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Found 221 with Last Name = 'sada' and Initial = 't'
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50260415(4-(2-Chloro-benzenesulfonyl)-2-(1-methyl-1,2,5,6-t...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50260414(4-(4-tert-Butyl-benzenesulfonyl)-2-(1-methyl-1,2,5...)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50260413(4-(4-Methyl-benzenesulfonyl)-2-(1-methyl-1,2,5,6-t...)
Affinity DataKi:  1.40E+4nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300564(2-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-3-(4-p...)
Affinity DataKi:  1.90E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50260418(4-Benzenesulfonyl-2-(1-methyl-1,2,5,6-tetrahydropy...)
Affinity DataKi:  2.70E+4nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300560(3-butyl-2-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl...)
Affinity DataKi:  3.20E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50260417(4-(2,5-Dichloro-benzenesulfonyl)-2-(1-methyl-1,2,5...)
Affinity DataKi:  3.50E+4nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300563(4-[2-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-4-o...)
Affinity DataKi:  3.70E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300565(2-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-3-(4-n...)
Affinity DataKi:  4.30E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50260420(4-(3-Nitrobenzenesulfonyl)-2-(1-methyl-1,2,5,6-tet...)
Affinity DataKi:  6.20E+4nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50260421(4-(4-Nitro-benzenesulfonyl)-2-(1-methyl-1,2,5,6-te...)
Affinity DataKi:  6.40E+4nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM46858(1-methyl-3,6-dihydro-2H-pyridine-5-carboxylic acid...)
Affinity DataKi:  8.60E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM46858(1-methyl-3,6-dihydro-2H-pyridine-5-carboxylic acid...)
Affinity DataKi:  8.60E+4nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50260419(4-(2-Nitrobenzenesulfonyl)-2-(1-methyl-1,2,5,6-tet...)
Affinity DataKi:  9.60E+4nMAssay Description:Displacement of [3H]Quinuclidinyl benzillate from muscarinic M1 receptor in Wistar rat cortex synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300561(3-isopropyl-2-(1-methyl-1,2,5,6-tetrahydropyridin-...)
Affinity DataKi:  9.70E+4nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300567(3-(3-hydroxy-phenyl)-2-(1-methyl-1,2,5,6-tetrahydr...)
Affinity DataKi:  1.02E+5nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300558(2-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-3-phen...)
Affinity DataKi:  1.05E+5nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300559(3-hexyl-2-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl...)
Affinity DataKi:  1.10E+5nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300562(3-(4-bromophenyl)-2-(1-methyl-1,2,5,6-tetrahydropy...)
Affinity DataKi:  1.22E+5nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300566(3-(4-methyl-2-nitro-phenyl)-2-(1-methyl-1,2,5,6-te...)
Affinity DataKi:  1.25E+5nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300556(3-benzyl-2-(1-methyl-1,2,5,6-tetrahydropyridin-3-y...)
Affinity DataKi:  1.49E+5nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300555(3-(4-chlorophenyl)-2-(1,2,5,6-tetrahydro-1-methylp...)
Affinity DataKi:  2.00E+5nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50300557(3-ethyl-2-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl...)
Affinity DataKi:  2.30E+5nMAssay Description:Displacement of [3H]QNB from muscarinic M1 receptor in Wistar rat brain cortex membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049128(5-(1-Hydroxy-ethyl)-2-propyl-3-[2'-(2H-tetrazol-5-...)
Affinity DataIC50:  4.90nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049118(2-Ethyl-5-(1-hydroxy-1-methyl-ethyl)-3-[2'-(2H-tet...)
Affinity DataIC50:  5.30nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049123(5-Hydroxymethyl-2-propyl-3-[2'-(2H-tetrazol-5-yl)-...)
Affinity DataIC50:  6.90nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50241364(4-(1-hydroxy-1-methylethyl)-2-propyl-1-{[2'-(1H-te...)
Affinity DataIC50:  8.10nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049107(2-Propyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50:  9.10nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049109(2-Butyl-5-(1-hydroxy-1-methyl-ethyl)-3-[2'-(2H-tet...)
Affinity DataIC50:  9.5nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049124(5-Methyl-2-propyl-3-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataIC50:  11nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049116(5-Ethyl-2-propyl-3-(2'-tetrazol-1-yl-biphenyl-4-yl...)
Affinity DataIC50:  12nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50188016(1-[bis(4-fluoro-phenyl)-methyl]-4-(2-pyrrolidin-1-...)
Affinity DataIC50:  17.6nMAssay Description:Inhibition of electric eel AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50188016(1-[bis(4-fluoro-phenyl)-methyl]-4-(2-pyrrolidin-1-...)
Affinity DataIC50:  18.8nMAssay Description:Inhibition of rat brain homogenate AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50188016(1-[bis(4-fluoro-phenyl)-methyl]-4-(2-pyrrolidin-1-...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human serum AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50006909(2-Butyl-5-chloro-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  22nMAssay Description:Inhibition of [125l]-All binding to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50006909(2-Butyl-5-chloro-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  22nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049132(3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-(1-hydroxy-1-...)
Affinity DataIC50:  28nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049112(3-(2'-Carboxy-biphenyl-4-ylmethyl)-5-(1-hydroxy-et...)
Affinity DataIC50:  28nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049122(2-Butyl-3-(2'-carboxy-biphenyl-4-ylmethyl)-5-(1-hy...)
Affinity DataIC50:  30nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50022775((m-Hydroxyphenyl)trimethylammonium dimethylcarbama...)
Affinity DataIC50:  35nMAssay Description:Inhibition of Wistar rat brain AChE by Ellman colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049117(3-(2'-Carboxy-biphenyl-4-ylmethyl)-2-ethyl-5-(1-hy...)
Affinity DataIC50:  37nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50022775((m-Hydroxyphenyl)trimethylammonium dimethylcarbama...)
Affinity DataIC50:  37.5nMAssay Description:Inhibition of rat brain homogenate AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50188013(1-[bis(4-fluoro-phenyl)-methyl]-4-1(benzyl)-4-(2-c...)
Affinity DataIC50:  37.5nMAssay Description:Inhibition of rat brain homogenate AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50022775((m-Hydroxyphenyl)trimethylammonium dimethylcarbama...)
Affinity DataIC50:  40nMAssay Description:Inhibition of Wistar rat brain homogenate AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50022775((m-Hydroxyphenyl)trimethylammonium dimethylcarbama...)
Affinity DataIC50:  41nMAssay Description:Inhibition of human serum AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50022775((m-Hydroxyphenyl)trimethylammonium dimethylcarbama...)
Affinity DataIC50:  42.1nMAssay Description:Inhibition of human serum AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50022775((m-Hydroxyphenyl)trimethylammonium dimethylcarbama...)
Affinity DataIC50:  45nMAssay Description:Inhibition of human serum AChE by Ellman colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049130(5-Isopropyl-2-propyl-3-[2'-(1H-tetrazol-5-yl)-biph...)
Affinity DataIC50:  46nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Mysore

Curated by ChEMBL
LigandPNGBDBM50022775((m-Hydroxyphenyl)trimethylammonium dimethylcarbama...)
Affinity DataIC50:  47.5nMAssay Description:Inhibition of electric eel AChE by Ellman colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50049113(5-Isopropenyl-2-propyl-3-[2'-(2H-tetrazol-5-yl)-bi...)
Affinity DataIC50:  50nMAssay Description:In vitro for inhibition of [125I]-angiotensin II (0.1 nM) binding to angiotensin II receptor type 1 in membrane fractions of bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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