TargetKynurenine/alpha-aminoadipate aminotransferase, mitochondrial(Homo sapiens (Human))
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
Affinity DataIC50: 910nMAssay Description:Inhibition of human recombinant MBP-KAT2 expressed in HEK293 cells assessed as conversion of L-kynurenine to kynurenic acid after 1 hrMore data for this Ligand-Target Pair
TargetKynurenine/alpha-aminoadipate aminotransferase, mitochondrial(Rattus norvegicus)
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat brain KAT2More data for this Ligand-Target Pair
TargetKynurenine/alpha-aminoadipate aminotransferase, mitochondrial(Homo sapiens (Human))
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of KAT2 in human prefrontal cortex homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of 3-HAO in human brain homogenates using [1-14C]-3-HANA as substrate assessed as [14C]-QUIN production after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
TargetKynurenine/alpha-aminoadipate aminotransferase, mitochondrial(Homo sapiens (Human))
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human recombinant MBP-KAT2 expressed in HEK293 cells assessed as conversion of L-kynurenine to kynurenic acid after 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of 3-HAO in Sprague-Dawley rat brain homogenates using [1-14C]-3-HANA as substrate assessed as [14C]-QUIN production after 1 hr by liquid ...More data for this Ligand-Target Pair
TargetKynurenine--oxoglutarate transaminase 1(Homo sapiens (Human))
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant MBP-KAT1 expressed in HEK293 cells assessed as conversion of L-kynurenine to kynurenic acid after 1 hrMore data for this Ligand-Target Pair
TargetKynurenine--oxoglutarate transaminase 1(Homo sapiens (Human))
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
University Of Piemonte Orientale Amedeo Avogadro
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of KAT1 in human prefrontal cortex homogenatesMore data for this Ligand-Target Pair