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Found 206 with Last Name = 'ye' and Initial = 'yp'
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147851((3R,4S)-4-(4-Chloro-phenyl)-1-methyl-3-propyl-pipe...)
Affinity DataKi:  6.5nMAssay Description:Ability to inhibit high affinity uptake of [3H]NE at Norepinephrine transporter (NET) using rat brain parietal/occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50115557(4-(4-Chloro-phenyl)-piperidine-3-carboxylic acid m...)
Affinity DataKi:  7.90nMAssay Description:Inhibition of high affinity uptake of [3H]NE by norepinephrine transporter in nerve endings obtained from rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127626(5-(3',4'-Dichloro-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  9.70nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127627(5-[5-(4-Methoxy-phenyl)-thiophen-2-ylmethylene]-3-...)
Affinity DataKi:  10.3nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127641(5-(5-Phenyl-thiophen-2-ylmethylene)-3-aza-tricyclo...)
Affinity DataKi:  13.5nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127642(5-(4-Furan-2-yl-benzylidene)-3-aza-tricyclo[4.4.2....)
Affinity DataKi:  13.9nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147854(3-[(3R,4S)-4-(4-Chloro-phenyl)-1-methyl-piperidin-...)
Affinity DataKi:  16nMAssay Description:Ability to inhibit high affinity uptake of [3H]DA at Dopamine transporter (DAT) using rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147831(2-[(3R,4S)-4-(4-Chloro-phenyl)-1-methyl-piperidin-...)
Affinity DataKi:  16nMAssay Description:Ability to inhibit high affinity uptake of [3H]DA at Dopamine transporter (DAT) using rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127644(5-(3'-Chloro-biphenyl-4-ylmethylene)-3-aza-tricycl...)
Affinity DataKi:  17.5nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127625(5-(4-Thiophen-2-yl-benzylidene)-3-aza-tricyclo[4.4...)
Affinity DataKi:  19.8nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147829((3R,4S)-3-Allyloxymethyl-4-(4-chloro-phenyl)-1-met...)
Affinity DataKi:  20nMAssay Description:Ability to inhibit high affinity uptake of [3H]NE at Norepinephrine transporter (NET) using rat brain parietal/occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147851((3R,4S)-4-(4-Chloro-phenyl)-1-methyl-3-propyl-pipe...)
Affinity DataKi:  20nMAssay Description:Ability to inhibit high affinity uptake of [3H]DA at Dopamine transporter (DAT) using rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127635(5-(4-Thiophen-3-yl-benzylidene)-3-aza-tricyclo[4.4...)
Affinity DataKi:  20.5nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127624(5-[4-(5-Methyl-thiophen-2-yl)-benzylidene]-3-aza-t...)
Affinity DataKi:  22.5nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127634(5-(4'-Methyl-biphenyl-4-ylmethylene)-3-aza-tricycl...)
Affinity DataKi:  22.7nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147840(3-[(3R,4S)-4-(4-Chloro-phenyl)-1-methyl-piperidin-...)
Affinity DataKi:  31nMAssay Description:Ability to inhibit high affinity uptake of [3H]NE at Norepinephrine transporter (NET) using rat brain parietal/occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147846((3R,4S)-3-(5-Benzo[1,3]dioxol-5-yl-[1,2,4]oxadiazo...)
Affinity DataKi:  32nMAssay Description:Ability to inhibit high affinity uptake of [3H]-5-HT at Serotonin transporter (SERT) using rat midbrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147833(CHEMBL103262 | N-Benzyl-2-[(3R,4S)-4-(4-chloro-phe...)
Affinity DataKi:  32nMAssay Description:Ability to inhibit high affinity uptake of [3H]NE at Norepinephrine transporter (NET) using rat brain parietal/occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127630(5-(4'-Cyano-biphenyl-4-ylmethylene)-3-aza-tricyclo...)
Affinity DataKi:  32.4nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147832(CHEMBL103805 | Phenyl-carbamic acid (3R,4S)-4-(4-c...)
Affinity DataKi:  33nMAssay Description:Ability to inhibit high affinity uptake of [3H]NE at Norepinephrine transporter (NET) using rat brain parietal/occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50115561(4-(4-Chloro-phenyl)-3-(3-methyl-[1,2,4]oxadiazol-5...)
Affinity DataKi:  34nMAssay Description:Inhibition of high affinity uptake of [3H]NE by norepinephrine transporter in nerve endings obtained from rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147857(CHEMBL103208 | [(3R,4S)-4-(4-Chloro-phenyl)-1-meth...)
Affinity DataKi:  36nMAssay Description:Ability to inhibit high affinity uptake of [3H]DA at Dopamine transporter (DAT) using rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147834(Adamantan-1-yl-carbamic acid (3R,4S)-4-(4-chloro-p...)
Affinity DataKi:  37nMAssay Description:Ability to inhibit high affinity uptake of [3H]-5-HT at Serotonin transporter (SERT) using rat midbrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127638(5-(4'-Methoxy-biphenyl-4-ylmethylene)-3-aza-tricyc...)
Affinity DataKi:  39nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147837((3R,4S)-4-(4-Chloro-phenyl)-3-(3-fluoro-propyl)-1-...)
Affinity DataKi:  43nMAssay Description:Ability to inhibit high affinity uptake of [3H]DA at Dopamine transporter (DAT) using rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147846((3R,4S)-3-(5-Benzo[1,3]dioxol-5-yl-[1,2,4]oxadiazo...)
