Compile Data Set for Download or QSAR
maximum 50k data
Found 152 with Last Name = 'renzetti' and Initial = 'ar'
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404016(CHEMBL2112922)
Affinity DataKi:  0.0500nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404016(CHEMBL2112922)
Affinity DataKi:  0.0501nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50472916(CHEMBL223221 | MEN-11690)
Affinity DataKi:  0.100nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404025(CHEMBL2112925)
Affinity DataKi:  0.126nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50366377(CHEMBL334721 | MEN-10627)
Affinity DataKi:  0.631nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404017(CHEMBL2112923)
Affinity DataKi:  0.631nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404023(CHEMBL159449)
Affinity DataKi:  1.60nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404021(CHEMBL161242)
Affinity DataKi:  1.60nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50472917(CHEMBL323884 | MEN-11749)
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404020(CHEMBL435324 | MEN-11558)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]NKA from human Tachykinin receptor 2 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404020(CHEMBL435324 | MEN-11558)
Affinity DataKi:  2nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50472911(CHEMBL407782 | MEN-11420)
Affinity DataKi:  2.5nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404019(CHEMBL345402)
Affinity DataKi:  2.5nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470323(CHEMBL327505)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029895(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029905(4'-(2-Butyl-4-methyl-6-oxo-6H-pyrimidin-1-ylmethyl...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029899(3-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029908(4'-(4-Butyl-6-oxo-1-thiophen-2-ylmethyl-1,6-dihydr...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029893(2-[4-Butyl-5-(2'-carboxy-biphenyl-4-ylmethyl)-2-me...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029906(2-[4-Butyl-5-(2'-carboxy-biphenyl-4-ylmethyl)-2-me...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029909(4'-[4-Butyl-1-(2-carboxy-benzyl)-6-oxo-1,6-dihydro...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029907(4'-(1-Benzyl-4-butyl-6-oxo-1,6-dihydro-pyrimidin-5...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029910(4'-(4-Butyl-6-oxo-1,6-dihydro-pyrimidin-5-ylmethyl...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029911(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029903(3-Benzyl-6-butyl-2-methyl-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404022(CHEMBL2112926)
Affinity DataKi:  4nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029894(4'-(4-Butyl-2-methyl-6-oxo-1,6-dihydro-pyrimidin-5...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029904(4'-[4-Butyl-1-(2-carboxy-benzyl)-2-methyl-6-oxo-1,...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029902(6-Butyl-2-methyl-5-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029897(4'-[4-Butyl-1-(4-carboxy-benzyl)-6-oxo-1,6-dihydro...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029901(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029892(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50241501(6-Butyl-2-methyl-5-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50241491(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029896(4'-(2-Butyl-6-oxo-6H-pyrimidin-1-ylmethyl)-bipheny...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470328(CHEMBL317300)
Affinity DataKi:  4.40nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470310(CHEMBL98592)
Affinity DataKi:  4.5nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404014(CHEMBL159585)
Affinity DataKi:  5nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404026(CHEMBL350596)
Affinity DataKi:  6.30nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404024(CHEMBL346285)
Affinity DataKi:  6.30nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470321(CHEMBL99008)
Affinity DataKi:  7.70nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50472912(CHEMBL116564 | MEN-11712)
Affinity DataKi:  7.90nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404015(CHEMBL161288)
Affinity DataKi:  7.90nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470340(CHEMBL98370)
Affinity DataKi:  8.80nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470326(CHEMBL319990)
Affinity DataKi:  9.10nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50472910(CHEMBL263194)
Affinity DataKi:  10nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50404018(CHEMBL2112924)
Affinity DataKi:  10nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Menarini Ricerche S.P.A. Laboratori Di Firenze

Curated by ChEMBL
LigandPNGBDBM50472908(CHEMBL336053)
Affinity DataKi:  10nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470313(CHEMBL441640)
Affinity DataKi:  12nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470330(CHEMBL318194)
Affinity DataKi:  12nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 152 total ) | Next | Last >>
Jump to: