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Found 53 with Last Name = 'sattler' and Initial = 'i'
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50080764((S)-2-({5-[(Benzyl-pyridin-3-yl-amino)-methyl]-2'-...)
Affinity DataIC50:  0.100nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50067563((S)-2-{[2'-Methyl-5-(pyridin-3-yloxymethyl)-biphen...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50072626((S)-2-[2-({(S)-2-[2-(4-Cyano-benzylsulfanyl)-acety...)
Affinity DataIC50:  5.40nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50104054(4-Methylsulfanyl-2-{[5-(5-phenyl-furan-2-ylmethoxy...)
Affinity DataIC50:  6nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50104052(2-{2-[(2-{2-[1-(4-Cyano-benzyl)-4,5-dihydro-1H-imi...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50104047((E)-N-[3-Benzoyl-4-(2-p-tolyl-acetylamino)-phenyl]...)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103281(1-(3-Benzoyl-4-diphenylacetylamino-phenylcarbamoyl...)
Affinity DataIC50:  36nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103269(1-{3-Benzoyl-4-[2-(4-bromo-phenyl)-acetylamino]-ph...)
Affinity DataIC50:  76nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103285(1-[3-Benzoyl-4-(2-p-tolyl-acetylamino)-phenylcarba...)
Affinity DataIC50:  77nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103271(1-(3-Benzoyl-4-phenylmethanesulfonylamino-phenylca...)
Affinity DataIC50:  85nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103280(1-(3-Benzoyl-4-p-tolylmethanesulfonylamino-phenylc...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103262(1-{3-Benzoyl-4-[2-(4-chloro-phenyl)-acetylamino]-p...)
Affinity DataIC50:  105nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103274(1-{3-Benzoyl-4-[2-(4-nitro-phenyl)-acetylamino]-ph...)
Affinity DataIC50:  115nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103261(1-{3-Benzoyl-4-[2-(2,4-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103270(1-{3-Benzoyl-4-[2-(2,6-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  340nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103272(1-[3-Benzoyl-4-(2-naphthalen-1-yl-acetylamino)-phe...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50104050(5-Phenyl-pentanoic acid [3-benzoyl-4-(2-p-tolyl-ac...)
Affinity DataIC50:  390nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103260(1-[3-Benzoyl-4-(2-o-tolyl-acetylamino)-phenylcarba...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103258(1-{3-Benzoyl-4-[2-(2,3-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  420nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50104055(CHEMBL276748 | N-[3-Benzoyl-4-(2-p-tolyl-acetylami...)
Affinity DataIC50:  455nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103277(1-[3-Benzoyl-4-(2-naphthalen-2-yl-acetylamino)-phe...)
Affinity DataIC50:  460nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103284(1-{3-Benzoyl-4-[2-(3,4-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  480nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50104048(CHEMBL106900 | N-[3-Benzoyl-4-(2-p-tolyl-acetylami...)
Affinity DataIC50:  530nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103276(1-{3-Benzoyl-4-[2-(3,5-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  535nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103259(1-[3-Benzoyl-4-(2-m-tolyl-acetylamino)-phenylcarba...)
Affinity DataIC50:  540nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103268(1-{3-Benzoyl-4-[2-(4-methoxy-phenyl)-acetylamino]-...)
Affinity DataIC50:  545nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103257(1-[3-Benzoyl-4-(4-carboxy-butyrylamino)-phenylcarb...)
Affinity DataIC50:  550nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103287(1-(3-Benzoyl-4-phenylacetylamino-phenylcarbamoyl)-...)
Affinity DataIC50:  650nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103278(1-[3-Benzoyl-4-(2-phenyl-propionylamino)-phenylcar...)
Affinity DataIC50:  650nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103266(1-[3-Benzoyl-4-(3-carboxy-propionylamino)-phenylca...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103283(1-{3-Benzoyl-4-[2-(4-trifluoromethyl-phenyl)-acety...)
Affinity DataIC50:  725nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50104053(CHEMBL329401 | N-[3-Benzoyl-4-(2-p-tolyl-acetylami...)
Affinity DataIC50:  925nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50104049(6-Phenyl-hexanoic acid [3-benzoyl-4-(2-p-tolyl-ace...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103282(1-[3-Benzoyl-4-(3-phenyl-propionylamino)-phenylcar...)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103256(1-[3-Benzoyl-4-(2-oxo-2-phenyl-acetylamino)-phenyl...)
Affinity DataIC50:  1.42E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103263(1-[3-Benzoyl-4-(3-methoxycarbonyl-propionylamino)-...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103267(1-[3-Benzoyl-4-(2-biphenyl-4-yl-acetylamino)-pheny...)
Affinity DataIC50:  1.98E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50104046(CHEMBL104134 | N-(2-Benzoyl-4-phenylacetylamino-ph...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50096841(CHEMBL91489 | N-[3-Benzoyl-4-(2-p-tolyl-acetylamin...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103264(1-[3-Benzoyl-4-(4-methoxycarbonyl-butyrylamino)-ph...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103273(1-{3-Benzoyl-4-[2-(2,5-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103265(1-{3-Benzoyl-4-[(naphthalene-1-carbonyl)-amino]-ph...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103286(1-(3-Benzoyl-4-benzoylamino-phenylcarbamoyl)-2-mer...)
Affinity DataIC50:  4.78E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50104057(CHEMBL106052 | N-[3-Benzoyl-4-(2-p-tolyl-acetylami...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50104056(CHEMBL90987 | N-[3-Benzoyl-4-(2-p-tolyl-acetylamin...)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103275(1-(4-Acetylamino-3-benzoyl-phenylcarbamoyl)-2-merc...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50103279(1-[3-Benzoyl-4-(3,5,5-trimethyl-hexanoylamino)-phe...)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50104051(CHEMBL105738 | N-[3-Benzoyl-4-(2-p-tolyl-acetylami...)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Leibniz-Institute For Natural Product Research And Infection Biology

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human recombinant DYRK1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
Philipps-UniversitäT Marburg

Curated by ChEMBL
LigandPNGBDBM50104045(CHEMBL106252 | N-[3-Benzoyl-4-(2-p-tolyl-acetylami...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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