Compile Data Set for Download or QSAR
maximum 50k data
Found 96 with Last Name = 'tevar' and Initial = 's'
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449244(CHEMBL3125150)
Affinity DataIC50:  0.670nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM20880((2S,3R,4R,5S,6R)-2-{4-chloro-3-[(4-ethoxyphenyl)me...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human SGLT2More data for this Ligand-Target Pair
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329198(2-(ethyl((5-(6-methyl-3-(1H-pyrazol-4-yl)imidazo[1...)
Affinity DataIC50:  8nMAssay Description:Inhibition of IRK4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: >10nMAssay Description:Inhibition of AKT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium/calmodulin-dependent protein kinase type IV(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: >10nMAssay Description:Inhibition of Camk4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: >10nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: >10nMAssay Description:Inhibition of CSNK1dMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: >10nMAssay Description:Inhibition of PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: >10nMAssay Description:Inhibition of ROCK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: >10nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTestis-specific serine/threonine-protein kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: >10nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: >10nMAssay Description:Inhibition of PLK3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: >10nMAssay Description:Inhibition of ERK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: >10nMAssay Description:Inhibition of IKK-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: >10nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: >10nMAssay Description:Inhibition of cMETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329198(2-(ethyl((5-(6-methyl-3-(1H-pyrazol-4-yl)imidazo[1...)
Affinity DataIC50:  13nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329201(3-((2,2-dimethylpiperidin-1-yl)methyl)-N-(6-methyl...)
Affinity DataIC50:  45nMAssay Description:Inhibition of LCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329196(3-(1-((2S,6R)-2,6-dimethylmorpholino)cyclopropyl)-...)
Affinity DataIC50:  45nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329196(3-(1-((2S,6R)-2,6-dimethylmorpholino)cyclopropyl)-...)
Affinity DataIC50:  50nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM20875(1-(2,4-dihydroxy-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihyd...)
Affinity DataIC50:  59nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM20875(1-(2,4-dihydroxy-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihyd...)
Affinity DataIC50:  61nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50093599(CHEMBL3585803)
Affinity DataIC50:  100nMAssay Description:Inhibition of rabbit lung ACE assessed as hippuryl-histidyl-leucine hydrolysis after 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50021153(1H-1-Benzazepine-1-acetic acid, 3-((1-(ethoxycarbo...)
Affinity DataIC50:  100nMAssay Description:Inhibition of rabbit lung ACE assessed as hippuryl-histidyl-leucine hydrolysis after 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50368166(Accupril | QUINAPRIL)
Affinity DataIC50:  110nMAssay Description:Inhibition of rabbit lung ACE assessed as hippuryl-histidyl-leucine hydrolysis after 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50017129((S)-1-((S)-2-((R)-1-ethoxy-1-oxo-4-phenylbutan-2-y...)
Affinity DataIC50:  123nMAssay Description:Inhibition of rabbit lung ACE assessed as hippuryl-histidyl-leucine hydrolysis after 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449247(CHEMBL3125147)
Affinity DataIC50:  126nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449242(CHEMBL3125151)
Affinity DataIC50:  135nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50:  140nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449239(CHEMBL3125155)
Affinity DataIC50:  147nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449240(CHEMBL3125154)
Affinity DataIC50:  149nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449252(CHEMBL3125142)
Affinity DataIC50:  150nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449251(CHEMBL3125143)
Affinity DataIC50:  152nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449243(CHEMBL3125152)
Affinity DataIC50:  163nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449248(CHEMBL3125146)
Affinity DataIC50:  175nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329198(2-(ethyl((5-(6-methyl-3-(1H-pyrazol-4-yl)imidazo[1...)
Affinity DataIC50:  180nMAssay Description:Inhibition of RSK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449253(CHEMBL3125141)
Affinity DataIC50:  186nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449250(CHEMBL3125144)
Affinity DataIC50:  190nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50021153(1H-1-Benzazepine-1-acetic acid, 3-((1-(ethoxycarbo...)
Affinity DataIC50:  212nMAssay Description:Inhibition of rabbit lung ACE assessed as hydrolysis of hippuryl-histidyl-leucine to hippuric acid and histidyl-leucine after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449241(CHEMBL3125153)
Affinity DataIC50:  214nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449247(CHEMBL3125147)
Affinity DataIC50:  220nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449245(CHEMBL3125149)
Affinity DataIC50:  227nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50084681(1-[2-(1-Ethoxycarbonyl-3-phenyl-propylamino)-propi...)
Affinity DataIC50:  253nMAssay Description:Inhibition of rabbit lung ACE assessed as hippuryl-histidyl-leucine hydrolysis after 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50084681(1-[2-(1-Ethoxycarbonyl-3-phenyl-propylamino)-propi...)
Affinity DataIC50:  253nMAssay Description:Inhibition of rabbit lung ACE assessed as hydrolysis of hippuryl-histidyl-leucine to hippuric acid and histidyl-leucine after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449249(CHEMBL3125145)
Affinity DataIC50:  257nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50367879(LISINOPRIL)
Affinity DataIC50:  262nMAssay Description:Inhibition of rabbit lung ACE assessed as hydrolysis of hippuryl-histidyl-leucine to hippuric acid and histidyl-leucine after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50438379(CHEMBL2413588)
Affinity DataIC50:  272nMAssay Description:Inhibition of rabbit lung ACE assessed as hydrolysis of hippuryl-histidyl-leucine to hippuric acid and histidyl-leucine after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449254(CHEMBL3125156)
Affinity DataIC50:  311nMAssay Description:Inhibition of SGLT2 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449242(CHEMBL3125151)
Affinity DataIC50:  315nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Csir-Indian Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50449239(CHEMBL3125155)
Affinity DataIC50:  315nMAssay Description:Inhibition of SGLT1 (unknown origin) expressed in HEK293 cells using 2-NBDG as substrate incubated for 30 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 96 total ) | Next | Last >>
Jump to: