TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of BTK (unknown origin) by FRET assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetNon-receptor tyrosine-protein kinase TYK2/Tyrosine-protein kinase JAK1/Tyrosine-protein kinase JAK2/Tyrosine-protein kinase JAK3(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: >5nMAssay Description:Inhibition of JAK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of TEC (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 5.90nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 6.20nMAssay Description:Inhibition of TEC (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of BTK (unknown origin) assessed as reduction in TNF productionMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of ITK (unknown origin) by FRET assayMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of ErbB4/HER4 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of TEC (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of EGFR exon 19 deletion and L858R mutant phosphorylation in human NCI-H1975 cellsMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Panjab University
Curated by ChEMBL
Panjab University
Curated by ChEMBL
Affinity DataIC50: 22.1nMAssay Description:Inhibition of human type-2 5-alpha reductase expressed in HEK293 cells using [3H]-androstenedione as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Panjab University
Curated by ChEMBL
Panjab University
Curated by ChEMBL
Affinity DataIC50: 26.5nMAssay Description:Inhibition of human type-2 5-alpha reductase expressed in HEK293 cells using [3H]-androstenedione as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Panjab University
Curated by ChEMBL
Panjab University
Curated by ChEMBL
Affinity DataIC50: 30.3nMAssay Description:Inhibition of human type-2 5-alpha reductase expressed in HEK293 cells using [3H]-androstenedione as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
TargetCytoplasmic tyrosine-protein kinase BMX(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of BMX (unknown origin)More data for this Ligand-Target Pair
TargetCytoplasmic tyrosine-protein kinase BMX(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of BMX (unknown origin)More data for this Ligand-Target Pair
TargetSTE20-like serine/threonine-protein kinase(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of SLK (unknown origin)More data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Panjab University
Curated by ChEMBL
Panjab University
Curated by ChEMBL
Affinity DataIC50: 54.1nMAssay Description:Inhibition of human type-2 5-alpha reductase expressed in HEK293 cells using [3H]-androstenedione as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of TEC (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of TEC (unknown origin)More data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Panjab University
Curated by ChEMBL
Panjab University
Curated by ChEMBL
Affinity DataIC50: 72.8nMAssay Description:Inhibition of human type-2 5-alpha reductase expressed in HEK293 cells using [3H]-androstenedione as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Inhibition of TEC (unknown origin) by FRET assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of LYN (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Panjab University
Curated by ChEMBL
Panjab University
Curated by ChEMBL
Affinity DataIC50: 213nMAssay Description:Inhibition of human type-2 5-alpha reductase expressed in HEK293 cells using [3H]-androstenedione as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Panjab University
Curated by ChEMBL
Panjab University
Curated by ChEMBL
Affinity DataIC50: 453nMAssay Description:Inhibition of human type-1 5-alpha reductase expressed in HEK293 cells using [3H]-androstenedione as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 652nMAssay Description:Inhibition of BTK (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of wild type EGFR phosphorylation in human H358 cellsMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of LYN (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of JAK3 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SYK (unknown origin) by FRET assayMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Shaanxi University Of Science & Technology
Curated by ChEMBL
Shaanxi University Of Science & Technology
Curated by ChEMBL
Affinity DataKd: 0.540nMAssay Description:Binding affinity to RPS6KA3 (unknown origin)More data for this Ligand-Target Pair