Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenergic receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenergic receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenergic receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Agonist activity at human alpha2C adrenoceptor expressed in CHO cells assessed as extracellular acidification measured after 4 mins by cytosensor mic...More data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Binding affinity at human alpha2A ARMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Binding affinity at human 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Displacement of [3H]RX821002 from human alpha2C adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair