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Found 49 with Last Name = 'swierczek' and Initial = 'k'
TargetAlkaline phosphatase, germ cell type(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131871(CHEMBL122097 | Methylsulfanylmethyl-phosphonothioi...)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of Human Placental alkaline Phosphatase (PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131868(7-Phosphonomethyl-naphthalene-1-carboxylic acid | ...)
Affinity DataKi:  1.30E+5nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131866(7-Thiophosphonomethyl-naphthalene-1-carboxylic aci...)
Affinity DataKi:  1.70E+5nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein tyrosine phosphatase receptor type C-associated protein(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131866(7-Thiophosphonomethyl-naphthalene-1-carboxylic aci...)
Affinity DataKi:  2.00E+5nMAssay Description:Inhibitory activity against Tyrosine phosphatase from Yersinia (Yop protein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, germ cell type(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131861(Benzyl-phosphonothioic acid | CHEMBL123163)
Affinity DataKi:  2.00E+5nMAssay Description:Inhibition of Human Placental alkaline Phosphatase (PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Rattus norvegicus)
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131868(7-Phosphonomethyl-naphthalene-1-carboxylic acid | ...)
Affinity DataKi:  3.00E+5nMAssay Description:Inhibitory activity against E. coli Alkaline PhosphataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, germ cell type(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131865(6-Thiophosphono-hexanoic acid methyl ester | CHEMB...)
Affinity DataKi:  3.30E+5nMAssay Description:Inhibition of Human Placental alkaline Phosphatase (PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, germ cell type(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131868(7-Phosphonomethyl-naphthalene-1-carboxylic acid | ...)
Affinity DataKi:  3.90E+5nMAssay Description:Inhibition of Human Placental alkaline Phosphatase (PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131860(6-Phosphono-hexanoic acid | CHEMBL122539)
Affinity DataKi:  4.30E+5nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, germ cell type(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131863(CHEMBL331460 | Phenylsulfanylmethyl-phosphonothioi...)
Affinity DataKi:  4.60E+5nMAssay Description:Inhibition of Human Placental alkaline Phosphatase (PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131863(CHEMBL331460 | Phenylsulfanylmethyl-phosphonothioi...)
Affinity DataKi:  4.70E+5nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131861(Benzyl-phosphonothioic acid | CHEMBL123163)
Affinity DataKi:  5.70E+5nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, germ cell type(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50080274(Benzyl-phosphonic acid | CHEMBL299737 | Phenyl-met...)
Affinity DataKi:  5.80E+5nMAssay Description:Inhibition of Human Placental alkaline Phosphatase (PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, germ cell type(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131870(Butyl-phosphonothioic acid | CHEMBL331046)
Affinity DataKi:  6.00E+5nMAssay Description:Inhibition of Human Placental alkaline Phosphatase (PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, tissue-nonspecific isozyme(Rattus norvegicus)
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131864(CHEMBL125296 | Propyl-phosphonic acid)
Affinity DataKi:  6.10E+5nMAssay Description:Inhibitory activity against E. coli Alkaline PhosphataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131862(CHEMBL122938 | methylphosphonic acid)
Affinity DataKi:  1.01E+6nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131865(6-Thiophosphono-hexanoic acid methyl ester | CHEMB...)
Affinity DataKi:  1.10E+6nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131871(CHEMBL122097 | Methylsulfanylmethyl-phosphonothioi...)
Affinity DataKi:  1.20E+6nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, germ cell type(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131866(7-Thiophosphonomethyl-naphthalene-1-carboxylic aci...)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of Human Placental alkaline Phosphatase (PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, germ cell type(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131867(6-Thiophosphono-hexanoic acid | CHEMBL123990)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of Human Placental alkaline Phosphatase (PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131867(6-Thiophosphono-hexanoic acid | CHEMBL123990)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, germ cell type(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131864(CHEMBL125296 | Propyl-phosphonic acid)
Affinity DataKi:  1.55E+6nMAssay Description:Inhibition of Human Placental alkaline Phosphatase (PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein tyrosine phosphatase receptor type C-associated protein(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131869(CHEMBL122577 | Methyl-phosphonothioic acid)
Affinity DataKi:  7.00E+6nMAssay Description:Inhibitory activity against Tyrosine phosphatase from Yersinia (Yop protein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, germ cell type(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131860(6-Phosphono-hexanoic acid | CHEMBL122539)
Affinity DataKi:  7.00E+6nMAssay Description:Inhibition of Human Placental alkaline Phosphatase (PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, germ cell type(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131862(CHEMBL122938 | methylphosphonic acid)
Affinity DataKi:  1.10E+7nMAssay Description:Inhibition of Human Placental alkaline Phosphatase (PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein tyrosine phosphatase receptor type C-associated protein(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131863(CHEMBL331460 | Phenylsulfanylmethyl-phosphonothioi...)
