Affinity DataIC50: 5nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 172nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 252nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 279nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
Affinity DataIC50: 302nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 788nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.58E+3nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Binding affinity for human cloned Histamine H1 receptor expressed in CHO cells using [3H]pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
TargetGeranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 2.08E+4nMAssay Description:Binding affinity for human cloned 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of HDAC in human leukemic CEM cellsMore data for this Ligand-Target Pair