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Found 47 with Last Name = 'tsai' and Initial = 'yc'
TargetMu-type opioid receptor(GUINEA PIG)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  38nMAssay Description:Binding affinity of the compound against mu opioid receptor was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50070947(2-ethyl-1'-methylspiro[2,3-dihydrobenzo[b]furan-3,...)
Affinity DataKi:  102nMAssay Description:Binding affinity of the compound against mu opioid receptor was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50070948(1',2-dimethylspiro[2,3-dihydrobenzo[b]furan-3,4'-(...)
Affinity DataKi:  124nMAssay Description:Binding affinity of the compound against mu opioid receptor was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50026752(1-Methyl-4-phenyl-piperidine-4-carboxylic acid eth...)
Affinity DataKi:  451nMAssay Description:Binding affinity of the compound against mu opioid receptor was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50070946(1',3'-dimethylspiro[2,3-dihydrobenzo[b]furan-3,4'-...)
Affinity DataKi:  505nMAssay Description:Binding affinity against Opioid receptor kappa 1 was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50070946(1',3'-dimethylspiro[2,3-dihydrobenzo[b]furan-3,4'-...)
Affinity DataKi:  505nMAssay Description:Binding affinity of the compound against Opioid receptor kappa 1 was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  510nMAssay Description:Binding affinity of the compound against Opioid receptor delta 1 was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286878(Butyl-carbamic acid 2'-hydroxy-[1,1']binaphthaleny...)
Affinity DataKi:  800nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 (KDR)More data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286878(Butyl-carbamic acid 2'-hydroxy-[1,1']binaphthaleny...)
Affinity DataKi:  800nMAssay Description:Dissociation constant of the compound (KI) for the Pancreatic cholesterol esterase-catalyzed hydrolysis of 4-nitrophenyl butyrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286878(Butyl-carbamic acid 2'-hydroxy-[1,1']binaphthaleny...)
Affinity DataKi:  800nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 (KDR)More data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50070947(2-ethyl-1'-methylspiro[2,3-dihydrobenzo[b]furan-3,...)
Affinity DataKi:  853nMAssay Description:Binding affinity of the compound against Opioid receptor delta 1 was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50070946(1',3'-dimethylspiro[2,3-dihydrobenzo[b]furan-3,4'-...)
Affinity DataKi:  1.01E+3nMAssay Description:Binding affinity against mu opioid receptor was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50070946(1',3'-dimethylspiro[2,3-dihydrobenzo[b]furan-3,4'-...)
Affinity DataKi:  1.02E+3nMAssay Description:Binding affinity of the compound against mu opioid receptor was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50070949(1'-methylspiro[2,3-dihydrobenzo[b]furan-3,4'-(hexa...)
Affinity DataKi:  1.65E+3nMAssay Description:Binding affinity of the compound against mu opioid receptor was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  1.87E+3nMAssay Description:Binding affinity of the compound against Opioid receptor kappa 1 was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50070948(1',2-dimethylspiro[2,3-dihydrobenzo[b]furan-3,4'-(...)
Affinity DataKi:  2.41E+3nMAssay Description:Binding affinity of the compound against Opioid receptor delta 1 was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286880(Butyric acid 2'-butylcarbamoyloxy-[1,1']binaphthal...)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 (KDR)More data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286880(Butyric acid 2'-butylcarbamoyloxy-[1,1']binaphthal...)
Affinity DataKi:  2.00E+4nMAssay Description:Dissociation constant of the compound (KI) for the Pancreatic cholesterol esterase-catalyzed hydrolysis of 4-nitrophenyl butyrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286880(Butyric acid 2'-butylcarbamoyloxy-[1,1']binaphthal...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 (KDR)More data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286879(Butyl-carbamic acid 2'-butylcarbamoyloxy-[1,1']bin...)
