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Found 2442 with Last Name = 'rivier' and Initial = 'j'
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM82286(CAS_59763-91-6 | PP, human | PP,SALMON)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085734(CHEMBL407628 | DiCyclo (4-10/5,5'-8) [Ac-D Nal, D ...)
Affinity DataKi:  0.100nMAssay Description:Competitive radioligand binding assay, in human HEK-293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085777(CHEMBL386166 | Gonadotropin Releasing Hormone anal...)
Affinity DataKi:  0.120nMAssay Description:Affinity for rat gonadotrophin releasing hormone (GnRH) receptor using HEK-293 cells transfected with rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085807(CHEMBL425966 | Gonadotropin Releasing Hormone anal...)
Affinity DataKi:  0.120nMAssay Description:Affinity for rat gonadotrophin releasing hormone (GnRH) receptor using HEK-293 cells transfected with rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085814(CHEMBL405548 | dicyclo(4-10/5,5-8)[Ac-D2Nal-DCpa-D...)
Affinity DataKi:  0.140nMAssay Description:Binding affinity of the compound towards Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085756(CHEMBL439532 | cyclo(1,1'-3)Ac-D-Asp (Gly)-D-Cpa-D...)
Affinity DataKi:  0.140nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK-293More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM86477(FE200041 | d-Phe-d-Phe-d-Nle-d-Arg-NH2)
Affinity DataKi:  0.146nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085791(CHEMBL265240 | Gonadotropin Releasing Hormone anal...)
Affinity DataKi:  0.150nMAssay Description:Affinity for rat gonadotrophin releasing hormone (GnRH) receptor using HEK-293 cells transfected with rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153477(CHEMBL3775524)
Affinity DataKi:  0.160nMAssay Description:Displacement of [125ITyr0-Glu1,Nle17]-PS-Svg in human CRF-R1 expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085715(CHEMBL266300 | DiCyclo (4-10/5,5'-8) [Ac-D Nal, D ...)
Affinity DataKi:  0.160nMAssay Description:Competitive radioligand binding assay, in human HEK-293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 2(Mus musculus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153480(CHEMBL3775195)
Affinity DataKi:  0.170nMAssay Description:Displacement of [125ITyr0-Glu1,Nle17]-PS-Svg in mouse CRF-R2 beta expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085742(CHEMBL414350 | cyclo(1,1'-3)Ac-D-Asp (beta-Ala)-D-...)
Affinity DataKi:  0.170nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK-293More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 2(Mus musculus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153499(CHEMBL3774658)
Affinity DataKi:  0.170nMAssay Description:Displacement of [125ITyr0-Glu1,Nle17]-PS-Svg in mouse CRF-R2 beta expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153473(CHEMBL3775796)
Affinity DataKi:  0.180nMAssay Description:Displacement of [125ITyr0-Glu1]-PD-Svg in human CRF-R1 expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085761(CHEMBL437038 | cyclo(1,1'-3)Ac-D-Asp (Gaba)-D-Cpa-...)
Affinity DataKi:  0.180nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK-293More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50231578(CHEMBL3349022)
Affinity DataKi:  0.200nMAssay Description:Affinity against Neuropeptide Y2 receptor on SK-N-BE2 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85813(Des-AA11-18[Cys7,21,D-Lys9 (Ac), Pro34]-NPY)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153499(CHEMBL3774658)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125ITyr0-Glu1,Nle17]-PS-Svg in human CRF-R1 expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153579(CHEMBL3774395)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125ITyr0-Glu1,Nle17]-PS-Svg in human CRF-R1 expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50231578(CHEMBL3349022)
Affinity DataKi:  0.200nMAssay Description:Affinity against Neuropeptide Y2 receptor on SK-N-BE2 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085718(CHEMBL410820 | DiCyclo (4-10/5,5'-8) [Ac-D Nal, D ...)
Affinity DataKi:  0.200nMAssay Description:Competitive radioligand binding assay, in human HEK-293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085719(CHEMBL438543 | DiCyclo (4-10/5,5'-8) [Ac-D Nal, D ...)
Affinity DataKi:  0.200nMAssay Description:Competitive radioligand binding assay, in human HEK-293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50231578(CHEMBL3349022)
Affinity DataKi:  0.200nMAssay Description:Affinity against Neuropeptide Y2 receptor on SK-N-BE2 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50231578(CHEMBL3349022)
Affinity DataKi:  0.200nMAssay Description:Affinity against Neuropeptide Y2 receptor on SK-N-BE2 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085710(CHEMBL414756 | DiCyclo (4-10/5,5'-8) [Ac-D Nal, D ...)
Affinity DataKi:  0.200nMAssay Description:Competitive radioligand binding assay, in human HEK-293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085799(CHEMBL439083 | Gonadotropin Releasing Hormone anal...)
