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Found 61 with Last Name = 'tsang' and Initial = 'm'
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50277623(CHEMBL451523 | N-(5-tert-butyl-2-methoxy-3-(3-(4-(...)
Affinity DataIC50:  3nMAssay Description:Inhibition of JNK2alpha2 (unknown origin) by by exchange curve binding kinetic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM175526(US9120744, CDE-002)
Affinity DataIC50:  58nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218689(CHEMBL245230 | N-(5-tert-butyl-2-methoxy-3-(3-naph...)
Affinity DataIC50:  79nMAssay Description:Binding affinity to p38alpha (unknown origin) assessed as inhibition of ATF2 phosphorylation preincubated for 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM50522442(CHEMBL383306)
Affinity DataIC50:  100nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM50522441(CHEMBL4557794)
Affinity DataIC50:  132nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM50522452(CHEMBL4469305)
Affinity DataIC50:  167nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50277623(CHEMBL451523 | N-(5-tert-butyl-2-methoxy-3-(3-(4-(...)
Affinity DataIC50:  480nMAssay Description:Inhibition of Abl (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM50241052(1,2,3,4,6-Pgg | 1,2,3,4,6-pentakis-O-(3,4,5-trihyd...)
Affinity DataIC50:  607nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50277623(CHEMBL451523 | N-(5-tert-butyl-2-methoxy-3-(3-(4-(...)
Affinity DataIC50:  880nMAssay Description:Inhibition of craf (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM50522447(CHEMBL4440070)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50277623(CHEMBL451523 | N-(5-tert-butyl-2-methoxy-3-(3-(4-(...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of Lyn (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218677(CHEMBL242005 | N-(5-tert-butyl-2-methoxy-3-(methyl...)
Affinity DataIC50:  2.70E+3nMAssay Description:Binding affinity to p38alpha (unknown origin) assessed as inhibition of ATF2 phosphorylation preincubated for 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-A receptor 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50277623(CHEMBL451523 | N-(5-tert-butyl-2-methoxy-3-(3-(4-(...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of HEK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM50522443(CHEMBL4474868)
Affinity DataIC50:  3.42E+3nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50277627(1-(5-tert-butyl-2-methoxyphenyl)-3-(naphthalen-1-y...)
Affinity DataIC50:  3.90E+3nMAssay Description:Binding affinity to p38alpha (unknown origin) assessed as inhibition of ATF2 phosphorylation preincubated for 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218695(CHEMBL390254 | N-(5-tert-butyl-2-methoxy-3-(methyl...)
Affinity DataIC50:  4.10E+3nMAssay Description:Binding affinity to p38alpha (unknown origin) assessed as inhibition of ATF2 phosphorylation preincubated for 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-A receptor 2(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50277623(CHEMBL451523 | N-(5-tert-butyl-2-methoxy-3-(3-(4-(...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of ECK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50277623(CHEMBL451523 | N-(5-tert-butyl-2-methoxy-3-(3-(4-(...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50277623(CHEMBL451523 | N-(5-tert-butyl-2-methoxy-3-(3-(4-(...)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of PKBalpha/Akt1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50277623(CHEMBL451523 | N-(5-tert-butyl-2-methoxy-3-(3-(4-(...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of bRaf (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM50522448(CHEMBL4439272)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM50522449(CHEMBL4437267)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM50522450(CHEMBL4570281)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM50522451(CHEMBL4463429)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM50522453(CHEMBL383459)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50277663(CHEMBL519511 | N-(5-tert-butyl-2-methoxyphenyl)ben...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to p38alpha (unknown origin) assessed as inhibition of ATF2 phosphorylation preincubated for 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM50522446(CHEMBL4521362)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM50522445(CHEMBL4555734)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAnthrax toxin receptor 2(Homo sapiens)
Instituto De Qu£Mica M£Dica (Iqm)

Curated by ChEMBL
LigandPNGBDBM50522444(CHEMBL4446670)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AF488-labelled PA binding to AF546- labelled GST-tagged CMG2 R40C/C178A double mutant (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50277662(CHEMBL484405 | N-(5-tert-butyl-2-methoxyphenyl)ben...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to p38alpha (unknown origin) assessed as inhibition of ATF2 phosphorylation preincubated for 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 1(Homo sapiens (Human))
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50326052((E)-2-benzylidene-3-(cyclohexylamino)-2,3-dihydro-...)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of Myc-tagged human Dusp1 expressed in TPA-induced human HeLa cells asssessed as decrease in dephosphorylation of pERK measured by immunos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 6(Homo sapiens (Human))
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50326052((E)-2-benzylidene-3-(cyclohexylamino)-2,3-dihydro-...)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibition of Myc-tagged human Dusp6 expressed in TPA-induced human HeLa cells asssessed as decrease in dephosphorylation of pERK measured by immunos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14846(1-(3-tert-butyl-1-cyclohexyl-1H-pyrazol-5-yl)-3-[4...)
