Affinity DataKi: 9nMAssay Description:Inhibition of CCR3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Inhibition of CCR3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 520nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 7.30E+3nMAssay Description:Inhibition of xanthine oxidase (unknown origin)More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Punjabi University
Curated by ChEMBL
Punjabi University
Curated by ChEMBL
Affinity DataKi: 8.10E+4nMAssay Description:Inhibition of forskolin-stimulated CFTR (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.540nMAssay Description:Inhibition of human CDK1 using Biotinaminohexyl-Ala-Arg-Arg-Pro-Met-Ser-Pro-Lys-LysLys-Ala-CONH2 peptide as substrate incubated for 20 to 30 mins by ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.601nMAssay Description:Inhibition of mouse macrophage COX2More data for this Ligand-Target Pair
Affinity DataIC50: 0.701nMAssay Description:Inhibition of mouse macrophage COX2More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of mouse macrophage COX2More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of bovine erythrocyte AchE using acetylthiocholine iodide as substrate after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of bovine erythrocyte AchE using acetylthiocholine iodide as substrate after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of mouse macrophage COX2More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Reversible inhibition of NH2-terminal 6His-tagged FAK catalytic domain (410 to 689 residues) (unknown origin) expressed in Sf9 insect cells using p(G...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of mouse macrophage COX2More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of mouse macrophage COX2More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of mouse macrophage COX2More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2 (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of mouse macrophage COX2More data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of mouse macrophage COX2More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of CDK2 (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Inhibition of mouse macrophage COX2More data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Inhibition of mouse macrophage COX2More data for this Ligand-Target Pair
Affinity DataIC50: 4.51nMAssay Description:Inhibition of mouse macrophage COX2More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of mouse macrophage COX2More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of human Syk expressed in Kluyveromyces lactis using Biot-(BA)3-DEEYEIP-NH2 as substrate in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of spleen tyrosine kinase (unknown origin)More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Punjabi University
Curated by ChEMBL
Punjabi University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of c-Kit by HTRF methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Punjabi University
Curated by ChEMBL
Punjabi University
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of c-Kit by HTRF methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Punjabi University
Curated by ChEMBL
Punjabi University
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of GnRH receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of TrkA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 7.70nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of TrkA (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 8nMAssay Description:Inhibition of spleen tyrosine kinase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of cRAF1 (unknown origin)More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Punjabi University
Curated by ChEMBL
Punjabi University
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of c-Kit by HTRF methodMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Punjabi University
Curated by ChEMBL
Punjabi University
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant GST-tagged PI3Kgamma incubated for 180 mins using [33P]gamma-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.10nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair