Affinity DataKi: 6nMAssay Description:Inhibition of human CA12 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of human CA2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of human CA9 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Inhibition of human CA2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Inhibition of human CA12 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Inhibition of human CA1 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Inhibition of human CA2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Inhibition of human CA2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Inhibition of human CA2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of human CA12 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Inhibition of human CA2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Inhibition of human CA12 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Inhibition of human CA1 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Inhibition of human CA12 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 750nMAssay Description:Inhibition of human CA1 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 780nMAssay Description:Inhibition of human CA12 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Inhibition of human CA12 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 840nMAssay Description:Inhibition of human CA12 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 860nMAssay Description:Inhibition of human CA2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 960nMAssay Description:Inhibition of human CA1 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.25E+3nMAssay Description:Inhibition of human CA9 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.25E+3nMAssay Description:Inhibition of human CA9 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.26E+3nMAssay Description:Inhibition of human CA9 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.44E+3nMAssay Description:Inhibition of human CA9 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.78E+3nMAssay Description:Inhibition of human CA9 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Inhibition of human CA2 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.37E+3nMAssay Description:Inhibition of human CA1 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.43E+3nMAssay Description:Inhibition of human CA9 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.46E+3nMAssay Description:Inhibition of human CA1 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.54E+3nMAssay Description:Inhibition of human CA9 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8.02E+3nMAssay Description:Inhibition of human CA1 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 9.07E+3nMAssay Description:Inhibition of human CA1 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Dipartimento Farmaco Chimico Tecnologico
Curated by ChEMBL
Dipartimento Farmaco Chimico Tecnologico
Curated by ChEMBL
Affinity DataIC50: 4.46nMAssay Description:Inhibition of human recombinant MAOA expressed in baculovirus infected BTI insect cells assessed as hydrogen peroxide production after 15 mins by Amp...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Dipartimento Farmaco Chimico Tecnologico
Curated by ChEMBL
Dipartimento Farmaco Chimico Tecnologico
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
Affinity DataIC50: 7.60nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
Affinity DataIC50: 9.5nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
Affinity DataIC50: 19.6nMAssay Description:Inhibition of human recombinant MAOB expressed in baculovirus infected BTI insect cells assessed as hydrogen peroxide production after 15 mins by Amp...More data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
Affinity DataIC50: 82.5nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of COX1 in human platelet microsomes assessed as reduction in formation of oxidized TMPD using arachidonic acid as substrate preincubated ...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
Affinity DataIC50: 115nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
Affinity DataIC50: 115nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of human COX2 expressed in baculovirus infected sf21 cells assessed as reduction in formation of oxidized TMPD using arachidonic acid as s...More data for this Ligand-Target Pair
Affinity DataIC50: 122nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair
Affinity DataIC50: 204nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
Affinity DataIC50: 218nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
Affinity DataIC50: 221nMAssay Description:Inhibition of human recombinant MAO-B expressed in BTI-TN-5B1-4 insect cells using p-tyramine substrate by Amplex Red MAO assayMore data for this Ligand-Target Pair