Affinity DataKi: 0.200nMAssay Description:In vitro inhibitory activity against glutamate carboxypeptidase II (GCP II) using N-acetyl-L-aspartyl-[3H]-L-glutamate as a substrateMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:In vitro inhibitory activity against glutamate carboxypeptidase II (GCP II) using N-acetyl-L-aspartyl-[3H]-L-glutamate as a substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of N-acetyl-L-aspartyl-[3H]-L-glutamate binding to glutamate carboxypeptidase II (GCP II)More data for this Ligand-Target Pair
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of N-acetyl-L-aspartyl-[3H]-L-glutamate binding to glutamate carboxypeptidase II (GCP II)More data for this Ligand-Target Pair
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
Affinity DataIC50: 580nMAssay Description:Inhibition of N-acetyl-L-aspartyl-[3H]-L-glutamate binding to glutamate carboxypeptidase II (GCP II)More data for this Ligand-Target Pair
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Inhibition of recombinant human MAO-BMore data for this Ligand-Target Pair
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant human MAO-AMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of N-acetyl-L-aspartyl-[3H]-L-glutamate binding to glutamate carboxypeptidase II (GCP II)More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of N-acetyl-L-aspartyl-[3H]-L-glutamate binding to glutamate carboxypeptidase II (GCP II)More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant human MAO-AMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of N-acetyl-L-aspartyl-[3H]-L-glutamate binding to glutamate carboxypeptidase II (GCP II)More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of N-acetyl-L-aspartyl-[3H]-L-glutamate binding to glutamate carboxypeptidase II (GCP II)More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of recombinant human MAO-AMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of N-acetyl-L-aspartyl-[3H]-L-glutamate binding to glutamate carboxypeptidase II (GCP II)More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of N-acetyl-L-aspartyl-[3H]-L-glutamate binding to glutamate carboxypeptidase II (GCP II)More data for this Ligand-Target Pair
TargetMembrane primary amine oxidase(Rattus norvegicus (Rat))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of recombinant human MAO-AMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of N-acetyl-L-aspartyl-[3H]-L-glutamate binding to glutamate carboxypeptidase II (GCP II)More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of recombinant human MAO-AMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of N-acetyl-L-aspartyl-[3H]-L-glutamate binding to glutamate carboxypeptidase II (GCP II)More data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of N-acetyl-L-aspartyl-[3H]-L-glutamate binding to glutamate carboxypeptidase II (GCP II)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-acetyl-L-aspartyl-[3H]-L-glutamate binding to glutamate carboxypeptidase II (GCP II)More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 2.45E+4nMAssay Description:Inhibition of recombinant human MAO-BMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 7.10E+4nMAssay Description:Inhibition of recombinant human MAO-BMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 8.10E+4nMAssay Description:Inhibition of recombinant human MAO-BMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
La Jolla Pharmaceutical
Curated by ChEMBL
La Jolla Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of recombinant human MAO-BMore data for this Ligand-Target Pair