Affinity DataKi:  2.90E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 (KDR)More data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286879(Butyl-carbamic acid 2'-butylcarbamoyloxy-[1,1']bin...)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 (KDR)More data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286879(Butyl-carbamic acid 2'-butylcarbamoyloxy-[1,1']bin...)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 (KDR)More data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50070947(2-ethyl-1'-methylspiro[2,3-dihydrobenzo[b]furan-3,...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity of the compound against Opioid receptor kappa 1 was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50026752(1-Methyl-4-phenyl-piperidine-4-carboxylic acid eth...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity of the compound against Opioid receptor kappa 1 was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50070948(1',2-dimethylspiro[2,3-dihydrobenzo[b]furan-3,4'-(...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity of the compound against Opioid receptor kappa 1 was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50070949(1'-methylspiro[2,3-dihydrobenzo[b]furan-3,4'-(hexa...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity of the compound against Opioid receptor kappa 1 was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50070949(1'-methylspiro[2,3-dihydrobenzo[b]furan-3,4'-(hexa...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity of the compound against Opioid receptor delta 1 was determined in brain membrane preparations from male Hartley guinea-pigsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
National Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50428362(15-O-Acetylganolucidate A | CHEMBL2331733)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of iNOS-mediated nitric oxide production in LPS-stimulated mouse RAW264.7 cells after 24 hrs by Griess reaction analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
National Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50428365(CHEMBL2331728)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of iNOS-mediated nitric oxide production in LPS-stimulated mouse RAW264.7 cells after 24 hrs by Griess reaction analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
National Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50428366(CHEMBL2203598)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of iNOS-mediated nitric oxide production in LPS-stimulated mouse RAW264.7 cells after 24 hrs by Griess reaction analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
National Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50428364(CHEMBL2331730)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of iNOS-mediated nitric oxide production in LPS-stimulated mouse RAW264.7 cells after 24 hrs by Griess reaction analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
National Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50428363(CHEMBL2331729)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of iNOS-mediated nitric oxide production in LPS-stimulated mouse RAW264.7 cells after 24 hrs by Griess reaction analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
National Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50428361(CHEMBL2331731 | Ethyl Lucidenate A)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of iNOS-mediated nitric oxide production in LPS-stimulated mouse RAW264.7 cells after 24 hrs by Griess reaction analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
National Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  1.64E+4nMAssay Description:Inhibition of iNOS-mediated nitric oxide production in LPS-stimulated mouse RAW264.7 cells after 24 hrs by Griess reaction analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
National Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50428360(CHEMBL2331732 | Ethyl Lucidenate F)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of iNOS-mediated nitric oxide production in LPS-stimulated mouse RAW264.7 cells after 24 hrs by Griess reaction analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
National Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50428359(CHEMBL2331734)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of iNOS-mediated nitric oxide production in LPS-stimulated mouse RAW264.7 cells after 24 hrs by Griess reaction analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
National Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50428358(CHEMBL2331735)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of iNOS-mediated nitric oxide production in LPS-stimulated mouse RAW264.7 cells after 24 hrs by Griess reaction analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
National Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50428357(CHEMBL2331727)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of iNOS-mediated nitric oxide production in LPS-stimulated mouse RAW264.7 cells after 24 hrs by Griess reaction analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286879(Butyl-carbamic acid 2'-butylcarbamoyloxy-[1,1']bin...)
Affinity DataKoff:  4.00E+3s-1Assay Description:Dissociation constant of the compound (KI) for the Pancreatic cholesterol esterase-catalyzed hydrolysis of 4-nitrophenyl butyrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286880(Butyric acid 2'-butylcarbamoyloxy-[1,1']binaphthal...)
Affinity DataKoff:  6.00E+3s-1Assay Description:Inhibition of Vascular endothelial growth factor receptor 2 (KDR)More data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286880(Butyric acid 2'-butylcarbamoyloxy-[1,1']binaphthal...)
Affinity DataKoff:  6.00E+3s-1Assay Description:Inhibition of Vascular endothelial growth factor receptor 2 (KDR)More data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286880(Butyric acid 2'-butylcarbamoyloxy-[1,1']binaphthal...)
Affinity DataKoff:  6.00E+3s-1Assay Description:Inhibition of Vascular endothelial growth factor receptor 2 (KDR)More data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286878(Butyl-carbamic acid 2'-hydroxy-[1,1']binaphthaleny...)
Affinity DataKoff:  5.00E+5s-1Assay Description:Inhibition of Vascular endothelial growth factor receptor 2 (KDR)More data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286878(Butyl-carbamic acid 2'-hydroxy-[1,1']binaphthaleny...)
Affinity DataKoff:  5.00E+5s-1Assay Description:Inhibition of Vascular endothelial growth factor receptor 2 (KDR)More data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286879(Butyl-carbamic acid 2'-butylcarbamoyloxy-[1,1']bin...)
Affinity DataKoff:  4.00E+3s-1Assay Description:Dissociation constant of the compound (KI) for the Pancreatic cholesterol esterase-catalyzed hydrolysis of 4-nitrophenyl butyrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286879(Butyl-carbamic acid 2'-butylcarbamoyloxy-[1,1']bin...)
Affinity DataKoff:  4.00E+3s-1Assay Description:Dissociation constant of the compound (KI) for the Pancreatic cholesterol esterase-catalyzed hydrolysis of 4-nitrophenyl butyrateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetBile salt-activated lipase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286878(Butyl-carbamic acid 2'-hydroxy-[1,1']binaphthaleny...)
Affinity DataKoff:  5.00E+5s-1Assay Description:Inhibition of Vascular endothelial growth factor receptor 2 (KDR)More data for this Ligand-Target Pair
In DepthDetails Article