Affinity DataKi: 0.25nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]-Naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 0.370nMAssay Description:Binding affinity against Opioid receptor mu 1 of guinea pig brain membranes using 0.5 nM of [3H]naloxone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Binding affinity against Opioid receptor mu 1 of guinea pig brain membranes using 0.5 nM of [3H]naloxone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.570nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]-Naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 0.760nMAssay Description:Binding affinity against Opioid receptor mu 1 of guinea pig brain membranes using 0.5 nM of [3H]naloxone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity of the compound towards sigma receptor using radiolabeled ligand [3H]-(+)-SKF- 10,047 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity towards sigma receptor using [3H]-(+)-SKF-10,047 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for sigma receptor in guinea pig brain membrane using radiolabeled ligand [3H]-(+)-SKF- 10,047 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for sigma receptor in guinea pig brain membrane using radiolabeled ligand [3H]-(+)-SKF- 10,047 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for sigma receptor in guinea pig brain membrane using radiolabeled ligand [3H]-(+)-SKF- 10,047 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]-Naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:In vivo binding affinity against kappa opioid receptor was measured by using labeled ligand [3H]-ethylketocyclazocine (1 nM) with 500 nM DADLE and 20...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]-Naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity against opioid receptor kappa from guinea pig brain membranes using [3H]ethylketocyclazocine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:In vivo binding affinity against kappa opioid receptor was measured by using labeled ligand [3H]-ethylketocyclazocine (1 nM) with 500 nM DADLE and 20...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity towards sigma receptor using [3H]-(+)-SKF-10,047 as radioligandMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by ChEMBL
Dupont Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity for sigma receptor in guinea pig brain membrane using radiolabeled ligand [3H]-(+)-SKF- 10,047 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity against Opioid receptor kappa 1 of guinea pig brain membranes using 1 nM of (-)-[3H]ethylketazocine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:In vivo binding affinity against delta Opioid receptor was measured by using labeled ligand [3H]-DADLE (1 nM) with 4 nM sufentanilMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity against Opioid receptor mu 1 of guinea pig brain membranes using 0.5 nM of [3H]naloxone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Binding affinity against Opioid receptor kappa 1 of guinea pig brain membranes using 1 nM of (-)-[3H]ethylketazocine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity against Opioid receptor kappa 1 of guinea pig brain membranes using 1 nM of (-)-[3H]ethylketazocine as radioligandMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by ChEMBL
Dupont Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity for sigma receptor in guinea pig brain membrane using radiolabeled ligand [3H]-(+)-SKF- 10,047 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Binding affinity against Opioid receptor delta 1 of guinea pig brain membranes using 1 nM of [3H]DADLE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:The compound was tested for binding activity towards opioid receptor kappa in guinea pig brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity against Opioid receptor delta 1 of guinea pig brain membranes using 1 nM of [3H]DADLE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]-Naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity for sigma receptor in guinea pig brain membrane using radiolabeled ligand [3H]-(+)-SKF- 10,047 was determinedMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by ChEMBL
Dupont Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity of the compound towards sigma receptor using radiolabeled ligand [3H]-(+)-SKF- 10,047 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity for sigma receptor using [3H]-(+)-SKF- 10,047More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity towards sigma receptor using [3H]-(+)-SKF-10,047 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity towards sigma receptor using [3H]-(+)-SKF-10,047 as radioligandMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by ChEMBL
Dupont Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by ChEMBL
Dupont Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity for sigma receptor in guinea pig brain membrane using radiolabeled ligand [3H]-(+)-SKF- 10,047 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity for sigma receptor in guinea pig brain membrane using radiolabeled ligand [3H]-(+)-SKF- 10,047 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity for sigma receptor in guinea pig brain membrane using radiolabeled ligand [3H]-(+)-SKF- 10,047 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity of the compound towards sigma receptor using radiolabeled ligand [3H]-(+)-SKF- 10,047 was determinedMore data for this Ligand-Target Pair