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Found 102 with Last Name = 'seto' and Initial = 'ct'
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50102186((Difluoro-phenyl-methyl)-phosphonic acid | CHEMBL5...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibitory activity against Yersinia Protein-tyrosine phosphatase 1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50081422(2-((R)-3-{(R)-3-[(S)-2-((S)-Benzyloxycarbonylamino...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibitory activity of the compound against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50081422(2-((R)-3-{(R)-3-[(S)-2-((S)-Benzyloxycarbonylamino...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibitory activity of the compound against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50079381((R)-2-Amino-3-methyl-pentanoic acid {(S)-1-[(6-ami...)
Affinity DataKi:  5.00E+4nMAssay Description:Compound was evaluated for its binding affinity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50102187(CHEMBL299446 | Furan-2-yl-oxo-acetic acid)
Affinity DataKi:  7.90E+4nMAssay Description:Inhibitory activity against Yersinia Protein-tyrosine phosphatase 1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50081425(2-((R)-3-{(R)-3-[(S)-2-Benzyloxycarbonylamino-3-(1...)
Affinity DataKi:  1.50E+5nMAssay Description:Inhibitory activity of the compound against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50081425(2-((R)-3-{(R)-3-[(S)-2-Benzyloxycarbonylamino-3-(1...)
Affinity DataKi:  1.50E+5nMAssay Description:Inhibitory activity of the compound against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50075312((Difluoro-naphthalen-2-yl-methyl)-phosphonic acid ...)
Affinity DataKi:  1.79E+5nMAssay Description:Inhibitory activity against Yersinia Protein-tyrosine phosphatase 1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Brown University

Curated by ChEMBL
LigandPNGBDBM50081425(2-((R)-3-{(R)-3-[(S)-2-Benzyloxycarbonylamino-3-(1...)
Affinity DataKi:  2.50E+5nMAssay Description:Inhibitory activity of the compound against papainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50462601(CHEMBL4250607)
Affinity DataKi:  2.75E+5nMAssay Description:Irreversible inhibition of human arginase 1 using thioarginine as substrate measured up to 360 mins by UV micro plate methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50462601(CHEMBL4250607)
Affinity DataKi:  3.22E+5nMAssay Description:Irreversible inhibition of human arginase 2 using thioarginine as substrate measured up to 360 mins by UV micro plate methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Brown University

Curated by ChEMBL
LigandPNGBDBM50081422(2-((R)-3-{(R)-3-[(S)-2-((S)-Benzyloxycarbonylamino...)
Affinity DataKi:  3.80E+5nMAssay Description:Inhibitory activity of the compound against papainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50462600(CHEMBL4238387)
Affinity DataKi:  3.82E+5nMAssay Description:Irreversible inhibition of human arginase 1 using thioarginine as substrate measured up to 360 mins by UV micro plate methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50079380(3-[Bis-(6-amino-hexyl)-amino]-tetrahydro-thiopyran...)
Affinity DataKi:  4.00E+5nMAssay Description:Compound was evaluated for its binding affinity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50081424(2-((R)-3-{(R)-3-[(S)-2-((S)-Benzyloxycarbonylamino...)
Affinity DataKi:  4.20E+5nMAssay Description:Inhibitory activity of the compound against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50462600(CHEMBL4238387)
Affinity DataKi:  4.37E+5nMAssay Description:Irreversible inhibition of human arginase 2 using thioarginine as substrate measured up to 360 mins by UV micro plate methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Brown University

Curated by ChEMBL
LigandPNGBDBM50081424(2-((R)-3-{(R)-3-[(S)-2-((S)-Benzyloxycarbonylamino...)
Affinity DataKi:  4.90E+5nMAssay Description:Inhibitory activity of the compound against papainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50079383((R)-2-Amino-3-methyl-pentanoic acid {(S)-1-[(6-ami...)
Affinity DataKi:  5.20E+5nMAssay Description:Compound was evaluated for its binding affinity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50079381((R)-2-Amino-3-methyl-pentanoic acid {(S)-1-[(6-ami...)
Affinity DataKi:  6.30E+5nMAssay Description:Compound was evaluated for its binding affinity against kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50079381((R)-2-Amino-3-methyl-pentanoic acid {(S)-1-[(6-ami...)
Affinity DataKi:  6.30E+5nMAssay Description:Compound was evaluated for its binding affinity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50079381((R)-2-Amino-3-methyl-pentanoic acid {(S)-1-[(6-ami...)
Affinity DataKi:  6.30E+5nMAssay Description:Compound was evaluated for its binding affinity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50079381((R)-2-Amino-3-methyl-pentanoic acid {(S)-1-[(6-ami...)
Affinity DataKi:  6.30E+5nMAssay Description:Compound was evaluated for its binding affinity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Brown University

