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Found 43 with Last Name = 'probert' and Initial = 'aw'
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50344821(10-hydroxymethyl-5-imino-(2S)-12,13-dioxa-4,6-diaz...)
Affinity DataIC50:  14nMAssay Description:Inhibition of Na+ influx in chinese hamster ovary cells expressing rat brain sodium channel type IIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172933(5-chloro-N'-(2-(trifluoromethyl)phenylsulfonyl)-1H...)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50017702(1-(bis(4-fluorophenyl)methyl)-4-cinnamylpiperazine...)
Affinity DataIC50:  420nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172933(5-chloro-N'-(2-(trifluoromethyl)phenylsulfonyl)-1H...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172943(5-chloro-N'-(o-tolylsulfonyl)-1H-indole-2-carbohyd...)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172934(5-chloro-N'-(m-tolylsulfonyl)-1H-indole-2-carbohyd...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172945(CHEMBL205902 | N'-(phenylsulfonyl)dibenzo[b,d]fura...)
Affinity DataIC50:  2.35E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM23619(2-{4-[4,4-bis(4-fluorophenyl)butyl]piperazin-1-yl}...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172944(5-bromo-N'-(phenylsulfonyl)benzofuran-2-carbohydra...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043993(CHEMBL282833 | N-[3-(2,6-Dimethyl-piperidin-1-yl)-...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172940(CHEMBL437702 | N'-[(3-methylphenyl)sulfonyl]dibenz...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, mitochondrial(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172933(5-chloro-N'-(2-(trifluoromethyl)phenylsulfonyl)-1H...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of rat BCATmMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50044001(CHEMBL93106 | N-[3-(2,6-Dimethyl-piperidin-1-yl)-p...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172931(CHEMBL205475 | N'-[(2-methylphenyl)sulfonyl]dibenz...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043984(2,2-Bis-(2-chloro-phenyl)-N-[3-(2,6-dimethyl-piper...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043992(1-[3-(2,6-Dimethyl-piperidin-1-yl)-propyl]-3,3-dip...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172942(5-chloro-N'-(phenylsulfonyl)benzofuran-2-carbohydr...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043990(1-Phenyl-cyclohexanecarboxylic acid [3-(2,6-dimeth...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043998(2,2-Bis-(4-chloro-phenyl)-N-[3-(2,6-dimethyl-piper...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50044000(2,2-Bis-(4-bromo-phenyl)-N-[3-(2,6-dimethyl-piperi...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172932(5-chloro-N'-(2-chlorophenylsulfonyl)-1H-indole-2-c...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043995(CHEMBL92071 | N-[3-(2,6-Dimethyl-piperidin-1-yl)-p...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043994(CHEMBL92918 | N-[3-(2,6-Dimethyl-piperidin-1-yl)-p...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043991(2-Cyclopentyl-N-[3-(2,6-dimethyl-piperidin-1-yl)-p...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172947(5-methoxy-N'-(phenylsulfonyl)benzofuran-2-carbohyd...)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172930(CHEMBL379025 | N'-[(2-chlorophenyl)sulfonyl]dibenz...)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043986(CHEMBL329245 | N-[3-(2,6-Dimethyl-piperidin-1-yl)-...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043997(9H-Xanthene-9-carboxylic acid [3-(2,6-dimethyl-pip...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172936(CHEMBL437697 | N'-(phenylsulfonyl)quinoline-6-carb...)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172937(5-bromo-N'-(phenylsulfonyl)-1H-indole-2-carbohydra...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172929(CHEMBL205220 | N'-(phenylsulfonyl)benzofuran-2-car...)
Affinity DataIC50:  1.83E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043996(9H-Fluorene-9-carboxylic acid [3-(2,6-dimethyl-pip...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043999(CHEMBL93838 | N-[3-(2,6-Dimethyl-piperidin-1-yl)-p...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172928(CHEMBL382232 | N'-(phenylsulfonyl)quinoline-3-carb...)
Affinity DataIC50:  3.33E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172941(CHEMBL205274 | N'-[(3-chlorophenyl)sulfonyl]dibenz...)
Affinity DataIC50: >3.50E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172935(CHEMBL207686 | N'-(phenylsulfonyl)-1H-indole-2-car...)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172946(CHEMBL205044 | N'-[(4-chlorophenyl)sulfonyl]dibenz...)
Affinity DataIC50:  3.72E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172938(CHEMBL380652 | N'-[(4-methylphenyl)sulfonyl]dibenz...)
Affinity DataIC50:  5.10E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172939(5-methoxy-N'-(phenylsulfonyl)-1H-indole-2-carbohyd...)
Affinity DataIC50:  5.68E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043987(3-(3-Dimethylamino-propyl)-5,5-diphenyl-imidazolid...)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043989(CHEMBL93271 | N-[3-(2,6-Dimethyl-piperidin-1-yl)-p...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043985(CHEMBL93065 | N-[3-(2,6-Dimethyl-piperidin-1-yl)-p...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50043988(3-[3-(2,6-Dimethyl-piperidin-1-yl)-propyl]-1,1-dip...)
Affinity DataIC50:  1.06E+5nMAssay Description:Inhibition of veratridine-induced Na+ influx in chinese hamster ovary cells expressing alpha subunit of rat brain type voltage-gated sodium channel t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed