Compile Data Set for Download or QSAR
maximum 50k data
Found 49 with Last Name = 'salvesen' and Initial = 'gs'
TargetCathepsin B(Rattus norvegicus)
Stanford University

LigandPNGBDBM36331(Ac-YFR-AMOK 10b)
Affinity DataIC50:  7.30nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Rattus norvegicus)
Stanford University

LigandPNGBDBM36328(Z-FR-AMOK 9b)
Affinity DataIC50:  15nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Homo sapiens (Human))
School Of Chemistry And Biochemistry And The Parker H. Petit Institute For Bioengineering And Bioscience

Curated by ChEMBL
LigandPNGBDBM50143613((E)-3-{(S)-N'-[(S)-2-((S)-2-Benzyloxycarbonylamino...)
Affinity DataIC50:  31nMAssay Description:Inhibitory concentration of the compound was evaluated for Irreversible Inhibition of S. mansoni LegumainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Homo sapiens (Human))
School Of Chemistry And Biochemistry And The Parker H. Petit Institute For Bioengineering And Bioscience

Curated by ChEMBL
LigandPNGBDBM50143614((E)-3-{(S)-N'-[(S)-2-((S)-2-Benzyloxycarbonylamino...)
Affinity DataIC50:  38nMAssay Description:Inhibitory concentration of the compound was evaluated for Irreversible Inhibition of S. mansoni LegumainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Homo sapiens (Human))
School Of Chemistry And Biochemistry And The Parker H. Petit Institute For Bioengineering And Bioscience

Curated by ChEMBL
LigandPNGBDBM50143612((S)-N'-[(S)-2-((S)-2-Benzyloxycarbonylamino-propio...)
Affinity DataIC50:  55nMAssay Description:Inhibitory concentration of the compound was evaluated for Irreversible Inhibition of S. mansoni LegumainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Rattus norvegicus)
Stanford University

LigandPNGBDBM36327(Z-FG-AOMK 9a)
Affinity DataIC50:  120nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Rattus norvegicus)
Stanford University

LigandPNGBDBM36330(AC-YFG-AMOK 10a)
Affinity DataIC50:  220nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81515(VEA-499)
Affinity DataIC50:  250nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81516(VEA-500)
Affinity DataIC50:  860nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Rattus norvegicus)
Stanford University

LigandPNGBDBM36329(Z-LG-AOMK 9c)
Affinity DataIC50:  920nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Homo sapiens (Human))
School Of Chemistry And Biochemistry And The Parker H. Petit Institute For Bioengineering And Bioscience

Curated by ChEMBL
LigandPNGBDBM50292159((S)-N'-[(S)-2-((S)-2-Benzyloxycarbonylamino-propio...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory concentration of the compound was evaluated for irreversible inhibition of S. mansoni LegumainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Rattus norvegicus)
Stanford University

LigandPNGBDBM36325(Cathepsin Inhibitor III)
Affinity DataIC50:  1.20E+3nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin Z(Rattus norvegicus)
Stanford University

LigandPNGBDBM36325(Cathepsin Inhibitor III)
Affinity DataIC50:  1.50E+3nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81515(VEA-499)
Affinity DataIC50:  3.60E+3nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81511(VEA-260)
Affinity DataIC50:  3.70E+3nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 6(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81517(VEA-561)
Affinity DataIC50:  4.20E+3nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 7(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81517(VEA-561)
Affinity DataIC50:  4.30E+3nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin Z(Rattus norvegicus)
Stanford University

LigandPNGBDBM36331(Ac-YFR-AMOK 10b)
Affinity DataIC50:  4.70E+3nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81517(VEA-561)
Affinity DataIC50:  5.70E+3nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPro-cathepsin H(Rattus norvegicus)
Stanford University

LigandPNGBDBM36325(Cathepsin Inhibitor III)
Affinity DataIC50:  6.60E+3nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81510(JCP-666)
Affinity DataIC50:  7.00E+3nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81511(VEA-260)
Affinity DataIC50:  7.10E+3nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPro-cathepsin H(Rattus norvegicus)
Stanford University

LigandPNGBDBM36330(AC-YFG-AMOK 10a)
Affinity DataIC50:  7.90E+3nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPro-cathepsin H(Rattus norvegicus)
Stanford University

LigandPNGBDBM36329(Z-LG-AOMK 9c)
Affinity DataIC50:  7.90E+3nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81513(VEA-422)
Affinity DataIC50:  1.04E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPro-cathepsin H(Rattus norvegicus)
Stanford University

LigandPNGBDBM36331(Ac-YFR-AMOK 10b)
Affinity DataIC50:  1.20E+4nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81512(VEA-417)
Affinity DataIC50:  1.31E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81514(VEA-401)
Affinity DataIC50:  1.34E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81510(JCP-666)
Affinity DataIC50:  1.38E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81516(VEA-500)
Affinity DataIC50: >2.00E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 7(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81514(VEA-401)
Affinity DataIC50: >2.00E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81513(VEA-422)
Affinity DataIC50:  2.24E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81514(VEA-401)
Affinity DataIC50:  2.31E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81517(VEA-561)
Affinity DataIC50: >2.50E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 1(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81512(VEA-417)
Affinity DataIC50:  3.25E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 7(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81511(VEA-260)
Affinity DataIC50:  3.65E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin Z(Rattus norvegicus)
Stanford University

LigandPNGBDBM36330(AC-YFG-AMOK 10a)
Affinity DataIC50:  3.90E+4nMpH: 5.5 T: 2°CAssay Description:Protease enzyme inhibition assay targeting diverse member of the cysteine protease families:cathepsin B, Z, and HMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 6(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81514(VEA-401)
Affinity DataIC50: >4.00E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 6(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81516(VEA-500)
Affinity DataIC50: >4.00E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 6(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81515(VEA-499)
Affinity DataIC50: >6.00E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 7(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81510(JCP-666)
Affinity DataIC50: >7.00E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 7(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81513(VEA-422)
Affinity DataIC50: >7.00E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 7(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81512(VEA-417)
Affinity DataIC50: >7.00E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 6(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81511(VEA-260)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 6(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81510(JCP-666)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 6(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81512(VEA-417)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 7(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81515(VEA-499)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 7(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81516(VEA-500)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 6(Homo sapiens (Human))
Stanford University

LigandPNGBDBM81513(VEA-422)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed