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Found 433 with Last Name = 'rao' and Initial = 'au'
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50386346(CHEMBL2048594)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50386346(CHEMBL2048594)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50386351(CHEMBL2048589)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50386346(CHEMBL2048594)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299031(2-(1,4'-bipiperidin-1'-yl)-6-(2-methoxypyridin-4-y...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50386364(CHEMBL2048592)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50386346(CHEMBL2048594)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50386351(CHEMBL2048589)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210759(US9290454, 4.4)
Affinity DataKi:  5.16nM ΔG°:  -51.3kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210749(US9290454, 3.1)
Affinity DataKi:  5.79nM ΔG°:  -51.0kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210750(US9290454, 3.2)
Affinity DataKi:  6.50nM ΔG°:  -50.6kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50386364(CHEMBL2048592)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210764(US9290454, 7.2)
Affinity DataKi:  7.79nM ΔG°:  -50.2kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299045(5-(2-(1,4'-bipiperidin-1'-yl)thiazolo[4,5-c]pyridi...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50386347(CHEMBL2048595)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210751(US9290454, 3.3)
Affinity DataKi:  8.20nM ΔG°:  -50.0kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210752(US9290454, 3.4)
Affinity DataKi:  8.84nM ΔG°:  -49.8kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299035(CHEMBL574387 | N-(5-(2-(1,4'-bipiperidin-1'-yl)thi...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299014(2-(1,4'-bipiperidin-1'-yl)-6-chlorothiazolo[4,5-c]...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210760(US9290454, 5.1)
Affinity DataKi:  10.2nM ΔG°:  -49.4kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210767(US9290454, 8.1)
Affinity DataKi:  10.9nM ΔG°:  -49.3kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50386350(CHEMBL2048590)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50386353(CHEMBL2048587)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210765(US9290454, 7.3)
Affinity DataKi:  12.7nM ΔG°:  -48.8kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299027(2-(1,4'-bipiperidin-1'-yl)-6-(2-fluoropyridin-4-yl...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210753(US9290454, 3.5)
Affinity DataKi:  13.1nM ΔG°:  -48.8kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210757(US9290454, 4.2)
Affinity DataKi:  13.6nM ΔG°:  -48.7kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50386352(CHEMBL2048588)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210768(US9290454, 8.2)
Affinity DataKi:  14.8nM ΔG°:  -48.4kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210766(US9290454, 7.4)
Affinity DataKi:  14.8nM ΔG°:  -48.4kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50386359(CHEMBL2048581)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50386347(CHEMBL2048595)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299034(5-(2-(1,4'-bipiperidin-1'-yl)thiazolo[4,5-b]pyridi...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299029(5-(2-(1,4'-bipiperidin-1'-yl)thiazolo[4,5-b]pyridi...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299049(5-(2-(1,4'-bipiperidin-1'-yl)thiazolo[4,5-c]pyridi...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210769(US9290454, 8.3)
Affinity DataKi:  17.0nM ΔG°:  -48.1kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210771(US9290454, 8.5)
Affinity DataKi:  17.2nM ΔG°:  -48.0kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210772(US9290454, 8.6)
Affinity DataKi:  17.3nM ΔG°:  -48.0kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50386359(CHEMBL2048581)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from mouse recombinant histamine H3 receptor after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210754(US9290454, 3.6 | US9290454, 3.7)
Affinity DataKi:  18.7nM ΔG°:  -47.8kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50299035(CHEMBL574387 | N-(5-(2-(1,4'-bipiperidin-1'-yl)thi...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse brain histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299040(2-(1,4'-bipiperidin-1'-yl)-6-(2-fluoropyridin-3-yl...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50299045(5-(2-(1,4'-bipiperidin-1'-yl)thiazolo[4,5-c]pyridi...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from mouse brain histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210758(US9290454, 4.3)
Affinity DataKi:  20.7nM ΔG°:  -47.5kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210763(US9290454, 7.1)
Affinity DataKi:  21.5nM ΔG°:  -47.4kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299041(5-(2-(1,4'-bipiperidin-1'-yl)thiazolo[4,5-c]pyridi...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM210756(US9290454, 4.1)
Affinity DataKi:  22.5nM ΔG°:  -47.3kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299017(5-(2-(1,4'-bipiperidin-1'-yl)thiazolo[4,5-b]pyridi...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299046(5-(2-(1,4'-bipiperidin-1'-yl)thiazolo[4,5-c]pyridi...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299036(2-(1,4'-bipiperidin-1'-yl)-6-(pyrimidin-5-yl)thiaz...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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