Affinity DataKi:  1.58E+7nMAssay Description:Inhibitory activity against Tyrosine phosphatase from Yersinia (Yop protein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131869(CHEMBL122577 | Methyl-phosphonothioic acid)
Affinity DataKi:  1.70E+7nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlkaline phosphatase, germ cell type(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131869(CHEMBL122577 | Methyl-phosphonothioic acid)
Affinity DataKi:  1.90E+7nMAssay Description:Inhibition of Human Placental alkaline Phosphatase (PLAP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131870(Butyl-phosphonothioic acid | CHEMBL331046)
Affinity DataKi:  2.00E+7nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein tyrosine phosphatase receptor type C-associated protein(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131867(6-Thiophosphono-hexanoic acid | CHEMBL123990)
Affinity DataKi:  2.90E+7nMAssay Description:Inhibitory activity against Tyrosine phosphatase from Yersinia (Yop protein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein tyrosine phosphatase receptor type C-associated protein(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131862(CHEMBL122938 | methylphosphonic acid)
Affinity DataKi:  3.00E+7nMAssay Description:Inhibitory activity against Tyrosine phosphatase from Yersinia (Yop protein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein tyrosine phosphatase receptor type C-associated protein(Homo sapiens (Human))
Utah State University

Curated by ChEMBL
LigandPNGBDBM50131860(6-Phosphono-hexanoic acid | CHEMBL122539)
Affinity DataKi:  4.20E+7nMAssay Description:Inhibitory activity against Tyrosine phosphatase from Yersinia (Yop protein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161093((R)-2-chloro-6-(2-hydroxy-3-(2-methyl-1-(naphthale...)
Affinity DataIC50:  43nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166511(3-[2-(3-Fluoro-phenyl)-ethyl]-2-(2-hydroxy-phenyl)...)
Affinity DataIC50:  95nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166504(5-Ethyl-3-[2-(2-fluoro-phenyl)-ethyl]-2-(2-hydroxy...)
Affinity DataIC50:  97nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166510(5-Ethyl-2-(2-hydroxy-phenyl)-6-methyl-3-phenethyl-...)
Affinity DataIC50:  100nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166517(5-Cyclopropyl-3-[2-(3-fluoro-phenyl)-ethyl]-2-(2-h...)
Affinity DataIC50:  120nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166507(2-(2-Hydroxy-phenyl)-3-phenethyl-4a,5,6,7,8,8a-hex...)
Affinity DataIC50:  140nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166503(3-[2-(3-Fluoro-phenyl)-ethyl]-2-(2-hydroxy-phenyl)...)
Affinity DataIC50:  140nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166505(3-[2-(3-Fluoro-phenyl)-ethyl]-2-(2-hydroxy-phenyl)...)
Affinity DataIC50:  160nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166512(3-[2-(3-Fluoro-phenyl)-ethyl]-2-(2-hydroxy-phenyl)...)
Affinity DataIC50:  170nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166514(2-(2-Hydroxy-phenyl)-5,6-dimethyl-3-phenethyl-3H-p...)
Affinity DataIC50:  200nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166509(3-[2-(3-Fluoro-phenyl)-ethyl]-2-(2-hydroxy-phenyl)...)
Affinity DataIC50:  200nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166508(2-(2-Hydroxy-phenyl)-3-phenethyl-3,4a,5,6,7,7a-hex...)
Affinity DataIC50:  200nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166516(2-(2-Hydroxy-phenyl)-5-methyl-3-phenethyl-6-triflu...)
Affinity DataIC50:  800nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166506(3-[2-(3-Fluoro-phenyl)-ethyl]-2-(2-hydroxy-phenyl)...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166515(3-[2-(2-Fluoro-phenyl)-ethyl]-2-(2-hydroxy-phenyl)...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50166513(2-(2-Hydroxy-phenyl)-6-methyl-3-phenethyl-3H-pyrim...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Nps Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50162542(2-Furan-2-yl-3-phenethyl-3H-quinazolin-4-one | CHE...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibitory concentration was evaluated for in vitro calcilytic activity against human calcium receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed