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Found 89 with Last Name = 'stephenson' and Initial = 'pt'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50316213(4-((3-(2-(6-(2,2-diphenylethylamino)-9-((2R,3R,4S,...)
Affinity DataIC50:  0.400nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50276291(CHEMBL472464 | N-benzyl-N-(1'-(2,6-dimethylbenzoyl...)
Affinity DataIC50:  0.5nMAssay Description:Antagonist activity at human recombinant CCR5 expressed in human HeLa-P4 cells assessed as inhibition of human HeLa-P4 cells binding to HIV1 gp160 ex...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50276259(CHEMBL481068 | exo-N-benzyl-N-((R)-1-(8-(2,6-dimet...)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at human recombinant CCR5 expressed in human HeLa-P4 cells assessed as inhibition of human HeLa-P4 cells binding to HIV1 gp160 ex...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50276260((R)-N-benzyl-N-(1-(1-(2,6-dimethylbenzoyl)piperidi...)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at human recombinant CCR5 expressed in human HeLa-P4 cells assessed as inhibition of human HeLa-P4 cells binding to HIV1 gp160 ex...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50276290(CHEMBL472260 | N-benzyl-N-(1'-(2,6-dimethylbenzoyl...)
Affinity DataIC50:  3nMAssay Description:Antagonist activity at human recombinant CCR5 expressed in human HeLa-P4 cells assessed as inhibition of human HeLa-P4 cells binding to HIV1 gp160 ex...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50316210(6-(2,2-diphenylethylamino)-9-((2R,3R,4S,5S)-5-(eth...)
Affinity DataIC50:  4nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50316212(6-(2,2-diphenylethylamino)-9-((2R,3R,4S,5S)-5-(eth...)
Affinity DataIC50:  4nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50316211(CHEMBL1096895 | N-(2-(3-(4-((diethylamino)methyl)b...)
Affinity DataIC50:  5nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50316205(CHEMBL1096889 | N-(2-(3-(2-(diisopropylamino)ethyl...)
Affinity DataIC50:  5nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50316202(6-(2,2-diphenylethylamino)-9-((2R,3R,4S,5S)-5-(eth...)
Affinity DataIC50:  5nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50233816((2S,3S,4R,5R)-5-(2-((3-(2-(cyclopentyl(isopropyl)a...)
Affinity DataIC50:  6nMAssay Description:Agonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50316209(CHEMBL1096893 | N-(2-(3-benzylureido)ethyl)-6-(2,2...)
Affinity DataIC50:  6nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50233816((2S,3S,4R,5R)-5-(2-((3-(2-(cyclopentyl(isopropyl)a...)
Affinity DataIC50:  6nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50316204(CHEMBL1096888 | N-(2-(3-(2-(cyclopentyl(isopropyl)...)
Affinity DataIC50:  7nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50276260((R)-N-benzyl-N-(1-(1-(2,6-dimethylbenzoyl)piperidi...)
Affinity DataIC50:  8nMAssay Description:Displacement of [125]Mip1beta form CCR5 receptor (unknown origin) expressed in MIP34.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50372023(CHEMBL403478)
Affinity DataIC50:  9nMAssay Description:Agonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50316206(CHEMBL1096890 | N-(2-(3-(2-(3,4-dihydroisoquinolin...)
Affinity DataIC50:  10nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50316208(6-(2,2-diphenylethylamino)-9-((2R,3R,4S,5S)-5-(eth...)
Affinity DataIC50:  10nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50372024(CHEMBL257213)
Affinity DataIC50:  11nMAssay Description:Agonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50233809((2S,3S,4R,5R)-5-(6-(2,2-diphenylethylamino)-2-((3-...)
Affinity DataIC50:  17nMAssay Description:Agonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50233809((2S,3S,4R,5R)-5-(6-(2,2-diphenylethylamino)-2-((3-...)
Affinity DataIC50:  17nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50276623((4-((1-benzhydrylazetidin-3-yl)(methyl)amino)piper...)
Affinity DataIC50:  24nMAssay Description:Antagonist activity at human recombinant CCR5 expressed in human HeLa-P4 cells assessed as inhibition of human HeLa-P4 cells binding to HIV1 gp160 ex...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50372026(CHEMBL257429)
Affinity DataIC50:  28nMAssay Description:Agonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50372029(CHEMBL256489)
Affinity DataIC50:  33nMAssay Description:Agonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50276672((4-(3-benzhydryl-3,8-diazabicyclo[3.2.1]octan-8-yl...)
