TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane by solid scintillation analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 0.570nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 0.570nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane after 180 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 0.590nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 0.590nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 0.710nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 0.740nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 0.790nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane by solid scintillation analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 0.860nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane by solid scintillation analysisMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: >1nMAssay Description:Binding affinity to VAChTMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: >1nMAssay Description:Binding affinity to VAChTMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane by solid scintillation analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane after 180 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane after 180 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane by solid scintillation analysisMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Binding affinity to VAChTMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by scintillation countingMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Homo sapiens (Human))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Binding affinity to EBPMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane after 180 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane after 180 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane after 180 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane after 180 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane after 180 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane by solid scintillation analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane after 180 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane by solid scintillation analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane after 180 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 6.80nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane after 180 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane by solid scintillation analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 8.20nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane after 180 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 9.20nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 180 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institute Of Radiopharmacy
Curated by ChEMBL
Institute Of Radiopharmacy
Curated by ChEMBL
Affinity DataKi: 14.2nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane by scintillation countingMore data for this Ligand-Target Pair