Affinity DataKi: 7nMAssay Description:Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Inhibition of CYP1A1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Inhibition of CYP1A1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Inhibition of CYP1A1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Inhibition of CYP1A1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Inhibition of CYP1A1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Inhibition of CYP1A1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Inhibition of CYP1A1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 660nMAssay Description:Inhibition of CYP1A1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 670nMAssay Description:Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Competitive inhibition of human recombinant ERAP2 expressed in baculovirus infected sf9 cells using R-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 750nMAssay Description:Inhibition of CYP1A1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: >800nMAssay Description:Inhibition of CYP1A1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: >800nMAssay Description:Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: 890nMAssay Description:Inhibition of CYP1A1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Competitive inhibition of human recombinant ERAP2 expressed in baculovirus infected sf9 cells using R-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 1.22E+3nMAssay Description:Inhibition of CYP1A1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Competitive inhibition of human recombinant IRAP expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by M...More data for this Ligand-Target Pair
Affinity DataKi: 1.64E+3nMAssay Description:Inhibition of CYP1A1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: >2.34E+3nMAssay Description:Inhibition of CYP1B1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
Affinity DataKi: >2.34E+3nMAssay Description:Inhibition of CYP1A1 EROD activity assessed as inhibition of deethylation of 7-ethoxyresorufin to resorufinMore data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 3.20E+3nMAssay Description:Competitive inhibition of human recombinant IRAP expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by M...More data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 3.80E+3nMAssay Description:Competitive inhibition of human recombinant IRAP expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by M...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 4.30E+3nMAssay Description:Competitive inhibition of human recombinant ERAP2 expressed in baculovirus infected sf9 cells using R-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 4.60E+3nMAssay Description:Competitive inhibition of human recombinant IRAP expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by M...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 4.70E+3nMAssay Description:Competitive inhibition of human recombinant ERAP1 expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 4.80E+3nMAssay Description:Competitive inhibition of human recombinant ERAP2 expressed in baculovirus infected sf9 cells using R-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 4.90E+3nMAssay Description:Competitive inhibition of human recombinant ERAP2 expressed in baculovirus infected sf9 cells using R-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 5.70E+3nMAssay Description:Competitive inhibition of human recombinant IRAP expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by M...More data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 8.70E+3nMAssay Description:Competitive inhibition of human recombinant IRAP expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by M...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 1.09E+4nMAssay Description:Competitive inhibition of human recombinant ERAP1 expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 1.30E+4nMAssay Description:Competitive inhibition of human recombinant IRAP expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by M...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 1.74E+4nMAssay Description:Competitive inhibition of human recombinant ERAP2 expressed in baculovirus infected sf9 cells using R-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 1.75E+4nMAssay Description:Competitive inhibition of human recombinant ERAP1 expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetInterleukin-1 receptor antagonist protein(Homo sapiens)
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 1.76E+4nMAssay Description:Competitive inhibition of human recombinant IRAP expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by M...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 1.77E+4nMAssay Description:Competitive inhibition of human recombinant ERAP2 expressed in baculovirus infected sf9 cells using R-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 1.85E+4nMAssay Description:Competitive inhibition of human recombinant ERAP1 expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 2.14E+4nMAssay Description:Competitive inhibition of human recombinant ERAP2 expressed in baculovirus infected sf9 cells using R-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 1(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 2.34E+4nMAssay Description:Competitive inhibition of human recombinant ERAP1 expressed in baculovirus infected sf9 cells using L-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
National Centre For Scientific Research "Demokritos
Curated by ChEMBL
Affinity DataKi: 2.74E+4nMAssay Description:Competitive inhibition of human recombinant ERAP2 expressed in baculovirus infected sf9 cells using R-AMC as substrate incubated for 5 to 10 mins by ...More data for this Ligand-Target Pair