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Found 576 with Last Name = 'ralph' and Initial = 'm'
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305511(5-(3-(4-(3,5-difluoro-2-methylphenoxy)piperidin-1-...)
Affinity DataKi:  0.400nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305512(2-methoxy-5-(3-(methoxymethyl)-5-(4-(o-tolyloxy)pi...)
Affinity DataKi:  2.20nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305510(5-(3-(4-(3-fluoro-2-methylphenoxy)piperidin-1-yl)-...)
Affinity DataKi:  2.60nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305509(5-(3-(4-(4-fluoro-2-methylphenoxy)piperidin-1-yl)-...)
Affinity DataKi:  4.20nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305508(2-methoxy-5-(3-methyl-5-(4-(o-tolyloxy)piperidin-1...)
Affinity DataKi:  5.40nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305518((R)-5-(3-(3-(3,5-difluoro-2-methylphenoxy)pyrrolid...)
Affinity DataKi:  5.80nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295778(2-(2,6-dimethylphenoxy)-5-(4-(6-methoxypyridin-3-y...)
Affinity DataKi:  5.90nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50262270(2-(4-fluoro-2-methylphenyl)-5-(4-(6-methoxypyridin...)
Affinity DataKi:  6nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50262270(2-(4-fluoro-2-methylphenyl)-5-(4-(6-methoxypyridin...)
Affinity DataKi:  6nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295779(2-(2-chloro-3,6-difluorophenoxy)-5-(4-(6-methoxypy...)
Affinity DataKi:  8.80nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295777(2-(4-fluoro-2-methylphenoxy)-5-(4-(6-methoxypyridi...)
Affinity DataKi:  9.40nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305506(5-(3-(3-(2-chloro-4-fluorophenoxy)azetidin-1-yl)-5...)
Affinity DataKi:  9.5nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50314514(5-(2,3-dimethylphenyl)-N-(2-methoxyethyl)-N-(6-met...)
Affinity DataKi:  11nMAssay Description:Antagonist activity at human cloned OT receptor by cell based beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295772(2-(4-(6-methoxypyridin-3-yl)-5-methyl-4H-1,2,4-tri...)
Affinity DataKi:  12.5nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50313813(CHEMBL1077300 | N-ethyl-3-(3-fluoro-2-methylphenox...)
Affinity DataKi:  13.9nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50314513(5-(2,3-dimethylphenyl)-N-isopropyl-N-(6-methoxypyr...)
Affinity DataKi:  14nMAssay Description:Antagonist activity at human cloned OT receptor by cell based beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295776(2-(3-fluoro-2-methylphenoxy)-5-(4-(6-methoxypyridi...)
Affinity DataKi:  14.6nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305524(5-(3-(3-(4-fluoro-2-methylphenoxy)azetidin-1-yl)-5...)
Affinity DataKi:  17.5nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305524(5-(3-(3-(4-fluoro-2-methylphenoxy)azetidin-1-yl)-5...)
Affinity DataKi:  17.5nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305517((R)-5-(3-(3-(4-fluoro-2-methylphenoxy)pyrrolidin-1...)
Affinity DataKi:  17.9nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305526(5-(3-(3-(4-fluoro-2-methylphenoxy)azetidin-1-yl)-5...)
Affinity DataKi:  18.4nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50313817(5-(3-(3-(3-fluoro-2-methylphenoxy)azetidin-1-yl)-5...)
Affinity DataKi:  19.7nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305508(2-methoxy-5-(3-methyl-5-(4-(o-tolyloxy)piperidin-1...)
Affinity DataKi:  21.6nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295771(2-(2-chlorophenoxy)-5-(4-(6-methoxypyridin-3-yl)-5...)
Affinity DataKi:  23.6nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305512(2-methoxy-5-(3-(methoxymethyl)-5-(4-(o-tolyloxy)pi...)
Affinity DataKi:  24.4nMAssay Description:Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50314512(5-(2,3-dimethylphenyl)-N-ethyl-N-(6-methoxypyridin...)
Affinity DataKi:  25nMAssay Description:Antagonist activity at human cloned OT receptor by cell based beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305523(5-(3-(3-(2-chloro-4-fluorophenoxy)azetidin-1-yl)-5...)
Affinity DataKi:  28.4nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305523(5-(3-(3-(2-chloro-4-fluorophenoxy)azetidin-1-yl)-5...)
Affinity DataKi:  28.4nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305516((R)-2-methoxy-5-(3-(methoxymethyl)-5-(3-(o-tolylox...)
Affinity DataKi:  28.5nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50314511(CHEMBL1092458 | N-ethyl-5-(3-fluoro-2-methylphenyl...)
Affinity DataKi:  29nMAssay Description:Antagonist activity at human cloned OT receptor by cell based beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305515((R)-5-(3-(3-(4-fluoro-2-methylphenoxy)pyrrolidin-1...)
Affinity DataKi:  31.8nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305522(5-(3-(3-(2-chlorophenoxy)azetidin-1-yl)-5-(methoxy...)
Affinity DataKi:  32.5nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305514((R)-2-methoxy-5-(3-methyl-5-(3-(o-tolyloxy)pyrroli...)
Affinity DataKi:  35.9nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50313812(3-(3,5-difluoro-2-methylphenoxy)-N-ethyl-N-(6-meth...)
Affinity DataKi:  36.7nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295780(2-(2,4-dichlorophenoxy)-5-(4-(6-methoxypyridin-3-y...)
Affinity DataKi:  37.5nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305525(5-(3-(3-(5-fluoro-2-methylphenoxy)azetidin-1-yl)-5...)
Affinity DataKi:  40nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50314515(CHEMBL1093776 | N-ethyl-N-(6-methoxypyridin-3-yl)-...)
Affinity DataKi:  41nMAssay Description:Antagonist activity at human cloned OT receptor by cell based beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50313816(5-(3-(3-(3,5-difluoro-2-methylphenoxy)azetidin-1-y...)
Affinity DataKi:  41.4nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50313815(CHEMBL1094050 | N-ethyl-3-(4-fluoro-2-methylphenox...)
Affinity DataKi:  43nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50314522(CHEMBL1089272 | N-ethyl-N-(6-methoxypyridin-3-yl)-...)
Affinity DataKi:  48nMAssay Description:Antagonist activity at human cloned OT receptor by cell based beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50313814(3-(2-chloro-4-fluorophenoxy)-N-ethyl-N-(6-methoxyp...)
Affinity DataKi:  48.4nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50295773(2-(2-ethylphenoxy)-5-(4-(6-methoxypyridin-3-yl)-5-...)
Affinity DataKi:  52.3nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta-lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50305521(5-(3-(3-(2-chlorophenoxy)azetidin-1-yl)-5-methyl-4...)
Affinity DataKi:  55.1nMAssay Description:Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50313811(3-(2-chloro-4-fluorophenoxy)-N-(6-methoxypyridin-3...)
Affinity DataKi:  67.2nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by beta lactamase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50314524(CHEMBL1093709 | N-ethyl-6-(4-methoxyphenyl)-N-(6-m...)
Affinity DataKi:  84nMAssay Description:Antagonist activity at human cloned OT receptor by cell based beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50314520(CHEMBL1093341 | N-ethyl-5-methoxy-N-(6-methoxypyri...)
Affinity DataKi:  85nMAssay Description:Antagonist activity at human cloned OT receptor by cell based beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50314516(CHEMBL1088765 | N-ethyl-N-(6-methoxypyridin-3-yl)-...)
Affinity DataKi:  85nMAssay Description:Antagonist activity at human cloned OT receptor by cell based beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50301772((R)-6-(2-methylpiperazin-1-yl)-2-(2-(2-(trifluorom...)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]meselurgine from human recombinant 5HT2C receptor expressed in Swiss mouse 3T3 cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50314502(CHEMBL1092098 | N-(6-methoxypyridin-3-yl)-N-methyl...)
Affinity DataKi:  90nMAssay Description:Antagonist activity at human cloned OT receptor by cell based beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50314518(CHEMBL1088767 | N-ethyl-1-(4-methoxyphenyl)-N-(6-m...)
Affinity DataKi:  91nMAssay Description:Antagonist activity at human cloned OT receptor by cell based beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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