Affinity DataKd:  23nMpH: 7.0 T: 2°CAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14835(1-(5-tert-Butyl-2-methyl-2H-pyrazol-3-yl)-3-[4-(2-...)
Affinity DataKd:  26nMpH: 7.0 T: 2°CAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14845(1-(2-Benzyl-5-tert-butyl-2H-pyrazol-3-yl)-3-[4-(2-...)
Affinity DataKd:  64nMpH: 7.0 T: 2°CAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14844(1-[5-tert-Butyl-2-(6-methyl-pyridin-3-yl)-2H-pyraz...)
Affinity DataKd:  0.180nMpH: 7.0 T: 2°CAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50277615(1-(5-tert-butyl-2-methoxyphenyl)-3-(4-(6-(morpholi...)
Affinity DataKd:  1.80nMAssay Description:Binding affinity to p38alpha (unknown origin) by exchange curve binding kinetic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataKd:  0.100nMAssay Description:Binding affinity to p38alpha (unknown origin) by exchange curve binding kinetic analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataKd:  0.0460nMpH: 7.0 T: 2°CAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14843(1-[5-(1-Methylcyclohexyl)-2-phenyl-2H-pyrazol-3-yl...)
Affinity DataKd:  1.90nMpH: 7.0 T: 2°CAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14839(1-(5-tert-Butyl-2-phenyl-2H-pyrazol-3-yl)-3-[4-(2-...)
Affinity DataKd:  0.230nMpH: 7.0 T: 2°CAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14838(1-(5-iso-Propyl-2-phenyl-2H-pyrazol-3-yl)-3-[4-(2-...)
Affinity DataKd:  3.40nMpH: 7.0 T: 2°CAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14842(1-[4-(2-Morpholin-4-yl-ethoxy)-naphthalen-1-yl]-3-...)
Affinity DataKd:  2.40E+3nMpH: 7.0 T: 2°CAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14834(1-[5-(2-Hydroxy-1,1-dimethylethyl)-2-p-tolyl-2H-py...)
Affinity DataKd:  56nMpH: 7.0 T: 2°CAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataKd:  20nMpH: 7.0 T: 2°CAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14847(1-[2-(3-Aminophenyl)-5-tert-butyl-2H-pyrazol-3-yl]...)
Affinity DataKd:  0.230nMpH: 7.0 T: 2°CAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14848(BIRB-796 Analog 39 | N-(3-{3-tert-butyl-5-[({4-[2-...)
Affinity DataKd:  9.90nMpH: 7.0 T: 2°CAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14849(1-[2-(4-Aminophenyl)-5-tert-butyl-2H-pyrazol-3-yl]...)
Affinity DataKd:  0.160nMpH: 7.0 T: 2°CAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14850(BIRB-796 Analog 41 | N-(4-{3-tert-butyl-5-[({4-[2-...)
Affinity DataKd:  64nMAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Mus musculus (mouse))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM14851(1-[5-tert-Butyl-2-(6-methoxypyridin-3-yl)-2H-pyraz...)
Affinity DataKd:  0.870nMAssay Description:UV thermal melt experiments were carried out in a quartz cuvette loaded with sample containing enzyme and each test compound using a spectrophotomete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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