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Found 40 with Last Name = 'wong' and Initial = 'mf'
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  0.100nMAssay Description:Binding affinity towards human Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 1.1 nM 3[H]-9-cis-RAMore data for this Ligand-Target Pair
In DepthDetails ArticleMMDB

TargetRetinoic acid receptor beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 1.1 nM 3[H]-9-cis-RAMore data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50032219((E)-4-(2-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydrona...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 0.82 nM 3[H]-all-trans-RAMore data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 0.82 nM 3[H]-all-trans-RAMore data for this Ligand-Target Pair
In DepthDetails ArticleMMDB

TargetRetinoic acid receptor beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50032219((E)-4-(2-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydrona...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 1.1 nM 3[H]-9-cis-RAMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity towards human Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticleMMDB

TargetRetinoic acid receptor beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 1.1 nM 3[H]-9-cis-RAMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290137((2E,4E)-3-Methyl-5-{2-[(E)-2-(3,3,6,6-tetramethyl-...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity towards human Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290137((2E,4E)-3-Methyl-5-{2-[(E)-2-(3,3,6,6-tetramethyl-...)
Affinity DataKi:  11nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 0.82 nM 3[H]-all-trans-RAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290137((2E,4E)-3-Methyl-5-{2-[(E)-2-(3,3,6,6-tetramethyl-...)
Affinity DataKi:  13nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 0.82 nM 3[H]-all-trans-RAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  27nMAssay Description:Binding affinity towards Retinoic acid receptor RXR-gamma by displacing 3.4 nM 3[H]-9-cis-RAMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290137((2E,4E)-3-Methyl-5-{2-[(E)-2-(3,3,6,6-tetramethyl-...)
Affinity DataKi:  32nMAssay Description:Binding affinity towards human Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  75nMAssay Description:Binding affinity towards Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi: >550nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 0.82 nM 3[H]-all-trans-RAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi: >800nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 1.1 nM 3[H]-9-cis-RAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290138((2Z,4E)-3-Methyl-5-{2-[(E)-2-(3,3,6,6-tetramethyl-...)
Affinity DataKi: >1.10E+3nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 0.82 nM 3[H]-all-trans-RAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290138((2Z,4E)-3-Methyl-5-{2-[(E)-2-(3,3,6,6-tetramethyl-...)
Affinity DataKi: >1.20E+3nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 1.1 nM 3[H]-9-cis-RAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290138((2Z,4E)-3-Methyl-5-{2-[(E)-2-(3,3,6,6-tetramethyl-...)
Affinity DataKi: >2.80E+3nMAssay Description:Binding affinity towards Retinoic acid receptor RXR-gamma by displacing 3.4 nM 3[H]-9-cis-RAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290138((2Z,4E)-3-Methyl-5-{2-[(E)-2-(3,3,6,6-tetramethyl-...)
Affinity DataKi: >4.00E+3nMAssay Description:Binding affinity towards human Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290138((2Z,4E)-3-Methyl-5-{2-[(E)-2-(3,3,6,6-tetramethyl-...)
Affinity DataKi: >4.00E+3nMAssay Description:Binding affinity towards human Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290137((2E,4E)-3-Methyl-5-{2-[(E)-2-(3,3,6,6-tetramethyl-...)
Affinity DataKi: >7.20E+3nMAssay Description:Binding affinity towards Retinoic acid receptor RXR-gamma by displacing 3.4 nM 3[H]-9-cis-RAMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030220(4-[(10R,13R)-17-(1,5-Dimethyl-hexyl)-10,13-dimethy...)
Affinity DataIC50:  60nMAssay Description:The 50% inhibitory concentration was measured as inhibition of RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030217(CHEMBL313213 | Hexadecanoic acid 1-hexadecanoylami...)
Affinity DataIC50:  720nMAssay Description:The 50% inhibitory concentration was measured as inhibition of RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030215(4-Hexadecanoylamino-naphthalene-1,5-disulfonic aci...)
Affinity DataIC50:  1.60E+3nMAssay Description:The 50% inhibitory concentration was measured as inhibition of RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030218(4-Hexadecanoylamino-3-hydroxy-naphthalene-1-sulfon...)
Affinity DataIC50:  3.20E+3nMAssay Description:The 50% inhibitory concentration was measured as inhibition of RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030218(4-Hexadecanoylamino-3-hydroxy-naphthalene-1-sulfon...)
Affinity DataIC50:  3.20E+3nMAssay Description:The 50% inhibitory concentration was measured as inhibition of RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030219(Biphenyl-4,4'-dicarboxylic acid bis-(3,6-disulfo-n...)
Affinity DataIC50:  3.40E+3nMAssay Description:The 50% inhibitory concentration was measured as inhibition of RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030216(4-[5-(3,6-disulfo-1-naphthyloxysulfonyl)-1-naphthy...)
Affinity DataIC50:  4.30E+3nMAssay Description:The 50% inhibitory concentration was measured as inhibition of RNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030217(CHEMBL313213 | Hexadecanoic acid 1-hexadecanoylami...)
Affinity DataIC50:  6.60E+3nMAssay Description:The 50% inhibitory concentration was measured as inhibition of DNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030215(4-Hexadecanoylamino-naphthalene-1,5-disulfonic aci...)
Affinity DataIC50:  6.70E+3nMAssay Description:The 50% inhibitory concentration was measured as inhibition of DNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030219(Biphenyl-4,4'-dicarboxylic acid bis-(3,6-disulfo-n...)
Affinity DataIC50:  6.90E+3nMAssay Description:The 50% inhibitory concentration was measured as inhibition of DNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030220(4-[(10R,13R)-17-(1,5-Dimethyl-hexyl)-10,13-dimethy...)
Affinity DataIC50:  7.90E+3nMAssay Description:The 50% inhibitory concentration was measured as inhibition of DNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030219(Biphenyl-4,4'-dicarboxylic acid bis-(3,6-disulfo-n...)
Affinity DataIC50:  1.44E+4nMAssay Description:The 50% inhibitory concentration was measured as inhibition of Ribonuclease H activity of reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030217(CHEMBL313213 | Hexadecanoic acid 1-hexadecanoylami...)
Affinity DataIC50:  1.68E+4nMAssay Description:The 50% inhibitory concentration was measured as inhibition of Ribonuclease H activity of reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030220(4-[(10R,13R)-17-(1,5-Dimethyl-hexyl)-10,13-dimethy...)
Affinity DataIC50:  2.18E+4nMAssay Description:The 50% inhibitory concentration was measured as inhibition of Ribonuclease H activity of reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030215(4-Hexadecanoylamino-naphthalene-1,5-disulfonic aci...)
Affinity DataIC50:  2.75E+4nMAssay Description:The 50% inhibitory concentration was measured as inhibition of Ribonuclease H activity of reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030218(4-Hexadecanoylamino-3-hydroxy-naphthalene-1-sulfon...)
Affinity DataIC50:  4.76E+4nMAssay Description:The 50% inhibitory concentration was measured as inhibition of Ribonuclease H activity of reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030216(4-[5-(3,6-disulfo-1-naphthyloxysulfonyl)-1-naphthy...)
Affinity DataIC50:  9.13E+4nMAssay Description:The 50% inhibitory concentration was measured as inhibition of DNA-dependent DNA polymerase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50030216(4-[5-(3,6-disulfo-1-naphthyloxysulfonyl)-1-naphthy...)
Affinity DataIC50:  2.15E+5nMAssay Description:The 50% inhibitory concentration was measured as inhibition of Ribonuclease H activity of reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed