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Found 90 with Last Name = 'sampe' and Initial = 'r'
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50106301(CHEMBL3598140)
Affinity DataIC50:  1.30nMAssay Description:Allosteric inverse agonist activity at 2-chloro-5-nitro-N-(2-(trifluoromethyl)phenyl)benzamide-ligated recombinant human N-terminal His6-tagged RORga...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50106301(CHEMBL3598140)
Affinity DataIC50:  5.5nMAssay Description:Allosteric inverse agonist activity at 2-chloro-5-nitro-N-o-tolylbenzamide-ligated recombinant human N-terminal His6-tagged RORgammat ligand binding ...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50106301(CHEMBL3598140)
Affinity DataIC50:  5.5nMAssay Description:Allosteric inverse agonist activity at 2-chloro-N-(2,6-dimethylphenyl)-5-nitrobenzamide-ligated recombinant human N-terminal His6-tagged RORgammat li...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50106301(CHEMBL3598140)
Affinity DataIC50:  17nMAssay Description:Allosteric inverse agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in Es...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50519883(CHEMBL4522217)
Affinity DataIC50:  40nMAssay Description:Allosteric inverse agonist activity at 2-chloro-N-(2,6-dimethylphenyl)-5-nitrobenzamide-ligated recombinant human N-terminal His6-tagged RORgammat li...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50557589(CHEMBL4791369)
Affinity DataIC50:  67nMAssay Description:Orthosteric inverse agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50519883(CHEMBL4522217)
Affinity DataIC50:  68nMAssay Description:Allosteric inverse agonist activity at 2-chloro-5-nitro-N-(2-(trifluoromethyl)phenyl)benzamide-ligated recombinant human N-terminal His6-tagged RORga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50557584(CHEMBL4799590)
Affinity DataIC50:  77nMAssay Description:Orthosteric inverse agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50519883(CHEMBL4522217)
Affinity DataIC50:  80nMAssay Description:Allosteric inverse agonist activity at 2-chloro-5-nitro-N-o-tolylbenzamide-ligated recombinant human N-terminal His6-tagged RORgammat ligand binding ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50557587(CHEMBL4793754)
Affinity DataIC50:  81nMAssay Description:Orthosteric inverse agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM55936(2-Chloro-5-nitrobenzanilide | 2-chloranyl-5-nitro-...)
Affinity DataIC50:  86nMAssay Description:Orthosteric inverse agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50557590(CHEMBL4790576)
Affinity DataIC50:  89nMAssay Description:Orthosteric inverse agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50557588(CHEMBL4784120)
Affinity DataIC50:  94nMAssay Description:Orthosteric inverse agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50557586(CHEMBL4779012)
Affinity DataIC50:  108nMAssay Description:Orthosteric inverse agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50557585(CHEMBL4740894)
Affinity DataIC50:  122nMAssay Description:Orthosteric inverse agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50557593(CHEMBL229948)
Affinity DataIC50:  131nMAssay Description:Orthosteric inverse agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104684((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104691(CHEMBL423508 | Diazo-[2-(4-hexadecanoyl-3-hydroxy-...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50557592(CHEMBL4791019)
Affinity DataIC50:  404nMAssay Description:Orthosteric inverse agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50519883(CHEMBL4522217)
Affinity DataIC50:  428nMAssay Description:Allosteric inverse agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in Es...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104690((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  520nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104674((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104693(4-Hydroxy-5-hydroxymethyl-3-octadec-9-enoyl-5H-fur...)
Affinity DataIC50:  900nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50557591(CHEMBL4763539)
Affinity DataIC50:  1.08E+3nMAssay Description:Orthosteric inverse agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104677(3-Hexadecanoyl-4-hydroxy-5-methylene-5H-furan-2-on...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104676((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104681(CHEMBL109357 | Methanesulfonic acid 4-hexadecanoyl...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104696(4-Hydroxy-5-hydroxymethyl-2-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104688(4-Hydroxy-5-hydroxymethyl-2-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104697((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104694((R)-4-hydroxy-5-(hydroxymethyl)-3-palmitoylfuran-2...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM46355(DIGOXIN | MLS000069819 | SMR000059217 | US10668094...)
Affinity DataIC50:  2.31E+3nMAssay Description:Orthosteric inverse agonist activity at recombinant human N-terminal His6-tagged RORgammat ligand binding domain (265 to 518 residues) expressed in E...More data for this Ligand-Target Pair
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104692(4-Hydroxy-5-nonyloxycarbonylmethyl-2-oxo-2,5-dihyd...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104700(3-Hexadecanoyl-4-hydroxy-5H-furan-2-one | CHEMBL32...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104703(4-Hydroxy-5-hydroxymethyl-2-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104673(4-Hydroxy-5-hydroxymethyl-2-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104683(3-Hexadecanoyl-4-hydroxy-5-methyl-5H-furan-2-one |...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104684((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory activity against vaccinia VH1-related phosphatase(VHR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104690((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibitory activity against vaccinia VH1-related phosphatase(VHR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104674((4-Hexadecanoyl-3-hydroxy-5-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibitory activity against vaccinia VH1-related phosphatase(VHR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104694((R)-4-hydroxy-5-(hydroxymethyl)-3-palmitoylfuran-2...)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104699(4-Hydroxy-5-methoxycarbonylmethyl-2-oxo-2,5-dihydr...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM-phase inducer phosphatase 2(Mus musculus)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104686(4-Hydroxy-5-hydroxymethyl-2-oxo-2,5-dihydro-furan-...)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibitory activity against cell division cycle 25BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104681(CHEMBL109357 | Methanesulfonic acid 4-hexadecanoyl...)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibitory activity against vaccinia VH1-related phosphatase(VHR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104677(3-Hexadecanoyl-4-hydroxy-5-methylene-5H-furan-2-on...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibitory activity against vaccinia VH1-related phosphatase(VHR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM46355(DIGOXIN | MLS000069819 | SMR000059217 | US10668094...)
Affinity DataIC50: >1.00E+4nMAssay Description:Orthosteric inverse agonist activity at 2-chloro-N-(2,6-dimethylphenyl)-5-nitrobenzamide-ligated recombinant human N-terminal His6-tagged RORgammat l...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM46355(DIGOXIN | MLS000069819 | SMR000059217 | US10668094...)
Affinity DataIC50: >1.00E+4nMAssay Description:Orthosteric inverse agonist activity at 2-chloro-5-nitro-N-(2-(trifluoromethyl)phenyl)benzamide-ligated recombinant human N-terminal His6-tagged RORg...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM46355(DIGOXIN | MLS000069819 | SMR000059217 | US10668094...)
Affinity DataIC50: >1.00E+4nMAssay Description:Orthosteric inverse agonist activity at 2-chloro-5-nitro-N-o-tolylbenzamide-ligated recombinant human N-terminal His6-tagged RORgammat ligand binding...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104683(3-Hexadecanoyl-4-hydroxy-5-methyl-5H-furan-2-one |...)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibitory activity against vaccinia VH1-related phosphatase(VHR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50104699(4-Hydroxy-5-methoxycarbonylmethyl-2-oxo-2,5-dihydr...)
Affinity DataIC50:  1.11E+4nMAssay Description:Inhibitory activity against vaccinia VH1-related phosphatase(VHR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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