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Found 228 with Last Name = 'quan' and Initial = 'c'
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200728((R)-1-(4-oxo-4-phenylbutanoyl)pyrrolidin-2-ylboron...)
Affinity DataKi:  1.70nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200729((R)-1-(2-(2,5-dichlorobenzamido)acetyl)pyrrolidin-...)
Affinity DataKi:  2.20nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200726((R)-1-(2-(cyclopentanecarboxamido)acetyl)pyrrolidi...)
Affinity DataKi:  2.30nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200721((R)-1-(2-(cyclohexanecarboxamido)acetyl)pyrrolidin...)
Affinity DataKi:  2.70nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200723((R)-1-(2-(1-oxoisoindolin-2-yl)acetyl)pyrrolidin-2...)
Affinity DataKi:  2.80nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200720((R)-1-(2-(2,6-dichlorobenzamido)acetyl)pyrrolidin-...)
Affinity DataKi:  4.40nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200732((R)-1-(2-isobutyramidoacetyl)pyrrolidin-2-ylboroni...)
Affinity DataKi:  4.5nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200725((R)-1-(2-(N-methylbenzamido)acetyl)pyrrolidin-2-yl...)
Affinity DataKi:  7.40nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200723((R)-1-(2-(1-oxoisoindolin-2-yl)acetyl)pyrrolidin-2...)
Affinity DataKi:  7.5nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200720((R)-1-(2-(2,6-dichlorobenzamido)acetyl)pyrrolidin-...)
Affinity DataKi:  12nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200733((R)-1-(2-(N-methylisobutyramido)acetyl)pyrrolidin-...)
Affinity DataKi:  13nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMax-like protein X(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388975(CHEMBL2063869)
Affinity DataKi:  14nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from MLXBIR3SG after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200721((R)-1-(2-(cyclohexanecarboxamido)acetyl)pyrrolidin...)
Affinity DataKi:  14nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMax-like protein X(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388974(CHEMBL2063868)
Affinity DataKi:  16nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from MLXBIR3SG after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388975(CHEMBL2063869)
Affinity DataKi:  17nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from cIAP1 BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200726((R)-1-(2-(cyclopentanecarboxamido)acetyl)pyrrolidi...)
Affinity DataKi:  20nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200730((R)-1-(2-acetamidoacetyl)pyrrolidin-2-ylboronic ac...)
Affinity DataKi:  23nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200727((R)-1-(2-benzamidoacetyl)pyrrolidin-2-ylboronic ac...)
Affinity DataKi:  25nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388975(CHEMBL2063869)
Affinity DataKi:  28nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200729((R)-1-(2-(2,5-dichlorobenzamido)acetyl)pyrrolidin-...)
Affinity DataKi:  29nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMax-like protein X(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388970(CHEMBL2063863)
Affinity DataKi:  30nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from MLXBIR3SG after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMax-like protein X(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388969(CHEMBL2063862)
Affinity DataKi:  30nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from MLXBIR3SG after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388974(CHEMBL2063868)
Affinity DataKi:  35nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388975(CHEMBL2063869)
Affinity DataKi:  43nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from cIAP2 BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200732((R)-1-(2-isobutyramidoacetyl)pyrrolidin-2-ylboroni...)
Affinity DataKi:  51nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200736((R)-1-(2-(N-methylacetamido)acetyl)pyrrolidin-2-yl...)
Affinity DataKi:  53nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200724((2R)-1-(2-(N-methyl-5-oxopyrrolidine-2-carboxamido...)
Affinity DataKi:  68nMAssay Description:Inhibition constant against DPP-4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMax-like protein X(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388968(CHEMBL2063866)
Affinity DataKi:  70nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from MLXBIR3SG after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMax-like protein X(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388972(CHEMBL2063865)
Affinity DataKi:  80nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from MLXBIR3SG after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMax-like protein X(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388973(CHEMBL2063867)
Affinity DataKi:  90nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from MLXBIR3SG after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200728((R)-1-(4-oxo-4-phenylbutanoyl)pyrrolidin-2-ylboron...)
Affinity DataKi:  94nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200724((2R)-1-(2-(N-methyl-5-oxopyrrolidine-2-carboxamido...)
Affinity DataKi:  101nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388975(CHEMBL2063869)
Affinity DataKi:  112nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR2 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200727((R)-1-(2-benzamidoacetyl)pyrrolidin-2-ylboronic ac...)
Affinity DataKi:  142nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200724((2R)-1-(2-(N-methyl-5-oxopyrrolidine-2-carboxamido...)
Affinity DataKi:  146nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200736((R)-1-(2-(N-methylacetamido)acetyl)pyrrolidin-2-yl...)
Affinity DataKi:  161nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388970(CHEMBL2063863)
Affinity DataKi:  190nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200725((R)-1-(2-(N-methylbenzamido)acetyl)pyrrolidin-2-yl...)
Affinity DataKi:  191nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200722((R)-1-(2-pivalamidoacetyl)pyrrolidin-2-ylboronic a...)
Affinity DataKi:  191nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200730((R)-1-(2-acetamidoacetyl)pyrrolidin-2-ylboronic ac...)
Affinity DataKi:  211nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200735((R)-1-(2-(methylsulfonamido)acetyl)pyrrolidin-2-yl...)
Affinity DataKi:  246nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200733((R)-1-(2-(N-methylisobutyramido)acetyl)pyrrolidin-...)
Affinity DataKi:  265nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200734((R)-1-((R)-2-acetamidopropanoyl)pyrrolidin-2-ylbor...)
Affinity DataKi:  350nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200731((R)-1-(2-(2-oxopyridin-1(2H)-yl)acetyl)pyrrolidin-...)
Affinity DataKi:  353nMAssay Description:Inhibitory constant against POPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200730((R)-1-(2-acetamidoacetyl)pyrrolidin-2-ylboronic ac...)
Affinity DataKi:  377nMAssay Description:Inhibition constant against DPP-4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388968(CHEMBL2063866)
Affinity DataKi:  410nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388969(CHEMBL2063862)
Affinity DataKi:  430nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMax-like protein X(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388971(CHEMBL2063864)
Affinity DataKi:  460nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from MLXBIR3SG after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50388973(CHEMBL2063867)
Affinity DataKi:  700nMAssay Description:Displacement of 5-FAM-conjugated AVP-diPhe-FAM from XIAP BIR3 domain after 30 mins by fluorescence polarization-based competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50200722((R)-1-(2-pivalamidoacetyl)pyrrolidin-2-ylboronic a...)
Affinity DataKi:  751nMAssay Description:Inhibitiory constant against FAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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