Curated by ChEMBL
LigandPNGBDBM50081423(2-{(R)-3-[(R)-3-((S)-2-Benzyloxycarbonylamino-3-ph...)
Affinity DataKi:  8.70E+5nMAssay Description:Inhibitory activity of the compound against papainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50081423(2-{(R)-3-[(R)-3-((S)-2-Benzyloxycarbonylamino-3-ph...)
Affinity DataKi:  1.10E+6nMAssay Description:Inhibitory activity of the compound against Cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50079380(3-[Bis-(6-amino-hexyl)-amino]-tetrahydro-thiopyran...)
Affinity DataKi:  1.40E+6nMAssay Description:Compound was evaluated for its binding affinity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50081423(2-{(R)-3-[(R)-3-((S)-2-Benzyloxycarbonylamino-3-ph...)
Affinity DataKi:  3.00E+6nMAssay Description:Inhibitory activity of the compound against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50079380(3-[Bis-(6-amino-hexyl)-amino]-tetrahydro-thiopyran...)
Affinity DataKi: >1.00E+7nMAssay Description:Compound was evaluated for its binding affinity against kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50079380(3-[Bis-(6-amino-hexyl)-amino]-tetrahydro-thiopyran...)
Affinity DataKi: >1.00E+7nMAssay Description:Compound was evaluated for its binding affinity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50079382((R)-2-Amino-3-methyl-pentanoic acid [(S)-1-(4-oxo-...)
Affinity DataKi:  1.60E+7nMAssay Description:Compound was evaluated for its binding affinity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50079382((R)-2-Amino-3-methyl-pentanoic acid [(S)-1-(4-oxo-...)
Affinity DataKi:  1.60E+7nMAssay Description:Compound was evaluated for its binding affinity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326496(4, 4'-[[2-[[(4-(4-Trifluoromethylthio)phenoxy phen...)
Affinity DataIC50:  30nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326497(4, 4'-[[2-[[(4-(4-Trifluoromethylthio)phenoxypheny...)
Affinity DataIC50:  50nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326498(4, 4'-[[2-[[(4-(4-Ethyl)phenoxyphenyl)amino]carbon...)
Affinity DataIC50:  70nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326499(4, 4'-[[2-[[(4-(4-n-Hexyl)phenoxyphenyl)amino]carb...)
Affinity DataIC50:  90nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326500(2,2'-(4,4'-(2-(3-(benzyloxy)phenylcarbamoyl)-1,4-p...)
Affinity DataIC50:  100nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326502(2,2'-(4,4'-(2-(4-(4-fluorophenoxy)phenylcarbamoyl)...)
Affinity DataIC50:  110nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326501(2,2'-(4,4'-(2-(4-(4-(methylthio)phenoxy)phenylcarb...)
Affinity DataIC50:  110nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326503(2,2'-(4,4'-(2-(4-(p-tolyloxy)phenylcarbamoyl)-1,4-...)
Affinity DataIC50:  190nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326504(2,2'-(4,4'-(2-(4-(4-butylphenoxy)phenylcarbamoyl)-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326505(2,2'-(4,4'-(2-(4-(3,4-dichlorophenoxy)phenylcarbam...)
Affinity DataIC50:  210nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50326496(4, 4'-[[2-[[(4-(4-Trifluoromethylthio)phenoxy phen...)
Affinity DataIC50:  220nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326506(2,2'-(4,4'-(2-(4-(3-chlorophenoxy)phenylcarbamoyl)...)
Affinity DataIC50:  220nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326507(2,2'-(4,4'-(2-(4-(o-tolyloxy)phenylcarbamoyl)-1,4-...)
Affinity DataIC50:  230nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326508(2,2'-(4,4'-(2-(4-phenoxyphenylcarbamoyl)-1,4-pheny...)
Affinity DataIC50:  240nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50326498(4, 4'-[[2-[[(4-(4-Ethyl)phenoxyphenyl)amino]carbon...)
Affinity DataIC50:  490nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase C(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50118096(2,2'-(4,4'-(1,4-phenylenebis(methylene))bis(oxy)bi...)
Affinity DataIC50:  700nMAssay Description:Concentration required for 50% Inhibition of activity against Yersinia Protein-tyrosine phosphataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326509(2,2'-(4,4'-(2-(4-(4-isopropylphenoxy)phenylcarbamo...)
Affinity DataIC50:  800nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326510(2,2'-(4,4'-(2-(4-(2,4-difluorophenoxy)phenylcarbam...)
Affinity DataIC50:  910nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Brown University

Curated by ChEMBL
LigandPNGBDBM50326511(2,2'-(4,4'-(2-(4-(4-methoxyphenoxy)phenylcarbamoyl...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Brown University

Curated by ChEMBL
LigandPNGBDBM50326499(4, 4'-[[2-[[(4-(4-n-Hexyl)phenoxyphenyl)amino]carb...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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