TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Inhibitory constant against amidase free Glutathionylspermidine Synthetase mutant (C79A)More data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 6.40E+3nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 6.40E+3nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 7.20E+3nMAssay Description:In vitro binding affinity for Histamine H3 receptorMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 7.20E+3nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 1.04E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 1.04E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 1.40E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 1.40E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 2.70E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 2.70E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 3.20E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 3.20E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 3.30E+4nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 3.30E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 6.00E+4nMAssay Description:Inhibition constant of the compound was evaluated against enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 8.10E+4nMAssay Description:Inhibition constant of the compound was evaluated against enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)
Curated by ChEMBL
University Of Antwerp (Uia)
Curated by ChEMBL
Affinity DataKi: 8.10E+4nMAssay Description:Concentration of the compound required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant human FGFR1 in the presence of ATP at Km concentrationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.270nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 0.290nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of FGFR1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR1 (398 to 822 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 0.437nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of FGFR2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 0.630nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR1 (398 to 822 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 0.790nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR1 (398 to 822 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 0.810nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 0.840nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 0.890nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 0.915nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 0.950nMAssay Description:The compounds were dissolved in 100% DMSO, and obtained solutions were serially diluted in reaction buffer (50 mM Tris pH 7.5, 10 mM MgCl2, 0.25 mM E...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of FGFR3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of FGFR2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.07nMAssay Description:The compounds were dissolved in 100% DMSO, and obtained solutions were serially diluted in reaction buffer (50 mM Tris pH 7.5, 10 mM MgCl2, 0.25 mM E...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged FGFR3 (436 to 806 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of FGFR1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human recombinant BACE1 by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.26nMAssay Description:The compounds were dissolved in 100% DMSO, and obtained solutions were serially diluted in reaction buffer (50 mM Tris pH 7.5, 10 mM MgCl2, 0.25 mM E...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human FGFR2 (399 to 821 residues) expressed in baculovirus expression system using IGF-1Rtide peptide...More data for this Ligand-Target Pair
Affinity DataIC50: 1.63nMAssay Description:The compounds were dissolved in 100% DMSO, and obtained solutions were serially diluted in reaction buffer (50 mM Tris pH 7.5, 10 mM MgCl2, 0.25 mM E...More data for this Ligand-Target Pair