEC50:  1.47nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50252898(Ac-His-DPhe(pF)-Arg-Trp-NH2 | CHEMBL444219)
Affinity DataEC50:  2.04nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50252897(Ac-His-DPhe(pNO2)-Arg-Trp-NH2 | CHEMBL451423)
Affinity DataEC50:  17.6nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50252896(Ac-His-DPhe(pCN)-Arg-Trp-NH2 | CHEMBL448536)
Affinity DataEC50:  2.85nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50252895(Ac-His-DPhe(pBz)-Arg-Trp-NH2 | CHEMBL455826)
Affinity DataEC50:  51.1nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50252894(Ac-His-DPhe(pt-Bu)-Arg-Trp-NH2 | CHEMBL488355)
Affinity DataEC50:  340nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50252893(Ac-His-DPhe(pCH3)-Arg-Trp-NH2 | CHEMBL503449)
Affinity DataEC50:  5.20nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50252892(Ac-His-DPhe(pNH2)-Arg-Trp-NH2 | CHEMBL500516)
Affinity DataEC50:  226nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50115366(2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionyl...)
Affinity DataEC50:  730nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50034922((S)-2-{(R)-2-[(S)-2-Acetylamino-3-(1H-imidazol-4-y...)
Affinity DataEC50:  3.26nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50252904(Ac-His-DPhe(m-Cl)-Arg-Trp-NH2 | CHEMBL510687)
Affinity DataEC50:  1.24E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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