Affinity DataKi:  0.220nMAssay Description:Affinity for rat gonadotrophin releasing hormone (GnRH) receptor using HEK-293 cells transfected with rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153481(CHEMBL3774868)
Affinity DataKi:  0.220nMAssay Description:Displacement of [125ITyr0-Glu1,Nle17]-PS-Svg in human CRF-R1 expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 2(Mus musculus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153574(CHEMBL3775778)
Affinity DataKi:  0.220nMAssay Description:Displacement of [125ITyr0-Glu1,Nle17]-PS-Svg in mouse CRF-R2 beta expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085797(CHEMBL407361 | Gonadotropin Releasing Hormone anal...)
Affinity DataKi:  0.220nMAssay Description:Affinity for rat gonadotrophin releasing hormone (GnRH) receptor using HEK-293 cells transfected with rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085720(CHEMBL404930 | DiCyclo (4-10/5,5'-8) [Ac-D Nal, D ...)
Affinity DataKi:  0.230nMAssay Description:Competitive radioligand binding assay, in human HEK-293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085737(CHEMBL438597 | DiCyclo (4-10/5,5'-8) [Ac-D Nal, D ...)
Affinity DataKi:  0.230nMAssay Description:Competitive radioligand binding assay, in human HEK-293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153497(CHEMBL3775030)
Affinity DataKi:  0.240nMAssay Description:Displacement of [125ITyr0-Glu1,Nle17]-PS-Svg in human CRF-R1 expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085783(CHEMBL438897 | Gonadotropin Releasing Hormone anal...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity of the compound towards Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085783(CHEMBL438897 | Gonadotropin Releasing Hormone anal...)
Affinity DataKi:  0.240nMAssay Description:Affinity for rat gonadotrophin releasing hormone (GnRH) receptor using HEK-293 cells transfected with rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085771(CHEMBL436657 | Gonadotropin Releasing Hormone anal...)
Affinity DataKi:  0.25nMAssay Description:Affinity for rat gonadotrophin releasing hormone (GnRH) receptor using HEK-293 cells transfected with rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153498(CHEMBL3774682)
Affinity DataKi:  0.25nMAssay Description:Displacement of [125ITyr0-Glu1,Nle17]-PS-Svg in human CRF-R1 expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085810(CHEMBL406809 | Gonadotropin Releasing Hormone anal...)
Affinity DataKi:  0.260nMAssay Description:Affinity of the compound for rat Gonadotropin-releasing hormone receptor membrane evaluated using HEK-293 cells transfected with rat Gonadotropin-rel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 2(Mus musculus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153579(CHEMBL3774395)
Affinity DataKi:  0.260nMAssay Description:Displacement of [125ITyr0-Glu1]-PD-Svg in mouse CRF-R2 beta expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085768(CHEMBL268538 | Gonadotropin Releasing Hormone anal...)
Affinity DataKi:  0.270nMAssay Description:Affinity for rat gonadotrophin releasing hormone (GnRH) receptor using HEK-293 cells transfected with rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085815(CHEMBL269726 | cyclo(4-10)[Ac-3Pro-DFpa-DTrp-c[Asp...)
Affinity DataKi:  0.270nMAssay Description:Binding affinity of the compound towards Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085732(CHEMBL406094 | DiCyclo (4-10/5,5'-8) [Ac-D Nal, D ...)
Affinity DataKi:  0.270nMAssay Description:Competitive radioligand binding assay, in human HEK-293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085735(CHEMBL412681 | Cyclo (5-8) [Ac-D Nal, D Cpa, D Pal...)
Affinity DataKi:  0.280nMAssay Description:Competitive radioligand binding assay, in human HEK-293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153579(CHEMBL3774395)
Affinity DataKi:  0.280nMAssay Description:Displacement of [125ITyr0-Glu1]-PD-Svg in human CRF-R1 expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50015490(CHEMBL438945 | H-YPSKPDNPGEDAPAEDMARYYSALRHYINLITR...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153482(CHEMBL3775357)
Affinity DataKi:  0.290nMAssay Description:Displacement of [125ITyr0-Glu1,Nle17]-PS-Svg in human CRF-R1 expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 2(Mus musculus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153577(CHEMBL3774465)
Affinity DataKi:  0.290nMAssay Description:Displacement of [125ITyr0-Glu1]-PD-Svg in mouse CRF-R2 beta expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50005530(CHEMBL267633 | D-Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-G...)
Affinity DataKi:  0.300nMAssay Description:Affinity against Neuropeptide Y2 receptor on SK-N-BE2 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50046551(CHEMBL2370625 | Tyr-c(Glu-Ser-Lys-Pro-Gly-Arg-His-...)
Affinity DataKi:  0.300nMAssay Description:Tested against neuropeptide Y1 receptors using SK-N-MC human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50153482(CHEMBL3775357)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125ITyr0-Glu1,Nle17]-PS-Svg in human CRF-R1 expressed in COS-M6 cells after 90 mins by gamma counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50046551(CHEMBL2370625 | Tyr-c(Glu-Ser-Lys-Pro-Gly-Arg-His-...)
Affinity DataKi:  0.300nMAssay Description:Tested against neuropeptide Y2 receptors using SK-N-BE2 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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