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Found 2616 with Last Name = 'stocks' and Initial = 'mj'
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50521218(CHEMBL4434674)
Affinity DataKi:  0.0794nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
TargetP2Y purinoceptor 12(Homo sapiens (Human))TBA
LigandPNGBDBM50167271(CHEMBL3798413)
In DepthDetails
TargetPlasma kallikrein(Homo sapiens (Human))
Kalvista Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM408717( N-[(3-fluoro-4-methoxypyridin-2-yl)methyl]-3-(met...)
Affinity DataKi:  3nMAssay Description:Reversible inhibition of human plasma kallikrein assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429537(CHEMBL2333770)
In DepthDetails PDB3D3D Structure (crystal)
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429541(CHEMBL2333766)
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429548(CHEMBL2333759)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429538(CHEMBL2333767)
Affinity DataKi:  20nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 12(Homo sapiens (Human))TBA
LigandPNGBDBM50268964(CHEMBL502519 | Sodium 1-Amino-4-[4-phenylamino-3-c...)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271558(CHEMBL4082045)
Affinity DataKi:  22nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(2-(4-(2-(5,5-difluoro-7-(thiophen-2-yl)-5H-4-lambda4,5-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazab...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429546(CHEMBL2333761)
Affinity DataKi:  28nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50373303(CHEMBL256141)
Affinity DataKi:  30nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429547(CHEMBL2333760)
Affinity DataKi:  33nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271558(CHEMBL4082045)
Affinity DataKi:  35nMAssay Description:Displacement of N-(2-(3-((7-Chloro-4-(1-methyl-2-oxo-4-thioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-4H-benzo[5,6]cyclohepta[1,2-d]thiazol-2-yl)-amino)pro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271558(CHEMBL4082045)
Affinity DataKi:  42nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429567(CHEMBL2333776)
Affinity DataKi:  47nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271558(CHEMBL4082045)
Affinity DataKi:  48nMAssay Description:Displacement of N-(2-(2-(2-(3-((7-Chloro-4-(1-methyl-2-oxo-4-thioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-4H-benzo[5,6]cyclohepta[1,2-d]thiazol-2-yl)amin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429561(CHEMBL2333353)
Affinity DataKi:  48nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429562(CHEMBL2333352)
Affinity DataKi:  69nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50373324(CHEMBL258406)
Affinity DataKi:  70nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429569(CHEMBL2333774)
Affinity DataKi:  75nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429545(CHEMBL2333762)
Affinity DataKi:  77nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 14(Homo sapiens (Human))TBA
LigandPNGBDBM50614414(CHEMBL5271821)
Affinity DataKi:  80nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271600(CHEMBL4086462)
Affinity DataKi:  83nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthranilate--CoA ligase(Pseudomonas aeruginosa (Gram- Bacteria))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50324670(((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...)
Affinity DataKi:  88nMAssay Description:Inhibition of recombinant Pseudomonas aeruginosa PqsA assessed as decrease in formation of anthranilyl-CoA by spectrophotometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50373323(CHEMBL255306)
Affinity DataKi:  90nMMore data for this Ligand-Target Pair
In DepthDetails
TargetAnthranilate--CoA ligase(Pseudomonas aeruginosa (Gram- Bacteria))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50465699(CHEMBL377483)
Affinity DataKi:  109nMAssay Description:Inhibition of recombinant Pseudomonas aeruginosa PqsA assessed as decrease in formation of anthranilyl-CoA by spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271596(CHEMBL4128126)
Affinity DataKi:  129nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271589(CHEMBL4128024)
Affinity DataKi:  145nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 14(Homo sapiens (Human))TBA
LigandPNGBDBM50343128(2-(benzo[d][1,3]dioxol-5-yl)-N-(3-ethylphenyl)-4-o...)
Affinity DataKi:  160nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429568(CHEMBL2333775)
Affinity DataKi:  171nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429544(CHEMBL2333763)
Affinity DataKi:  172nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429540(CHEMBL2333768)
Affinity DataKi:  175nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271599(CHEMBL4128208)
Affinity DataKi:  275nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429559(CHEMBL2333355)
Affinity DataKi:  313nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271569(CHEMBL4128318)
Affinity DataKi:  398nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50521218(CHEMBL4434674)
Affinity DataKi:  501nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50521218(CHEMBL4434674)
Affinity DataKi:  501nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429565(CHEMBL2333349)
Affinity DataKi:  607nMMore data for this Ligand-Target Pair
In DepthDetails
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50521218(CHEMBL4434674)
Affinity DataKi:  631nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271597(CHEMBL4127983)
Affinity DataKi:  1.55E+3nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429549(CHEMBL2333758)
Affinity DataKi:  2.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50205417(CHEMBL220200 | UTP-gamma-S)
Affinity DataKi:  3.47E+3nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429539(CHEMBL2333769)
Affinity DataKi: >5.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429551(CHEMBL2333757)
Affinity DataKi: >5.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429550(CHEMBL2331579)
Affinity DataKi: >5.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429542(CHEMBL2333765)
Affinity DataKi: >5.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429543(CHEMBL2333764)
Affinity DataKi: >5.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50429566(CHEMBL2333348)
Affinity DataKi: >5.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetP2Y purinoceptor 2(Homo sapiens (Human))
University Park Nottingham

Curated by ChEMBL
LigandPNGBDBM50271598(CHEMBL4128059)
Affinity DataKi:  5.25E+3nMAssay Description:Displacement of (E)-2-((5-(7-Chloro-2-((3-((2-(6-(3-(5,5-difluoro-7,9-dimethyl-5H-5-lambda4,6-lambda4-dipyrrolo[1,2-c:2,1-f ][1,3,2]diazaborinin-3-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50373301(CHEMBL256944)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
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