Affinity DataKi: 1.60nMAssay Description:Binding affinity towards human Dopamine Receptor D4 was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-YM 09151 from D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonism of dopamine-stimulated [35S]GTP-gamma-S binding against human Dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:D4 receptor functional activity was measured inhibition of quinpirole stimulated [35S]GTP-gamma-S binding from cell membranes.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]-YM 09151 from D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity towards human Dopamine Receptor D4 was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor of rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]-YM 09151 from D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Binding affinity towards human Dopamine Receptor D4 was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]-YM 09151 from D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity towards human Dopamine Receptor D4 was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity towards human Dopamine Receptor D4 was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Antagonism of dopamine-stimulated [35S]GTP-gamma-S binding against human Dopamine receptor D2 in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]-YM 09151 from D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Dopamine receptor D2 functional activity was assessed via inhibition of forskolin stimulated cAMP production from Whole cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]-YM 09151 from D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-YM 09151 from D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Antagonism of dopamine-stimulated [35S]GTP-gamma-S binding against human Dopamine receptor D4 in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity towards human dopamine D4 receptor was determined via standard competitive displacement assays using [3H]-YM 09151 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]-YM 09151 from D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]-YM 09151 from D4 receptorMore data for this Ligand-Target Pair