TargetLeukotriene B4 receptor 2(Homo sapiens (Human))
The University of Tokyo
Curated by PDSP Ki Database
The University of Tokyo
Curated by PDSP Ki Database
TargetLeukotriene B4 receptor 2(Homo sapiens (Human))
The University of Tokyo
Curated by PDSP Ki Database
The University of Tokyo
Curated by PDSP Ki Database
Affinity DataKi: 90nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 2(Homo sapiens (Human))
The University of Tokyo
Curated by PDSP Ki Database
The University of Tokyo
Curated by PDSP Ki Database
Affinity DataKi: 130nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 2(Homo sapiens (Human))
The University of Tokyo
Curated by PDSP Ki Database
The University of Tokyo
Curated by PDSP Ki Database
Affinity DataKi: 470nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
Affinity DataKi: 580nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 610nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 790nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
Affinity DataKi: 880nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 940nM ΔG°: -35.8kJ/molepH: 4.5 T: 2°CAssay Description:β-Gal activity was measured by using 4-methylumbelliferyll-β-D-galactopyranoside in buffer B (0.15 M sodium citrate, pH 4.5, and 0.2 M NaCl...More data for this Ligand-Target Pair
Affinity DataKi: 990nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nM ΔG°: -35.4kJ/molepH: 4.5 T: 2°CAssay Description:β-Gal activity was measured by using 4-methylumbelliferyll-β-D-galactopyranoside in buffer B (0.15 M sodium citrate, pH 4.5, and 0.2 M NaCl...More data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 2(Homo sapiens (Human))
The University of Tokyo
Curated by PDSP Ki Database
The University of Tokyo
Curated by PDSP Ki Database
Affinity DataKi: 1.20E+3nM ΔG°: -35.2kJ/molepH: 4.5 T: 2°CAssay Description:β-Gal activity was measured by using 4-methylumbelliferyll-β-D-galactopyranoside in buffer B (0.15 M sodium citrate, pH 4.5, and 0.2 M NaCl...More data for this Ligand-Target Pair
Affinity DataKi: 1.46E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
Affinity DataKi: 1.62E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.67E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.26E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 7.84E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 8.64E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 9.90E+3nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
Affinity DataKi: 1.26E+4nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
Affinity DataKi: 1.26E+4nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (guinea pig) transgenic mouse muscle membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.47E+4nM ΔG°: -25.8kJ/molepH: 4.5 T: 2°CAssay Description:β-Gal activity was measured by using 4-methylumbelliferyll-β-D-galactopyranoside in buffer B (0.15 M sodium citrate, pH 4.5, and 0.2 M NaCl...More data for this Ligand-Target Pair
Affinity DataKi: 4.90E+4nM ΔG°: -25.6kJ/molepH: 4.5 T: 2°CAssay Description:β-Gal activity was measured by using 4-methylumbelliferyll-β-D-galactopyranoside in buffer B (0.15 M sodium citrate, pH 4.5, and 0.2 M NaCl...More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]-WEB 2086 from Platelet activating factor receptor (PAF)More data for this Ligand-Target Pair
Affinity DataKi: 5.33E+4nM ΔG°: -25.4kJ/molepH: 4.5 T: 2°CAssay Description:β-Gal activity was measured by using 4-methylumbelliferyll-β-D-galactopyranoside in buffer B (0.15 M sodium citrate, pH 4.5, and 0.2 M NaCl...More data for this Ligand-Target Pair