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Found 145 with Last Name = 'richards' and Initial = 'ng'
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50378579(CHEMBL1627258)
Affinity DataKi:  2.5nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as assessed as overall inhibition constant for ammonia dependent production of i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392270(CHEMBL2153507)
Affinity DataKi:  8nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as overall inhibition constant for glutamine dependent production of inorganic p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50378579(CHEMBL1627258)
Affinity DataKi:  24nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as overall inhibition constant for glutamine dependent production of inorganic p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392270(CHEMBL2153507)
Affinity DataKi:  33nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as assessed as overall inhibition constant for ammonia dependent production of i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50378579(CHEMBL1627258)
Affinity DataKi:  280nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as assessed as initial inhibition constant for ammonia dependent production of i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392271(CHEMBL2153508)
Affinity DataKi:  310nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as assessed as overall inhibition constant for ammonia dependent production of i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392270(CHEMBL2153507)
Affinity DataKi:  450nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as assessed as initial inhibition constant for ammonia dependent production of i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392270(CHEMBL2153507)
Affinity DataKi:  490nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as initial inhibition constant for glutamine dependent production of inorganic p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392271(CHEMBL2153508)
Affinity DataKi:  840nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as overall inhibition constant for glutamine dependent production of inorganic p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50378579(CHEMBL1627258)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as initial inhibition constant for glutamine dependent production of inorganic p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392271(CHEMBL2153508)
Affinity DataKi:  3.04E+3nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as assessed as initial inhibition constant for ammonia dependent production of i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50392271(CHEMBL2153508)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 cells assessed as initial inhibition constant for glutamine dependent production of inorganic p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50378579(CHEMBL1627258)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 insect cells assessed as overall inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAsparagine synthetase [glutamine-hydrolyzing](Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50378579(CHEMBL1627258)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of human recombinant ASNS expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144869(CHEMBL411775 | Tyr-c[Asp-His-DPhe-Arg-Trp-Asn-Ala-...)
Affinity DataIC50:  0.260nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144869(CHEMBL411775 | Tyr-c[Asp-His-DPhe-Arg-Trp-Asn-Ala-...)
Affinity DataIC50:  0.960nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144877(CHEMBL269274)
Affinity DataIC50:  1.46nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataIC50:  4.22nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-NDP-MSH; ND = not determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144877(CHEMBL269274)
Affinity DataIC50:  4.45nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144871(CHEMBL428134)
Affinity DataIC50:  4.74nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144882(CHEMBL266288)
Affinity DataIC50:  5.48nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50155865(CHEMBL2373991 | CUDPUATUYCRFFNAFCYCRKL)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]-hAGRP(87-132) from mouse Melanocortin 4 ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144871(CHEMBL428134)
Affinity DataIC50:  29.8nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50155865(CHEMBL2373991 | CUDPUATUYCRFFNAFCYCRKL)
Affinity DataIC50:  140nMAssay Description:Displacement of [125I]-hAGRP(87-132) from mouse Melanocortin 3 ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50410195(CHEMBL2096710)
Affinity DataIC50:  275nMAssay Description:Displacement of [125I]-hAGRP(87-132) from mouse Melanocortin 4 ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144880(CHEMBL406032 | Tyr-c[Asp-His-Phe-Arg-Trp-Asn-Ala-P...)
Affinity DataIC50:  290nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144880(CHEMBL406032 | Tyr-c[Asp-His-Phe-Arg-Trp-Asn-Ala-P...)
Affinity DataIC50:  540nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144879(CHEMBL406550 | Tyr-c[Asp-DPhe-Arg-Trp-Asn-Ala-Phe-...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144878(CHEMBL402258 | Tyr-c[Asp-Arg-Phe-Phe-Asn-Ala-Phe-D...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144874(CHEMBL440633 | Tyr-c[Asp-Phe-Arg-Trp-Asn-Ala-Phe-D...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144878(CHEMBL402258 | Tyr-c[Asp-Arg-Phe-Phe-Asn-Ala-Phe-D...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144879(CHEMBL406550 | Tyr-c[Asp-DPhe-Arg-Trp-Asn-Ala-Phe-...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144881(CHEMBL413465 | Tyr-c[Asp-Trp-Arg-Phe-Asn-Ala-Phe-D...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144874(CHEMBL440633 | Tyr-c[Asp-Phe-Arg-Trp-Asn-Ala-Phe-D...)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144870(CHEMBL410091 | Tyr-c[Asp-Trp-Arg-DPhe-Asn-Ala-Phe-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144870(CHEMBL410091 | Tyr-c[Asp-Trp-Arg-DPhe-Asn-Ala-Phe-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144881(CHEMBL413465 | Tyr-c[Asp-Trp-Arg-Phe-Asn-Ala-Phe-D...)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50410195(CHEMBL2096710)
Affinity DataIC50:  1.17E+4nMAssay Description:Displacement of [125I]-hAGRP(87-132) from mouse Melanocortin 3 ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422954(CHEMBL2304247)
Affinity DataEC50:  6.20nMAssay Description:Displacement of MT2 from mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422955(CHEMBL2304248)
Affinity DataEC50:  8.30E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422956(CHEMBL2304249)
Affinity DataEC50:  6.24E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422955(CHEMBL2304248)
Affinity DataEC50:  1.75E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422954(CHEMBL2304247)
Affinity DataEC50:  6.10nMAssay Description:Displacement of MT2 from mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422954(CHEMBL2304247)
Affinity DataEC50:  93nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422957(CHEMBL2304250)
Affinity DataEC50:  3.77E+4nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422956(CHEMBL2304249)
Affinity DataEC50:  1.14E+4nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422954(CHEMBL2304247)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422954(CHEMBL2304247)
Affinity DataEC50: >100nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422956(CHEMBL2304249)
Affinity DataEC50:  120nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422954(CHEMBL2304247)
Affinity DataEC50:  6.90nMAssay Description:Displacement of MT2 from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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