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Found 164 with Last Name = 'yasumatsu' and Initial = 'i'
TargetTyrosine-protein kinase Fer(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50501949(CHEMBL4461851)
Affinity DataIC50:  0.490nMAssay Description:Inhibition of recombinant N-terminal His-tagged human FER (SH2 domain to C-terminal) expressed in Escherichia coli assessed as decrease in FL-Peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fer(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50501965(CHEMBL4457164)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of recombinant N-terminal His-tagged human FER (SH2 domain to C-terminal) expressed in Escherichia coli assessed as decrease in FL-Peptide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fer(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50501961(CHEMBL4456804)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of recombinant N-terminal His-tagged human FER (SH2 domain to C-terminal) expressed in Escherichia coli assessed as decrease in FL-Peptide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560578(CHEMBL4795328)
Affinity DataIC50:  3.30nMAssay Description:Inhibition G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560569(CHEMBL4741874)
Affinity DataIC50:  4.30nMAssay Description:Inhibition G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase Fer(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50501963(CHEMBL4524587)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of recombinant N-terminal His-tagged human FER (SH2 domain to C-terminal) expressed in Escherichia coli assessed as decrease in FL-Peptide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560575(CHEMBL4756618)
Affinity DataIC50:  6.30nMAssay Description:Inhibition G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fer(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50501959(CHEMBL4557212)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant N-terminal His-tagged human FER (SH2 domain to C-terminal) expressed in Escherichia coli assessed as decrease in FL-Peptide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560572(CHEMBL4747198)
Affinity DataIC50:  11nMAssay Description:Inhibition G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336049(CHEMBL1669334 | N-benzyl-4-(6-(cyclopropylmethylam...)
Affinity DataIC50:  12nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336052(CHEMBL1669337 | N-cinnamyl-4-(6-(cyclopropylmethyl...)
Affinity DataIC50:  13nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560576(CHEMBL4741567)
Affinity DataIC50:  14nMAssay Description:Inhibition G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fer(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50501957(CHEMBL4455220)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant N-terminal His-tagged human FER (SH2 domain to C-terminal) expressed in Escherichia coli assessed as decrease in FL-Peptide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560577(CHEMBL4783331)
Affinity DataIC50:  15nMAssay Description:Inhibition G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336057(CHEMBL1669342 | N-(4-acetamidobenzyl)-4-(6-(cyclop...)
Affinity DataIC50:  15nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336055(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  15nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560578(CHEMBL4795328)
Affinity DataIC50:  15nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560568(CHEMBL4752510)
Affinity DataIC50:  15nMAssay Description:Inhibition G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336065(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  16nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336056(4-((4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  17nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336051(CHEMBL1669336 | N-(4-chlorobenzyl)-4-(6-(cycloprop...)
Affinity DataIC50:  17nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336050(CHEMBL1669335 | N-(3-chlorobenzyl)-4-(6-(cycloprop...)
Affinity DataIC50:  17nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560561(CHEMBL4759665)
Affinity DataIC50:  17nMAssay Description:Inhibition G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336064(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  18nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336060(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  21nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336061(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  22nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336058(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  23nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fer(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50501950(CHEMBL4548027)
Affinity DataIC50:  25nMAssay Description:Inhibition of recombinant N-terminal His-tagged human FER (SH2 domain to C-terminal) expressed in Escherichia coli assessed as decrease in FL-Peptide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560575(CHEMBL4756618)
Affinity DataIC50:  27nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560571(CHEMBL4753571)
Affinity DataIC50:  28nMAssay Description:Inhibition G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fer(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50501960(CHEMBL4564799)
Affinity DataIC50:  31nMAssay Description:Inhibition of recombinant N-terminal His-tagged human FER (SH2 domain to C-terminal) expressed in Escherichia coli assessed as decrease in FL-Peptide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560569(CHEMBL4741874)
Affinity DataIC50:  32nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336063(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  42nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560577(CHEMBL4783331)
Affinity DataIC50:  43nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560572(CHEMBL4747198)
Affinity DataIC50:  44nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325416((S)-4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  47nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325375((S)-4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  55nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325375((S)-4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  55nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fer(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50501948(CHEMBL4470327)
Affinity DataIC50:  57nMAssay Description:Inhibition of recombinant N-terminal His-tagged human FER (SH2 domain to C-terminal) expressed in Escherichia coli assessed as decrease in FL-Peptide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336059(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  71nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325371(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  73nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560568(CHEMBL4752510)
Affinity DataIC50:  74nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325370(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  79nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560570(CHEMBL4747939)
Affinity DataIC50:  83nMAssay Description:Inhibition G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560563(CHEMBL4779949)
Affinity DataIC50:  93nMAssay Description:Inhibition G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336062((S)-4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  97nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325415((R)-4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  100nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50560576(CHEMBL4741567)
Affinity DataIC50:  109nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325418((S)-4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  110nMAssay Description:Inhibition of purified His-tagged IKK-beta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336054(2-(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyri...)
Affinity DataIC50:  110nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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