Affinity DataKi: 1.20nMAssay Description:Dissplacement of [3H]-CGS- from Adenosine A2a receptor of rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 10.4nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 13.7nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 13.7nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 18.3nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 30.4nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 42.4nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 61.2nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 116nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 121nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 236nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 280nMAssay Description:Binding affinity towards dopamine transporter using [3H]- mazindol as radioligand in rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 320nMAssay Description:Inhibition of high affinity uptake of [3H]dopamine into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 540nMAssay Description:Binding affinity towards dopamine transporter using [3H]- mazindol as radioligand in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 651nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 706nMAssay Description:Dissplacement of [3H]-CGS- from Adenosine A2a receptor of rat striatal homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of high affinity uptake of [3H]dopamine into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 4.20E+3nMAssay Description:Binding affinity towards dopamine transporter using [3H]- mazindol as radioligand in rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 4.20E+3nMAssay Description:Binding affinity towards dopamine transporter using [3H]- mazindol as radioligand in rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 8.50E+3nMAssay Description:Inhibition of high affinity uptake of [3H]dopamine into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 8.50E+3nMAssay Description:Inhibition of high affinity uptake of [3H]dopamine into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.04E+4nMAssay Description:Binding affinity towards dopamine transporter using [3H]- mazindol as radioligand in rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.38E+4nMAssay Description:Inhibition of high affinity uptake of [3H]dopamine into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.30E+4nMAssay Description:Inhibition of high affinity uptake of [3H]dopamine into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.94E+4nMAssay Description:Binding affinity towards dopamine transporter using [3H]- mazindol as radioligand in rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.94E+4nMAssay Description:Binding affinity towards dopamine transporter using [3H]- mazindol as radioligand in rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.40E+4nMAssay Description:Binding affinity towards dopamine transporter using [3H]- mazindol as radioligand in rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.50E+4nMAssay Description:Inhibition of high affinity uptake of [3H]dopamine into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.80E+4nMAssay Description:Inhibition of high affinity uptake of [3H]dopamine into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 4.77E+4nMAssay Description:Binding affinity towards dopamine transporter using [3H]- mazindol as radioligand in rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 4.77E+4nMAssay Description:Inhibition of high affinity uptake of [3H]dopamine into striatal nerve endings (synaptosomes)More data for this Ligand-Target Pair