Affinity DataIC50:  41nMAssay Description:Antagonist activity at human recombinant CCR5 expressed in human HeLa-P4 cells assessed as inhibition of human HeLa-P4 cells binding to HIV1 gp160 ex...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50316203(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)te...)
Affinity DataIC50:  45nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50276793(CHEMBL459986 | rac-N-(2-(3-(2,2-diphenylethyl)pipe...)
Affinity DataIC50:  56nMAssay Description:Antagonist activity at human recombinant CCR5 expressed in human HeLa-P4 cells assessed as inhibition of human HeLa-P4 cells binding to HIV1 gp160 ex...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50372027(CHEMBL270378)
Affinity DataIC50:  60nMAssay Description:Agonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50233810(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-t...)
Affinity DataIC50:  65nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50233810(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-t...)
Affinity DataIC50:  65nMAssay Description:Agonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50372025(CHEMBL401571)
Affinity DataIC50:  100nMAssay Description:Agonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50276792((3-((1-benzhydrylpiperidin-4-yl)(methyl)amino)azet...)
Affinity DataIC50:  102nMAssay Description:Antagonist activity at human recombinant CCR5 expressed in human HeLa-P4 cells assessed as inhibition of human HeLa-P4 cells binding to HIV1 gp160 ex...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50276217(CHEMBL471403 | N-((4-benzyl-1'-(2,6-dimethylbenzoy...)
Affinity DataIC50:  145nMAssay Description:Antagonist activity at human recombinant CCR5 expressed in human HeLa-P4 cells assessed as inhibition of human HeLa-P4 cells binding to HIV1 gp160 ex...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050632(8-ETHYL-6-METHOXY-3-METHYL-8H-1,3A,7,8,9-PENTAAZA-...)
Affinity DataIC50:  156nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050632(8-ETHYL-6-METHOXY-3-METHYL-8H-1,3A,7,8,9-PENTAAZA-...)
Affinity DataIC50:  190nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050636(8-Cyclopropyl-4-methyl-8H-1,3a,7,8,9-pentaaza-dibe...)
Affinity DataIC50:  217nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050633(8-Ethyl-4-methyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,...)
Affinity DataIC50:  245nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050628(8-Ethyl-6-methoxy-8H-1,3a,7,8,9-pentaaza-dibenzo[e...)
Affinity DataIC50:  258nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50316207(6-(2,2-diphenylethylamino)-9-((2R,3R,4S,5S)-5-(eth...)
Affinity DataIC50:  305nMAssay Description:Agonist activity at adenosine A2A receptor in fMLP-stimulated human neutrophils assessed as inhibition of superoxide production by colorimetric analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50276671((4-(8-benzhydryl-3,8-diazabicyclo[3.2.1]octan-3-yl...)
Affinity DataIC50:  313nMAssay Description:Antagonist activity at human recombinant CCR5 expressed in human HeLa-P4 cells assessed as inhibition of human HeLa-P4 cells binding to HIV1 gp160 ex...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050640(8-Ethyl-3-methyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,...)
Affinity DataIC50:  425nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050628(8-Ethyl-6-methoxy-8H-1,3a,7,8,9-pentaaza-dibenzo[e...)
Affinity DataIC50:  598nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280306(8-Ethyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,h]azulene...)
Affinity DataIC50:  775nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50372022(CHEMBL404123)
Affinity DataIC50:  1.00E+3nMAssay Description:Agonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50372028(CHEMBL404521)
Affinity DataIC50:  1.01E+3nMAssay Description:Agonist activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050634((8-Ethyl-3-methyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e...)
Affinity DataIC50:  1.10E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50280315(3,8-Diethyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,h]azu...)
Affinity DataIC50:  1.10E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050640(8-Ethyl-3-methyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,...)
Affinity DataIC50:  1.22E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50276261((S)-N-benzyl-N-(1-(1-(2,6-dimethylbenzoyl)piperidi...)
Affinity DataIC50:  1.23E+3nMAssay Description:Antagonist activity at human recombinant CCR5 expressed in human HeLa-P4 cells assessed as inhibition of human HeLa-P4 cells binding to HIV1 gp160 ex...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM1517(2-ethyl-7-methyl-2,4,9,15-tetraazatricyclo[9.4.0.0...)
Affinity DataIC50:  1.50E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
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