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TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31373(CHEMBL28137 | terephthalamide scaffold, 9)
Affinity DataKi:  780nM ΔG°:  -34.9kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31374(CHEMBL286715 | terephthalamide scaffold, 10)
Affinity DataKi:  840nM ΔG°:  -34.7kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31381(CHEMBL282624 | terephthalamide scaffold, 29)
Affinity DataKi:  1.01E+3nM ΔG°:  -34.2kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31379(CHEMBL28872 | terephthalamide scaffold, 27)
Affinity DataKi:  1.79E+3nM ΔG°:  -32.8kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31378(CHEMBL284686 | terephthalamide scaffold, 26)
Affinity DataKi:  1.85E+3nM ΔG°:  -32.7kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31380(terephthalamide scaffold, 28)
Affinity DataKi:  2.31E+3nM ΔG°:  -32.2kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31390(terephthalamide scaffold, 37)
Affinity DataKi:  2.44E+3nM ΔG°:  -32.0kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31387(terephthalamide scaffold, 34)
Affinity DataKi:  3.14E+3nM ΔG°:  -31.4kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31385(CHEMBL281240 | terephthalamide scaffold, 17)
Affinity DataKi:  3.31E+3nM ΔG°:  -31.3kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31376(CHEMBL433422 | terephthalamide scaffold, 24)
Affinity DataKi:  5.85E+3nM ΔG°:  -29.9kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31383(terephthalamide scaffold, 31)
Affinity DataKi:  7.63E+3nM ΔG°:  -29.2kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31386(terephthalamide scaffold, 33)
Affinity DataKi:  8.34E+3nM ΔG°:  -29.0kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31393(terephthalamide scaffold, 40)
Affinity DataKi:  8.36E+3nM ΔG°:  -29.0kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31392(terephthalamide scaffold, 39)
Affinity DataKi:  8.76E+3nM ΔG°:  -28.9kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31388(terephthalamide scaffold, 35)
Affinity DataKi:  8.92E+3nM ΔG°:  -28.8kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31377(terephthalamide scaffold, 25)
Affinity DataKi:  1.09E+4nM ΔG°:  -28.3kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31375(CHEMBL28504 | terephthalamide scaffold, 23)
Affinity DataKi:  1.10E+4nM ΔG°:  -28.3kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31391(terephthalamide scaffold, 38)
Affinity DataKi:  1.14E+4nM ΔG°:  -28.2kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31384(terephthalamide scaffold, 32)
Affinity DataKi:  1.32E+4nM ΔG°:  -27.9kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31404(terephthalamide scaffold, 50)
Affinity DataKi:  8.21E+4nMAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31394(terephthalamide scaffold, 41)
Affinity DataKi:  1.38E+5nM ΔG°:  -22.0kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31395(terephthalamide scaffold, 42)
Affinity DataKi:  2.60E+5nM ΔG°:  -20.5kJ/molepH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31401(terephthalamide scaffold, 47)
Affinity DataKi:  4.50E+5nMAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31396(terephthalamide scaffold, 43)
Affinity DataKi:  7.80E+5nMAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Burkholderia cenocepacia)
H�Pital De Bic�Tre

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Burkholderia cenocepacia 07-34 beta-lactamase PenB1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional dihydrofolate reductase-thymidylate synthase(Cryptosporidium parvum)
Yale University

Curated by ChEMBL
LigandPNGBDBM50496577(CHEMBL3134008)
Affinity DataIC50:  2.30E+5nMAssay Description:Inhibition of DHFR activity of Cryptosporidium hominis thymidylate synthase-dihydrofolate reductase by steady state kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBifunctional dihydrofolate reductase-thymidylate synthase(Cryptosporidium parvum)
Yale University

Curated by ChEMBL
LigandPNGBDBM50496577(CHEMBL3134008)
Affinity DataIC50:  5.70E+5nMAssay Description:Inhibition of thymidylate synthase activity of Cryptosporidium hominis thymidylate synthase-dihydrofolate reductase by steady state kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBifunctional dihydrofolate reductase-thymidylate synthase(Cryptosporidium parvum)
Yale University

Curated by ChEMBL
LigandPNGBDBM50496578(CHEMBL3134009)
Affinity DataIC50:  8.00E+5nMAssay Description:Inhibition of DHFR activity of Cryptosporidium hominis thymidylate synthase-dihydrofolate reductase by steady state kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50496577(CHEMBL3134008)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human DHFRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31405(terephthalamide scaffold, 51)
Affinity DataAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31382(terephthalamide scaffold, 30)
Affinity DatapH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31399(terephthalamide scaffold, 22)
Affinity DataAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31403(terephthalamide scaffold, 49)
Affinity DataAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31402(terephthalamide scaffold, 48)
Affinity DataAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31397(terephthalamide scaffold, 44)
Affinity DataAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31389(CHEMBL29180 | terephthalamide scaffold, 36)
Affinity DatapH: 7.4 T: 25°CAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31400(terephthalamide scaffold, 46)
Affinity DataAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Yale University

LigandPNGBDBM31398(terephthalamide scaffold, 45)
Affinity DataAssay Description:Fluorescence polarization experiments were conducted on a Photon Technology International instrument using a 0.3 cm path length cuvette. Spectra were...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed