Affinity DataKi: 0.398nMAssay Description:Antagonist activity at human recombinant EP1 receptor expressed in CHO-K1 cells assessed as inhibition of PGE2-mediated intracellular calcium mobiliz...More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Antagonist activity against human EP1 receptor expressed in CHOK1 cells assessed as inhibition of PGE2-induced intracellular calcium mobilization by ...More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Antagonist activity at human recombinant EP3 receptor expressed in CHO-K1 cells assessed as inhibition of PGE2-mediated intracellular calcium mobiliz...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01nMAssay Description:Displacement of [3H]PGE2 from human prostanoid EP1 receptor expressed in CHO-K1 cells after 30 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Displacement of [3H]PGE2 from human EP1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.31nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 7.94nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 19.9nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 19.9nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 25.1nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 25.1nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 25.1nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 25.1nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 39.8nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 39.8nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Displacement of [3H]PGE2 from human prostanoid EP1 receptor expressed in CHO-K1 cells after 30 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Displacement of [3H]PGE2 from human prostanoid EP1 receptor expressed in CHO-K1 cells after 30 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:Displacement of [3H]PGE2 from human prostanoid EP1 receptor expressed in CHO-K1 cells after 30 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:Displacement of [3H]PGE2 from human prostanoid EP1 receptor expressed in CHO-K1 cells after 30 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 79.4nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of rat P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [3H]PGE2 from human prostanoid EP1 receptor expressed in CHO-K1 cells after 30 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Displacement of [3H]PGE2 from human prostanoid EP1 receptor expressed in CHO-K1 cells after 30 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of rat P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Displacement of [3H]GW875240X from human prostanoid EP1 receptor expressed in CHO-K1 cells after 45 mins by topcount liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair