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Found 40 with Last Name = 'takai' and Initial = 'a'
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375611(CHEMBL408120)
Affinity DataKi:  3.40nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375608(CHEMBL406220)
Affinity DataKi:  4.5nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375616(CHEMBL405248)
Affinity DataKi:  8nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375613(CHEMBL261577)
Affinity DataKi:  8.40nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375612(CHEMBL427915)
Affinity DataKi:  17.3nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375609(CHEMBL406283)
Affinity DataKi:  19.6nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375614(CHEMBL259235)
Affinity DataKi:  21.3nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375610(CHEMBL436904)
Affinity DataKi:  23.9nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375617(CHEMBL261094)
Affinity DataKi:  32.5nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University

Curated by ChEMBL
LigandPNGBDBM50375615(CHEMBL261583)
Affinity DataKi:  49.7nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  1nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40777(Hemicalyculin A (5))
Affinity DataIC50:  1nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40787(Des-N-methylcalyculin A (20))
Affinity DataIC50:  1nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40782(C1/C34-Calyculin A (15))
Affinity DataIC50:  1.10nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40785(Calyculinamide A (18))
Affinity DataIC50:  1.5nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40780(Calyculin A 21-acetate (13))
Affinity DataIC50:  2.10nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40790(Calyculin C (24))
Affinity DataIC50:  2.60nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40785(Calyculinamide A (18))
Affinity DataIC50:  5nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  7.5nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  8.20nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40782(C1/C34-Calyculin A (15))
Affinity DataIC50:  9nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  9nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40787(Des-N-methylcalyculin A (20))
Affinity DataIC50:  11nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40780(Calyculin A 21-acetate (13))
Affinity DataIC50:  13nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  14nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40777(Hemicalyculin A (5))
Affinity DataIC50:  14nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40781(Calyculin J (14))
Affinity DataIC50:  20nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40790(Calyculin C (24))
Affinity DataIC50:  29nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  55nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40781(Calyculin J (14))
Affinity DataIC50:  105nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  112nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  185nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40784(Dephosphonocalyculin A (17))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40778(11,13-O-isopropylidene-calyculin A (6))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40779(Calyculin A 11,13,21-triacetate (12))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40778(11,13-O-isopropylidene-calyculin A (6))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40783(C9/C35-calyculin (16))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40784(Dephosphonocalyculin A (17))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40783(C9/C35-calyculin (16))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University of Tokyo

LigandPNGBDBM40779(Calyculin A 11,13,21-triacetate (12))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed