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Found 64 with Last Name = 'whisstock' and Initial = 'jc'
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi:  0.0410nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518240(CHEMBL4439523)
Affinity DataKi:  0.0510nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518249(CHEMBL4588827)
Affinity DataKi:  0.140nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518247(CHEMBL4454304)
Affinity DataKi:  0.210nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518253(CHEMBL4579797)
Affinity DataKi:  0.450nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518252(CHEMBL4592533)
Affinity DataKi:  0.610nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518255(CHEMBL4443353)
Affinity DataKi:  0.660nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518243(CHEMBL4435567)
Affinity DataKi:  0.660nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518239(CHEMBL4453437)
Affinity DataKi:  1.10nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518245(CHEMBL4471930)
Affinity DataKi:  1.20nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518251(CHEMBL4515559)
Affinity DataKi:  1.80nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518244(CHEMBL4550948)
Affinity DataKi:  2nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518246(CHEMBL4563203)
Affinity DataKi:  2.5nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518254(CHEMBL4585149)
Affinity DataKi:  4.70nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518250(CHEMBL4483688)
Affinity DataKi:  8.30nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518249(CHEMBL4588827)
Affinity DataKi:  11nMAssay Description:Inhibition of bovine cationic trypsin using Bz-FVR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518248(CHEMBL4580142)
Affinity DataKi:  16nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518238(CHEMBL4558203)
Affinity DataKi:  16nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi:  28nMAssay Description:Inhibition of bovine cationic trypsin using Bz-FVR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50339789((S)-2-((2S,3R)-3-amino-2-hydroxy-4-(4-methoxypheny...)
Affinity DataKi:  43nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518242(CHEMBL4458397)
Affinity DataKi:  120nMAssay Description:Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518240(CHEMBL4439523)
Affinity DataKi:  160nMAssay Description:Inhibition of bovine cationic trypsin using Bz-FVR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataKi:  190nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50124947(CHEMBL453539)
Affinity DataKi:  200nMAssay Description:Inhibition of recombinant human matriptase catalytic domain pre-incubated for 60 mins before Boc QAR-AMC substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50339790((S)-2-((2S,3R)-3-amino-4-(4-(benzyloxy)phenyl)-2-h...)
Affinity DataKi:  490nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50339784((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi:  900nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50339785((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi:  1.45E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50339791((S)-2-((2S,3R)-3-amino-2-hydroxy-4-(naphthalen-2-y...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50339792((S)-2-((2S,3R)-3-amino-2-hydroxyheptanamido)-4-met...)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518249(CHEMBL4588827)
Affinity DataKi:  7.80E+3nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XI(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518249(CHEMBL4588827)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of activated beta-factor 11 (unknown origin) using Bz-FVRpNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50339787((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi: >1.50E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50339786((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi: >1.50E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50339788((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi: >1.50E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518240(CHEMBL4439523)
Affinity DataKi:  2.90E+4nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518249(CHEMBL4588827)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of plasma KLK (unknown origin) using Ac-NLTR-pNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518240(CHEMBL4439523)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of matriptase (unknown origin) using Boc-QAR-MCA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XI(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of activated beta-factor 11 (unknown origin) using Bz-FVRpNA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518240(CHEMBL4439523)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human thrombin using Ac-ATPR-pNA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XII(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518249(CHEMBL4588827)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of activated beta-factor 12 (unknown origin) using Ac-QRFR-pNA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518249(CHEMBL4588827)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of uPA (unknown origin) using Z-Pyr-Gly-Arg-MCA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor IX(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of activated beta-factor 9 (unknown origin) using Boc-QGR-MCA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of tPA (unknown origin) using Z-Pyr-Gly-Arg-MCA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of plasma KLK (unknown origin) using Ac-NLTR-pNA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518240(CHEMBL4439523)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of plasma KLK (unknown origin) using Ac-NLTR-pNA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of uPA (unknown origin) using Z-Pyr-Gly-Arg-MCA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518240(CHEMBL4439523)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of uPA (unknown origin) using Z-Pyr-Gly-Arg-MCA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518249(CHEMBL4588827)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of tPA (unknown origin) using Z-Pyr-Gly-Arg-MCA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50518241(CHEMBL4569923)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human thrombin using Ac-ATPR-pNA as substrate after 30 mins relative to untreated controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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