Affinity DataKi:  44nMAssay Description:Ability to inhibit high affinity uptake of [3H]DA at Dopamine transporter (DAT) using rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127628(5-(4-Pyrrol-1-yl-benzylidene)-3-aza-tricyclo[4.4.2...)
Affinity DataKi:  45.9nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127632(Acetic acid 5-biphenyl-4-ylmethylene-3-aza-tricycl...)
Affinity DataKi:  46nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147831(2-[(3R,4S)-4-(4-Chloro-phenyl)-1-methyl-piperidin-...)
Affinity DataKi:  46nMAssay Description:Ability to inhibit high affinity uptake of [3H]NE at Norepinephrine transporter (NET) using rat brain parietal/occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127630(5-(4'-Cyano-biphenyl-4-ylmethylene)-3-aza-tricyclo...)
Affinity DataKi:  47nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147857(CHEMBL103208 | [(3R,4S)-4-(4-Chloro-phenyl)-1-meth...)
Affinity DataKi:  48nMAssay Description:Ability to inhibit high affinity uptake of [3H]NE at Norepinephrine transporter (NET) using rat brain parietal/occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147846((3R,4S)-3-(5-Benzo[1,3]dioxol-5-yl-[1,2,4]oxadiazo...)
Affinity DataKi:  52nMAssay Description:Ability to inhibit high affinity uptake of [3H]NE at Norepinephrine transporter (NET) using rat brain parietal/occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147830((3R,4S)-4-(4-Chloro-phenyl)-1-methyl-piperidine-3-...)
Affinity DataKi:  53nMAssay Description:Ability to inhibit high affinity uptake of [3H]DA at Dopamine transporter (DAT) using rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147843((E)-3-[(3R,4S)-4-(4-Chloro-phenyl)-1-methyl-piperi...)
Affinity DataKi:  53nMAssay Description:Ability to inhibit high affinity uptake of [3H]DA at Dopamine transporter (DAT) using rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147852(3-[(3R,4S)-4-(4-Chloro-phenyl)-1-methyl-piperidin-...)
Affinity DataKi:  56nMAssay Description:Ability to inhibit high affinity uptake of [3H]NE at Norepinephrine transporter (NET) using rat brain parietal/occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147834(Adamantan-1-yl-carbamic acid (3R,4S)-4-(4-chloro-p...)
Affinity DataKi:  56nMAssay Description:Ability to inhibit high affinity uptake of [3H]NE at Norepinephrine transporter (NET) using rat brain parietal/occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147834(Adamantan-1-yl-carbamic acid (3R,4S)-4-(4-chloro-p...)
Affinity DataKi:  56nMAssay Description:Ability to inhibit high affinity uptake of [3H]DA at Dopamine transporter (DAT) using rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127632(Acetic acid 5-biphenyl-4-ylmethylene-3-aza-tricycl...)
Affinity DataKi:  57nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127622(5-(4'-Methylamino-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  57.9nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147829((3R,4S)-3-Allyloxymethyl-4-(4-chloro-phenyl)-1-met...)
Affinity DataKi:  60nMAssay Description:Ability to inhibit high affinity uptake of [3H]DA at Dopamine transporter (DAT) using rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127643(5-(3',5'-Dichloro-biphenyl-4-ylmethylene)-3-aza-tr...)
Affinity DataKi:  61nMAssay Description:Ability to inhibit [3H]NE reuptake at norepinephrine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147833(CHEMBL103262 | N-Benzyl-2-[(3R,4S)-4-(4-chloro-phe...)
Affinity DataKi:  66nMAssay Description:Ability to inhibit high affinity uptake of [3H]-5-HT at Serotonin transporter (SERT) using rat midbrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147840(3-[(3R,4S)-4-(4-Chloro-phenyl)-1-methyl-piperidin-...)
Affinity DataKi:  68nMAssay Description:Ability to inhibit high affinity uptake of [3H]DA at Dopamine transporter (DAT) using rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50115567(CHEMBL321454 | [4-(4-Chloro-phenyl)-piperidin-3-yl...)
Affinity DataKi:  69nMAssay Description:Inhibition of high affinity uptake of [3H]NE by norepinephrine transporter in nerve endings obtained from rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127641(5-(5-Phenyl-thiophen-2-ylmethylene)-3-aza-tricyclo...)
Affinity DataKi:  71nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127625(5-(4-Thiophen-2-yl-benzylidene)-3-aza-tricyclo[4.4...)
Affinity DataKi:  73nMAssay Description:Ability to inhibit [3H]5-HT reuptake at serotonin transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147850(CHEMBL103291 | [(3R,4S)-4-(4-Chloro-phenyl)-1-meth...)
Affinity DataKi:  79nMAssay Description:Ability to inhibit high affinity uptake of [3H]DA at Dopamine transporter (DAT) using rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147857(CHEMBL103208 | [(3R,4S)-4-(4-Chloro-phenyl)-1-meth...)
Affinity DataKi:  82nMAssay Description:Ability to inhibit high affinity uptake of [3H]-5-HT at Serotonin transporter (SERT) using rat midbrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50127644(5-(3'-Chloro-biphenyl-4-ylmethylene)-3-aza-tricycl...)
Affinity DataKi:  89nMAssay Description:Ability to inhibit [3H]DA reuptake at dopamine transporter from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50147832(CHEMBL103805 | Phenyl-carbamic acid (3R,4S)-4-(4-c...)
Affinity DataKi:  91nMAssay Description:Ability to inhibit high affinity uptake of [3H]DA at Dopamine transporter (DAT) using rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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