Found 251 with Last Name = 'xie' and Initial = 'p' 
Affinity DataKi: 0.00260nMAssay Description:Antagonist activity at cloned muscarinic M2 receptor-Gqi5 chimeric protein expressed in CHO cells assessed as acetylcholine-induced change in cytosol...More data for this Ligand-Target Pair
Affinity DataKi: 0.00340nMAssay Description:Antagonist activity at AT1 receptor in rat aortic ringsMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nM ΔG°: -58.2kJ/molepH: 7.0 T: 2°CAssay Description:BRAF kinase activity was quantified using an ELISA-based MEK phosphorylation assay. IC50 values were derived from the sigmoidal dose-response curve f...More data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKi: 0.200nMAssay Description:Antagonist activity at cloned muscarinic M1 receptor expressed in CHO cells assessed as acetylcholine-induced change in cytosolic calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Antagonist activity at cloned muscarinic M2 receptor-Gqi5 chimeric protein expressed in CHO cells assessed as acetylcholine-induced change in cytosol...More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Antagonist activity at oxytocin receptor in Wistar rat uterus assessed as inhibition of oxytocin-induced uterotonic activity treated 1 min prior to o...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Antagonist activity at cloned muscarinic M2 receptor-Gqi5 chimeric protein expressed in CHO cells assessed as acetylcholine-induced change in cytosol...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Antagonist activity at cloned muscarinic M1 receptor expressed in CHO cells assessed as acetylcholine-induced change in cytosolic calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as histamine-induced contractionsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonist activity at MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Antagonist activity at cloned muscarinic M3 receptor expressed in CHO cells assessed as acetylcholine-induced change in cytosolic calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Antagonist activity at cloned muscarinic M2 receptor-Gqi5 chimeric protein expressed in CHO cells assessed as acetylcholine-induced change in cytosol...More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Antagonist activity at human recombinant EP1 receptor expressed in CHO cells assessed as luciferase activity by Schild assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Antagonist activity at cloned muscarinic M3 receptor expressed in CHO cells assessed as acetylcholine-induced change in cytosolic calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Antagonist activity at cloned muscarinic M2 receptor-Gqi5 chimeric protein expressed in CHO cells assessed as acetylcholine-induced change in cytosol...More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Antagonist activity at cloned muscarinic M3 receptor expressed in CHO cells assessed as acetylcholine-induced change in cytosolic calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Antagonist activity at human recombinant CXCR3 receptor assessed as human IP10-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Antagonist activity at human histamine H4 receptor expressed in human SK-N-MC cells assessed as inhibition of 2-[3-(imidazol-4-yl)-propyl]-1-(4-iodo-...More data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Antagonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as reduction in PACAP38-induced calcium mobilization by FLIPR ...More data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Antagonist activity at cloned muscarinic M1 receptor expressed in CHO cells assessed as acetylcholine-induced change in cytosolic calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Antagonist activity at cloned muscarinic M1 receptor expressed in CHO cells assessed as acetylcholine-induced change in cytosolic calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Antagonist activity at cloned muscarinic M2 receptor-Gqi5 chimeric protein expressed in CHO cells assessed as acetylcholine-induced change in cytosol...More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Antagonist activity at histamine H3 receptor in guinea pig jejunum assessed as electrically evoked contractionsMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Antagonist activity at cloned muscarinic M1 receptor expressed in CHO cells assessed as acetylcholine-induced change in cytosolic calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Antagonist activity at oxytocin receptor in Wistar rat uterus assessed as inhibition of oxytocin-induced uterotonic activity treated 1 min prior to o...More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Antagonist activity rat recombinant histamine H3 receptor expressed in human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Antagonist activity at MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Antagonist activity rat recombinant histamine H3 receptor expressed in human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Antagonist activity at human recombinant CXCR3 receptor assessed as human IP10-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Antagonist activity at cloned muscarinic M3 receptor expressed in CHO cells assessed as acetylcholine-induced change in cytosolic calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Antagonist activity at MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 38nM ΔG°: -44.1kJ/molepH: 7.0 T: 2°CAssay Description:BRAF kinase activity was quantified using an ELISA-based MEK phosphorylation assay. IC50 values were derived from the sigmoidal dose-response curve f...More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Antagonist activity at wild type guinea pig NK3 receptor A1142.58T mutant expressed in HEK293 cells assessed as inhibition of [MePhe7]NKB-induced acc...More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Antagonist activity at human recombinant CXCR3 receptor assessed as human IP10-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Antagonist activity at rat Alpha-1D adrenoceptor assessed as inhibition if norepenephrine-induced contraction of thoracic aortaMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Antagonist activity at histamine H3 receptor in guinea pig jejunum assessed as electrically evoked contractionsMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Antagonist activity at vasopressin V1a receptor in phenoxybenzamine-treated Wistar rat uterus assessed as inhibition of vasopressin-induced arteial v...More data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Antagonist activity at histamine H3 receptor in guinea pig jejunum assessed as electrically evoked contractionsMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Antagonist activity at cloned muscarinic M1 receptor expressed in CHO cells assessed as acetylcholine-induced change in cytosolic calcium concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as histamine-induced contractionsMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as histamine-induced contractionsMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Antagonist activity at histamine H3 receptor in guinea pig jejunum assessed as electrically evoked contractionsMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Antagonist activity at histamine H3 receptor in guinea pig jejunum assessed as electrically evoked contractionsMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Antagonist activity at MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Antagonist activity at oxytocin receptor in Wistar rat uterus assessed as inhibition of oxytocin-induced uterotonic activity treated 1 min prior to o...More data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:Antagonist activity at wild type guinea pig NK3 receptor expressed in HEK293 cells assessed as inhibition of [MePhe7]NKB-induced accumulation of [3H]...More data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Antagonist activity rat recombinant histamine H3 receptor expressed in human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Antagonist activity at MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Antagonist activity at oxytocin receptor in Wistar rat uterus assessed as inhibition of oxytocin-induced uterotonic activity treated 1 min prior to o...More data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Antagonist activity at MTL receptor in rabbit duodenum homogenateMore data for this Ligand-Target Pair
